中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [12]
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Structure-based optimization of indoline-containing compounds as second generation inhibitors of NF-KB-inducing kinase (NIK) 期刊论文  OAI收割
JOURNAL OF MOLECULAR STRUCTURE, 2024, 卷号: 1295, 页码: 19
作者:  
Cheng, Jing;  Yan, Ziqin;  Li, Xinzhi;  Liu, Chen;  Tong, Linjiang
  |  收藏  |  浏览/下载:8/0  |  提交时间:2023/12/08
Selective degradation of cellular BRD3 and BRD4-L promoted by PROTAC molecules in six cancer cell lines 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 254, 页码: 17
作者:  
Yan, Ziqin;  Lyu, Xilin;  Lin, Dongze;  Wu, Gaoxing;  Gong, Yang
  |  收藏  |  浏览/下载:25/0  |  提交时间:2023/10/17
Cryo-EM structure of the human chemerin receptor 1-Gi protein complex bound to the C-terminal nonapeptide of chemerin 期刊论文  OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2023, 卷号: 120, 期号: 11, 页码: 8
作者:  
Wang, Junlin;  Chen, Geng;  Liao, Qiwen;  Lyu, Wenping;  Liu, Aijun
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/04/09
Discovery of a selective and covalent small-molecule inhibitor of BFL-1 protein that induces robust apoptosis in cancer cells 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 236, 页码: 114327
作者:  
Feng, Xuexin;  Yan, Ziqin;  Zhou, Feilong;  Lou, Jianfeng;  Lyu, Xilin
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/03/21
Structure-Based Discovery of MDM2/4 Dual Inhibitors that Exert Antitumor Activities against MDM4-Overexpressing Cancer Cells 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 8, 页码: 6207-6230
作者:  
Zhang, Shiyan;  Yan, Ziqin;  Li, Yafang;  Gong, Yang;  Lyu, Xilin
  |  收藏  |  浏览/下载:21/0  |  提交时间:2022/08/16
Synthesis and bioactivity studies of covalent inhibitors derived from (-)-Chaetominine 期刊论文  OAI收割
JOURNAL OF MOLECULAR STRUCTURE, 2021, 卷号: 1241, 页码: 14
作者:  
Zhou, Xian;  Feng, Xuexin;  Wang, Dachi;  Chen, Deheng;  Wu, Gaoxing
  |  收藏  |  浏览/下载:88/0  |  提交时间:2021/08/17
Deleterious mutation V369M in the mouse GCGR gene causes abnormal plasma amino acid levels indicative of a possible liver & ndash;alpha-cell axis 期刊论文  OAI收割
BIOSCIENCE REPORTS, 2021, 卷号: 41, 期号: 6, 页码: 12
作者:  
Liu, Qiaofeng;  Lin, Guangyao;  Chen, Yan;  Feng, Wenbo;  Xu, Yingna
  |  收藏  |  浏览/下载:37/0  |  提交时间:2021/11/24
Current trends in drug metabolism and pharmacokinetics 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2019, 卷号: 9, 期号: 6, 页码: 1113-1144
作者:  
Li, Yuhua;  Meng, Qiang;  Yang, Mengbi;  Liu, Dongyang;  Hou, Xiangyu
  |  收藏  |  浏览/下载:34/0  |  提交时间:2020/07/01
Palladium-catalyzed carbonylative Sonogashira cross-coupling for the synthesis of alkynones with formic acid as the CO source 期刊论文  OAI收割
MONATSHEFTE FUR CHEMIE, 2019, 卷号: 150, 期号: 2, 页码: 309-315
作者:  
Lyu, Xue;  Sun, Guanglong;  Zhou, Yang;  Wang, Yingying;  Lei, Min
  |  收藏  |  浏览/下载:27/0  |  提交时间:2020/07/01
currenttrendsindrugmetabolismandpharmacokinetics 期刊论文  OAI收割
actapharmaceuticasinicab, 2019, 卷号: 9, 期号: 6, 页码: 1113
作者:  
Liu Dongyang;  Hou Xiangyu;  Tang Lan;  Wang Xin;  Lyu Yuanfeng
  |  收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01