中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [17]
采集方式
OAI收割 [17]
内容类型
期刊论文 [17]
发表日期
2019 [17]
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浏览/检索结果:
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发表日期:2019
专题:上海药物研究所
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Discovery and biological evaluation of vinylsulfonamide derivatives as highly potent, covalent TEAD autopalmitoylation inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 184, 页码: 15
作者:
Lu, Wenchao
;
Wang, Jun
;
Li, Yong
;
Tao, Hongru
;
Xiong, Huan
  |  
收藏
  |  
浏览/下载:81/0
  |  
提交时间:2020/07/01
Hippo pathway
TEAD transcription factor
Covalent inhibitor
Palmitoylation inhibitor
Simultaneous determination of alflutinib and its active metabolite in human plasma using liquid chromatography-tandem mass spectrometry
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2019, 卷号: 176, 页码: 6
作者:
Liu, Xiaoyun
;
Li, Wei
;
Zhang, Yifan
;
Jian, Yong
;
Zhao, Qianyu
  |  
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2020/07/01
LC-MS/MS
Alflutinib
AST2818
Pharmacokinetics
Human plasma
A New Sesquiterpenoid from Chrysanthemum indicum
期刊论文
OAI收割
CHEMISTRY OF NATURAL COMPOUNDS, 2019, 页码: 4
作者:
Chen, Jia
;
Yang, Xu
;
Li, Bo
;
Yang, Kun
;
Wang, Yiqin
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2020/07/01
Chrysanthemum indicum
sesquiterpenoid
glucoside
nitric oxide production
Recent progress in drug delivery
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2019, 卷号: 9, 期号: 6, 页码: 1145-1162
作者:
Li, Chong
;
Wang, Jiancheng
;
Wang, Yiguang
;
Gao, Huile
;
Wei, Gang
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2020/07/01
Pharmaceutics
Drug delivery system
Basic research
Application
Delivery strategy
Organo-Catalyzed Asymmetric Amination of 4-Arylisoquinoline-1,3(2H,4H)-dione Derivatives in the Construction of Quaternary Stereocenters
期刊论文
OAI收割
ADVANCED SYNTHESIS & CATALYSIS, 2019, 页码: 6
作者:
Cheng, Cheng
;
Li, Ying-Xian
;
Zhang, Ji-Quan
;
Zhao, Yong-Long
;
Zhang, Lin
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2020/07/01
Isoquinoline-1,3(2H,4H)-dione
Amination reaction
Asymmetric catalysis
Bifunctional catalyst
Canescones A-E: aromatic polyketide dimers with PTP1B inhibitory activity from Penicillium canescens
期刊论文
OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 18, 页码: 3274-3281
作者:
Zang, Yi
;
Gong, Yi-Hua
;
Li, Xu-Wen
;
Li, Xiao-Nian
;
Liu, Jun-Jun
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2020/07/01
Small molecule IVQ, as a prodrug of gluconeogenesis inhibitor QVO, efficiently ameliorates glucose homeostasis in type 2 diabetic mice
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2019, 卷号: 40, 期号: 9, 页码: 1193-1204
作者:
Zhou, Ting-ting
;
Zhao, Tong
;
Ma, Fei
;
Zhang, Yi-nan
;
Jiang, Jing
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/07/01
type 2 diabetes mellitus
hepatic gluconeogenesis
AMPK signaling pathway
(E)-3-(2-(quinoline-4-yl)vinyl)-1H-indol-6-ol (QVO)
4-[2-(1H-indol-3-yl)vinyl]quinoline (IVQ)
prodrug
Metal-free quinolylation of the primary amino groups of amino acid derivatives and peptides with dihydrooxazolo[3,2-a]quinoliniums
期刊论文
OAI收割
GREEN CHEMISTRY, 2019, 卷号: 21, 期号: 15, 页码: 4231-4237
作者:
Liu, Peng
;
Li, Bo
;
Xi, Mengyu
;
Chen, Zhaoqiang
;
Sun, Haiguo
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/07/01
Crystal Transformation of -CD-MOF Facilitates Loading of Dimercaptosuccinic Acid
期刊论文
OAI收割
AAPS PHARMSCITECH, 2019, 卷号: 20, 期号: 6, 页码: 9
作者:
Xiong, Yuehuai
;
Wu, Li
;
Guo, Tao
;
Wang, Caifen
;
Wu, Wenting
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2020/07/01
beta-cyclodextrin metal-organic frameworks
crystal transformation
drug loading
dimercaptosuccinic acid
Chain-Length- and Saturation-Tuned Mechanics of Fluid Nanovesicles Direct Tumor Delivery
期刊论文
OAI收割
ACS NANO, 2019, 卷号: 13, 期号: 7, 页码: 7676-7689
作者:
Dai, Zhuo
;
Yu, Miaorong
;
Yi, Xin
;
Wu, Zeming
;
Tian, Falin
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2020/07/01
SUVs
liposome
chain length and saturation
membrane mechanics
vesicle rigidity
ECM penetration
tumor delivery