中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [102]
采集方式
OAI收割 [102]
内容类型
期刊论文 [102]
发表日期
2024 [2]
2023 [6]
2022 [5]
2021 [10]
2020 [8]
2019 [6]
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Biochemist... [1]
Biophysics [1]
Cell Biolo... [1]
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共102条,第1-10条
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专题:上海药物研究所
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A novel strategy for treating oncogene-mutated tumors by targeting tumor microenvironment and synergistically enhancing anti-PD-1 immunotherapy
期刊论文
OAI收割
CANCER COMMUNICATIONS, 2024, 页码: 5
作者:
Liu, Yingqiang
;
Tong, Linjiang
;
Zhang, Mengge
;
Zhang, Qi
;
Liu, Qiupei
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/03/13
Pharmacologically significant constituents collectively responsible for anti-sepsis action of XueBiJing, a Chinese herb-based intravenous formulation
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 16
作者:
Cheng, Chen
;
Ren, Chao
;
Li, Mu-zi
;
Liu, Yi-hui
;
Yao, Ren-qi
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/02/27
Traditional Chinese medicine
XueBiJing
sepsis
mortality
pharmacokinetic compatibility
polypharmacology
The novel norcantharidin derivative DCZ5417 suppresses multiple myeloma progression by targeting the TRIP13-MAPK-YWHAE signaling pathway
期刊论文
OAI收割
JOURNAL OF TRANSLATIONAL MEDICINE, 2023, 卷号: 21, 期号: 1, 页码: 17
作者:
Wang, Yingcong
;
Dong, Sanfeng
;
Hu, Ke
;
Xu, Li
;
Feng, Qilin
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/01/26
Norcantharidin
Derivative
DCZ5417
TRIP13
Anti-myeloma
MAPK
Design, synthesis and biological evaluation of chalcone derivatives as potent and orally active hCYP3A4 inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 95, 页码: 9
作者:
Lu, Shiwei
;
Zhang, Feng
;
Gong, Jiahao
;
Huang, Jian
;
Zhu, Guanghao
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/12/08
Cytochrome P450 3A4 (CYP3A4)
Inhibitors
Isoquinoline chalcones
Orally active
Anxiolytic effect of antidiabetic metformin is mediated by AMPK activation in mPFC inhibitory neurons
期刊论文
OAI收割
MOLECULAR PSYCHIATRY, 2023, 页码: 11
作者:
Zhang, Yong-mei
;
Zong, Hai-chao
;
Qi, Ying-bei
;
Chang, Liu-liu
;
Gao, Ya-nan
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/12/08
Discovery and Structural Optimization of Covalent ZAP-70 Kinase Inhibitors against Psoriasis
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 15
作者:
Rao, Danni
;
Yang, Tao
;
Feng, Huixu
;
An, Qi
;
Zhang, Shaofeng
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/10/17
Investigation of targets and anticancer mechanisms of covalently acting natural products by functional proteomics
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 卷号: 44, 期号: 8, 页码: 1701-1711
作者:
Zhao, Wen-si
;
Chen, Kai-feng
;
Liu, Man
;
Jia, Xing-long
;
Huang, Yu-qi
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/03/27
natural products
proteomics
ABPP
eriocalyxin B
parthenolide
Intranasal delivery of replicating mRNA encoding hACE2-targeting antibody against SARS-CoV-2 Omicron infection in the hamster
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2023, 卷号: 209, 页码: 9
作者:
Zhang, Ya-Nan
;
Zhang, Hong-Qing
;
Wang, Gui-Feng
;
Zhang, Zhe-Rui
;
Li, Jia-Qi
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/04/10
Omicron
VEEV VRP
Replicable mRNA
Energy sensor AMPK gamma regulates translation via phosphatase PPP6C independent of AMPK alpha
期刊论文
OAI收割
MOLECULAR CELL, 2022, 卷号: 82, 期号: 24, 页码: 4700-+
作者:
Zhou, Qi
;
Hao, Bingbing
;
Cao, Xiaolei
;
Gao, Lin
;
Yu, Zhenyue
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/04/10
Discovery of CECR2 Bromodomain Inhibitors with High Selectivities over BPTF Bromodomain
期刊论文
OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2022, 页码: 2072-2080
作者:
Lu, Haibo
;
Zu, Shijia
;
Duan, Zhe
;
Feng, Yueyao
;
Wang, Jie
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/08/16
CECR2 bromodomain
BPTF bromodomain
Inhibitors
Structure-activity relationships
chemical probe