中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 2022 [40]
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Discovery of Highly Potent Nicotinamide Phosphoribosyltransferase Degraders for Efficient Treatment of Ovarian Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 15
作者:  
Bi, Kaijian;  Cheng, Junfei;  He, Shipeng;  Fang, Yuxin;  Huang, Min
  |  收藏  |  浏览/下载:16/0  |  提交时间:2023/04/10
ASK120067 potently suppresses B-cell or T-cell malignancies in vitro and in vivo by inhibiting BTK and ITK 期刊论文  OAI收割
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13, 页码: 9
作者:  
Song, Peiran;  Bai, Gang;  Chan, Shingpan;  Zhang, Tao;  Tong, Linjiang
  |  收藏  |  浏览/下载:27/0  |  提交时间:2023/04/10
Identification of Novel Antifungal Skeleton of Hydroxyethyl Naphthalimides with Synergistic Potential for Chemical and Dynamic Treatments 期刊论文  OAI收割
MOLECULES, 2022, 卷号: 27, 期号: 23, 页码: 22
作者:  
Zhang, Pengli;  Tangadanchu, Vijai Kumar Reddy;  Zhou, Chenghe
  |  收藏  |  浏览/下载:19/0  |  提交时间:2023/04/10
Discovery of Novel N-(5-(Pyridin-3-yl)-1H-indazol-3-yl)benzamide Derivatives as Potent Cyclin-Dependent Kinase 7 Inhibitors for the Treatment of Autosomal Dominant Polycystic Kidney Disease 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 19
作者:  
Yang, Bowen;  Zhang, Haoran;  Li, Na;  Gao, Lixin;  Jiang, Hong
  |  收藏  |  浏览/下载:20/0  |  提交时间:2023/04/10
Design and exploration of gut-restricted bifunctional molecule with TGR5 agonistic and DPP4 inhibitory effects for treating ulcerative colitis 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 242, 页码: 114697
作者:  
Han, Fanghui
  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/03/21
Molecular Determinants for the High-Affinity Blockade of Human Ether-a-go-go-Related Gene K+ Channel by Tolterodine 期刊论文  OAI收割
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 2022, 卷号: 80, 期号: 5, 页码: 679-689
作者:  
Wang, Na;  Yang, Yang;  Wen, Jing;  Fan, Xin-Rong;  Li, Jian
  |  收藏  |  浏览/下载:26/0  |  提交时间:2022/12/13
Structure-based design of a novel inhibitor of the ZIKA virus NS2B/ NS3 protease 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 128, 页码: 7
作者:  
Xiong, Yanchao;  Cheng, Fei;  Zhang, Junyi;  Su, Haixia;  Hu, Hangchen
  |  收藏  |  浏览/下载:24/0  |  提交时间:2022/11/11
Discovery and characterization of a novel cGAS covalent inhibitor for the treatment of inflammatory bowel disease 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 10
作者:  
Song, Jia;  Yang, Rui-rui;  Chang, Jie;  Liu, Ya-dan;  Lu, Cheng-hao
  |  收藏  |  浏览/下载:48/0  |  提交时间:2022/11/11
Discovery of potent ebola entry inhibitors with (3S,4aS,8aS)-2-(3-amino-2-hydroxypropyl) decahydroisoquinoline-3-carboxamide scaffold 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 240, 页码: 12
作者:  
Han, Sheng;  Li, Heng;  Chen, Weixiong;  Yang, Li;  Tong, Xiankun
  |  收藏  |  浏览/下载:21/0  |  提交时间:2022/11/11
New Rufomycins from Streptomyces atratus MJM3502 Expand Anti- Mycobacterium tuberculosis Structure-Activity Relationships 期刊论文  OAI收割
ORGANIC LETTERS, 2022, 页码: 6
作者:  
Zhou, Bin;  Shetye, Gauri;  Wolf, Nina M.;  Chen, Shao-Nong;  Qader, Mallique
  |  收藏  |  浏览/下载:20/0  |  提交时间:2022/12/13