中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [38]
采集方式
OAI收割 [38]
内容类型
期刊论文 [38]
发表日期
2021 [38]
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内容类型:期刊论文
发表日期:2021
专题:上海药物研究所
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Histone lysine methacrylation is a dynamic post-translational modification regulated by HAT1 and SIRT2
期刊论文
OAI收割
CELL DISCOVERY, 2021, 卷号: 7, 期号: 1, 页码: 14
作者:
Delaney, Kyle
;
Tan, Minjia
;
Zhu, Zhesi
;
Gao, Jinjun
;
Dai, Lunzhi
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/06/15
Structures of the human cholecystokinin receptors bound to agonists and antagonists
期刊论文
OAI收割
NATURE CHEMICAL BIOLOGY, 2021, 卷号: 17, 期号: 12, 页码: 1230-1237
作者:
Zhang, Xuefeng
;
He, Chenglin
;
Wang, Mu
;
Zhou, Qingtong
;
Yang, Dehua
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/03/21
Structure-Based Design of Dual-Acting Compounds Targeting Adenosine A(2A) Receptor and Histone Deacetylase as Novel Tumor Immunotherapeutic Agents
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 22, 页码: 16573-16597
作者:
Yan, Wenzhong
;
Ling, Lijun
;
Wu, Yiran
;
Yang, Kexin
;
Liu, Ruiquan
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2022/06/15
Genetically-engineered "all-in-one" vaccine platform for cancer immunotherapy
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 11, 页码: 3622-3635
作者:
Wu, Aihua
;
Chen, Yingzhi
;
Wang, Hairui
;
Chang, Ya
;
Zhang, Meng
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2022/01/18
Trichosanthin
Legumain
TRP2
Transcutaneous immunization
Adjuvant
Cancer vaccine
Protein engineering
Synthesis and bioactivity studies of covalent inhibitors derived from (-)-Chaetominine
期刊论文
OAI收割
JOURNAL OF MOLECULAR STRUCTURE, 2021, 卷号: 1241, 页码: 14
作者:
Zhou, Xian
;
Feng, Xuexin
;
Wang, Dachi
;
Chen, Deheng
;
Wu, Gaoxing
  |  
收藏
  |  
浏览/下载:88/0
  |  
提交时间:2021/08/17
Chaetominine
Cellular growth inhibition
Cancer cell line
Covalent warhead
DRAK2 aggravates nonalcoholic fatty liver disease progression through SRSF6-associated RNA alternative splicing
期刊论文
OAI收割
CELL METABOLISM, 2021, 卷号: 33, 期号: 10, 页码: 2004-+
作者:
Li, Yufeng
;
Xu, Junyu
;
Lu, Yuting
;
Bian, Hua
;
Yang, Lin
  |  
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2022/01/18
Constitutive signal bias mediated by the human GHRHR splice variant 1
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 40, 页码: 10
作者:
Cong, Zhaotong
;
Zhou, Fulai
;
Zhang, Chao
;
Zou, Xinyu
;
Zhang, Huibing
  |  
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2021/12/01
class B1 GPCR
receptor bias
cancer
cell proliferation
PARP14 inhibits microglial activation via LPAR5 to promote post-stroke functional recovery
期刊论文
OAI收割
AUTOPHAGY, 2021, 卷号: 17, 期号: 10, 页码: 2905-2922
作者:
Tang, Ying
;
Liu, Jinchang
;
Wang, Yu
;
Yang, Li
;
Han, Bing
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2022/01/04
Autophagy
functional recovery
ischemic stroke
lysophosphatidic acid receptor 5
microglial activation
poly (ADP-ribose) polymerase 14
Insights into agonist-elicited activation of the human glucose-dependent insulinotropic polypeptide receptor
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2021, 卷号: 192, 页码: 16
作者:
Yuliantie, Elita
;
van der Velden, Wijnand J. C.
;
Labroska, Viktorija
;
Dai, Antao
;
Zhao, Fenghui
  |  
收藏
  |  
浏览/下载:94/0
  |  
提交时间:2021/11/04
Glucose-dependent insulinotropic polypeptide receptor
G protein-coupled receptor
GPCR structure-function relationship
ERK
cAMP
Arrestin
Ligand recognition and G-protein coupling selectivity of cholecystokinin A receptor
期刊论文
OAI收割
NATURE CHEMICAL BIOLOGY, 2021, 卷号: 17, 期号: 12, 页码: 1238-1244
作者:
Liu, Qiufeng
;
Yang, Dehua
;
Zhuang, Youwen
;
Croll, Tristan I.
;
Cai, Xiaoqing
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/03/22
a Receptor
Structural Basis
Binding-site
Cck1 Receptor
Agonist
Activation
Mechanism
Optimization
Discovery
Rat