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Chinese Academy of Sciences Institutional Repositories Grid
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The Tyrosine Kinase Inhibitor Bafetinib Inhibits PAR2-induced Activation of TRPV4 In Vitro and Pain In Vivo1 期刊论文  OAI收割
出版物, 2111, 页码: 1-44
作者:  
1M S Grace;  T Lieu;  B Darby;  F C Abogadie;  N Veldhuis N W Bunnett;  P McIntyre
  |  收藏  |  浏览/下载:220/0  |  提交时间:2017/07/24
Development of Potent MALT1 Inhibitors Featuring a Novel "2-Thioxo-2,3-dihydrothiazolo[4,5-d]pyrimidin-7(6H)-one" Scaffold for the Treatment of B Cell Lymphoma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 4, 页码: 2884-2906
作者:  
Liang, Xuewu;  Yu, Haolan;  Liang, Renwen;  Feng, Zhuanghui;  Saidahmatov, Abdusaid
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/04/09
Design, synthesis and biological evaluation of betulinic acid derivatives as potential inhibitors of 3CL-protease of SARS-CoV-2 期刊论文  OAI收割
STEROIDS, 2024, 卷号: 202, 页码: 8
作者:  
Liu, Yaowen;  Nie, Tianqing;  Hou, Jinjun;  Long, Huali;  Zhang, Zijia
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/03/13
Extracellular Matrix-Trapped Bioinspired Lipoprotein Prolongs Tumor Retention to Potentiate Antitumor Immunity 期刊论文  OAI收割
ADVANCED MATERIALS, 2024, 页码: 14
作者:  
Wu, Yao;  Li, Yongping;  Hu, Zixin;  Li, Yuan;  Zhang, Shixuan
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/02/27
A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects 期刊论文  OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:  
Yang, Xin-Mei;  Yang, Yang;  Yao, Bu-Fan;  Ye, Pan-Pan;  Xu, Yan
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/12/11
C-terminal modification and functionalization of proteins via a self-cleavage tag triggered by a small molecule 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 13
作者:  
Zeng, Yue;  Shi, Wei;  Liu, Zhi;  Xu, Hao;  Liu, Liya
  |  收藏  |  浏览/下载:6/0  |  提交时间:2024/02/19
Selective activator of human ClpP triggers cell cycle arrest to inhibit lung squamous cell carcinoma 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 7069
作者:  
Zhou, Lin-Lin;  Zhang, Tao;  Xue, Yun;  Yue, Chuan;  Pan, Yihui
  |  收藏  |  浏览/下载:3/0  |  提交时间:2024/03/27
Deubiquitylating Enzymes in Cancer and Immunity 期刊论文  OAI收割
ADVANCED SCIENCE, 2023, 页码: 37
作者:  
Ren, Jiang;  Yu, Peng;  Liu, Sijia;  Li, Ran;  Niu, Xin
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/12/08
Structure-based development and preclinical evaluation of the SARS-CoV-2 3C-like protease inhibitor simnotrelvir 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 15
作者:  
Jiang, Xiangrui;  Su, Haixia;  Shang, Weijuan;  Zhou, Feng;  Zhang, Yan
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/03/25
Assessment of the structure-activity relationship and antileukemic activity of diacylpyramide compounds as human ClpP agonists 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 258, 页码: 17
作者:  
Zhang, Ranran;  Wang, Pengyu;  Wei, Bingyan;  Chen, Liang;  Song, Xiaomin
  |  收藏  |  浏览/下载:20/0  |  提交时间:2023/10/17