中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [81]
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A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects 期刊论文  OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:  
Yang, Xin-Mei;  Yang, Yang;  Yao, Bu-Fan;  Ye, Pan-Pan;  Xu, Yan
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/12/11
Five undescribed abietane-type diterpenes of Callicarpa macrophylla 期刊论文  OAI收割
FITOTERAPIA, 2023, 卷号: 170, 页码: 10
作者:  
Du, Gao-Xiang;  Chen, Tong;  Wang, Ge;  Liu, Ying-Bo;  Zheng, Liu
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/10/17
Diterpenoids from Euphorbia lactea and their anti-HIV-1 activity 期刊论文  OAI收割
PHYTOCHEMISTRY, 2023, 卷号: 213, 页码: 11
作者:  
Zhao, Ye;  Hua, Chen;  Sha, Yi-ou;  Wu, Pei-Qian;  Liu, Qun-Fang
  |  收藏  |  浏览/下载:15/0  |  提交时间:2023/10/17
Novel thieno[2,3-b]quinoline-procaine hybrid molecules: A new class of allosteric SHP-1 activators evolved from PTP1B inhibitors 期刊论文  OAI收割
CHINESE CHEMICAL LETTERS, 2023, 卷号: 34, 期号: 8, 页码: 6
作者:  
Xu, Lei;  Xuyan, Xuyang;  Minmi, Minmin;  Wang, Zhiji;  Shee, Chao
  |  收藏  |  浏览/下载:27/0  |  提交时间:2023/10/17
Selective Electrochemical Benzylic C(sp(3))-H Oxidations in Fluoroalcohols 期刊论文  OAI收割
CHEMISTRYSELECT, 2023, 卷号: 8, 期号: 27, 页码: 4
作者:  
Shen, Haiwei;  Yang, Bo;  Lin, Jiusheng;  Zheng, Mingyue;  Jiang, Hualiang
  |  收藏  |  浏览/下载:18/0  |  提交时间:2023/10/17
Comparative Characterization of the Ginsenosides from Six Panax Herbal Extracts and Their In Vitro Rat Gut Microbial Metabolites by Advanced Liquid Chromatography-Mass Spectrometry Approaches 期刊论文  OAI收割
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2023, 卷号: 71, 期号: 24, 页码: 9391-9403
作者:  
Mi, Yue-Guang;  Xu, Xiao-Yan;  Hong, Li-Li;  Jiang, Mei-Ting;  Chen, Bo-Xue
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/10/17
Discovery of novel non-peptidic and non-covalent small-molecule 3CL(pro) inhibitors as potential candidate for COVID-19 treatment 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 4
作者:  
Jiang, Zhidong;  Feng, Bo;  Zhang, Yumin;  Nie, Tianqing;  Liu, Hong
  |  收藏  |  浏览/下载:9/0  |  提交时间:2023/10/17
Synthesis, cytotoxicity, and pharmacokinetic evaluations of niclosamide analogs for anti-SARS-CoV-2 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 253, 页码: 11
作者:  
Li, Rui;  Zhang, Zherui;  Huang, Shuhong;  Peng, Ke;  Jiang, Hualiang
  |  收藏  |  浏览/下载:8/0  |  提交时间:2023/10/17
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors 期刊论文  OAI收割
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1, 页码: 17-27
作者:  
Zang, Yi;  Su, Mingbo;  Wang, Qingxing;  Cheng, Xi;  Zhang, Wenru
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/03/27
Structure-Based Design of Tropane Derivatives as a Novel Series of CCR5 Antagonists with Broad-Spectrum Anti-HIV-1 Activities and Improved Oral Bioavailability 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 24, 页码: 16526-16540
作者:  
Xie, Xiong;  Zheng, Yu-Gui;  Chen, Huan;  Li, Jian
  |  收藏  |  浏览/下载:26/0  |  提交时间:2023/04/10