中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [13]
昆明植物研究所 [4]
宁波材料技术与工程研... [2]
青岛生物能源与过程研... [1]
海洋研究所 [1]
武汉植物园 [1]
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OAI收割 [23]
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期刊论文 [20]
学位论文 [2]
会议论文 [1]
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2022 [1]
2021 [5]
2020 [1]
2019 [2]
2018 [5]
2016 [2]
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Chemistry [1]
Materials ... [1]
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Design and exploration of gut-restricted bifunctional molecule with TGR5 agonistic and DPP4 inhibitory effects for treating ulcerative colitis
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 242, 页码: 114697
作者:
Han, Fanghui
;
Ning, Mengmeng
;
Wang, Kai
;
Gu, Yipei
;
Qu, Hui
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/03/21
Bifunctional molecule
Gut-restricted
Ulcerative colitis
TGR5
DPP4
Distal mutation V486M disrupts the catalytic activity of DPP4 by affecting the flap of the propeller domain
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:
Li, Teng-teng
;
Peng, Cheng
;
Wang, Ji-qiu
;
Xu, Zhi-jian
;
Su, Ming-bo
  |  
收藏
  |  
浏览/下载:65/0
  |  
提交时间:2022/01/18
DPP4
distal mutation
enzymatic activity
molecular dynamics simulation
structure-function mechanism
滇牡丹降血糖活性成分的比较分析和挖掘
学位论文
OAI收割
2021
作者:
黄骞
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/03/20
The Involvement of the Mammalian Target of Rapamycin, Protein Tyrosine Phosphatase 1b and Dipeptidase 4 Signaling Pathways in Cancer and Diabetes: A Narrative Review
期刊论文
OAI收割
MINI-REVIEWS IN MEDICINAL CHEMISTRY, 2021, 卷号: 21, 期号: 7, 页码: 803-815
作者:
Zhang, Jiajia
;
Wu, Ning
;
Shi, Dayong
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2021/05/11
Signaling pathway
mammalian target of rapamycin
protein tyrosine phosphatase 1b
dipeptidase 4
cancer
diabetes
pharmacology
target compounds
Diarylheptanoid-flavanone Hybrids as Multiple-target Antidiabetic Agents from Alpinia katsumadai
期刊论文
OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2021, 卷号: 39, 期号: 11, 页码: 3051-3063
作者:
He,Xiao-Feng
;
Chen,Ji-Jun
;
Li,Tian-Ze
;
Hu,Jing
;
Huang,Xiao-Yan
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2022/04/02
Alpinia katsumadai
Katsumadainols B-1-B-15
Natural products
Structure elucidation
Biological activity
TYROSINE-PHOSPHATASE 1B
GLYCOGEN-PHOSPHORYLASE
ALPHA-GLUCOSIDASE
ABSOLUTE-CONFIGURATION
STRUCTURE ELUCIDATION
DUAL INHIBITION
SEEDS
CONSTITUENT
DERIVATIVES
CHALCONE
Chemical profiling and antidiabetic potency of Paeonia delavayi: Comparison between different parts and constituents
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2021, 卷号: 198, 页码: 113998
作者:
Huang,Qian
;
Chen,Ji-Jun
;
Pan,Yang
;
He,Xiao-Feng
;
Wang,Yuan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2022/04/02
Paeonia delavayi
Chemical comparison
LCMS analyses
Antidiabetic effects
PTP1B/TCPTP selective inhibitors
LIQUID-CHROMATOGRAPHY
MULTIPLE CONSTITUENTS
RAPID IDENTIFICATION
GLYCOSIDES
ROOT
DERIVATIVES
TARGETS
CAPSULE
L.
Dipeptidyl peptidase 4 inhibitor sitagliptin protected against dextran sulfate sodium-induced experimental colitis by potentiating the action of GLP-2
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:
Ning, Meng-meng
;
Yang, Wen-ji
;
Guan, Wen-bo
;
Gu, Yi-pei
;
Feng, Ying
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/07/01
ulcerative colitis
dextran sulfate sodium
dipeptidyl peptidase 4
sitagliptin
glucagon-like peptide-2
GLP-2(3-33)
apoptosis
proliferation
芍药籽活性成分的研究
学位论文
OAI收割
: 中国科学院昆明植物研究所, 2019
作者:
张晨晨
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2022/08/29
芍药籽
二苯乙烯类化合物
降糖活性
质谱裂解途径
Alogliptin alleviates liver fibrosis via suppression of activated hepatic stellate cell
期刊论文
OAI收割
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2019, 卷号: 511, 期号: 2, 页码: 387-393
作者:
Zhang, Hanyan
;
Sun, Dandan
;
Wang, Guanzhen
;
Cui, Shichao
;
Field, Robert A.
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/07/01
DPP4
Alogliptin
Liver fibrosis
Hepatic stellate cell
A novel non-enzymatic hydrolytic probe for dipeptidyl peptidase IV specific recognition and imaging
期刊论文
OAI收割
CHEMICAL COMMUNICATIONS, 2018, 卷号: 54, 期号: 63, 页码: 8773-8776
作者:
Xing, Jie
;
Gong, Qiuyu
;
Zhang, Renshuai
;
Sun, Shan
;
Zou, Ruifen
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2018/12/21