中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [47]
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A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects 期刊论文  OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:  
Yang, Xin-Mei;  Yang, Yang;  Yao, Bu-Fan;  Ye, Pan-Pan;  Xu, Yan
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/12/11
Discovery, SAR Study of GST Inhibitors from a Novel Quinazolin-4(1H)-one Focused DNA-Encoded Library 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 15
作者:  
Wen, Xin;  Zhang, Minmin;  Duan, Zhiqiang;  Suo, Yanrui;  Lu, Weiwei
  |  收藏  |  浏览/下载:30/0  |  提交时间:2023/10/17
Controlled sequential in situ self-assembly and disassembly of a fluorogenic cisplatin prodrug for cancer theranostics 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 1
作者:  
Xidan Wen;  Rui Zhang;  Yuxuan Hu;  Luyan Wu;  He Bai
  |  收藏  |  浏览/下载:14/0  |  提交时间:2023/05/22
Intranasal delivery of replicating mRNA encoding hACE2-targeting antibody against SARS-CoV-2 Omicron infection in the hamster 期刊论文  OAI收割
ANTIVIRAL RESEARCH, 2023, 卷号: 209, 页码: 9
作者:  
Zhang, Ya-Nan;  Zhang, Hong-Qing;  Wang, Gui-Feng;  Zhang, Zhe-Rui;  Li, Jia-Qi
  |  收藏  |  浏览/下载:18/0  |  提交时间:2023/04/10
Identification and evaluation of a lipid-lowering small compound in preclinical models and in a Phase I trial 期刊论文  OAI收割
CELL METABOLISM, 2022, 卷号: 34, 期号: 5, 页码: 667-+
作者:  
Wang, Jiang;  Zhao, Jing;  Yan, Cong;  Xi, Cong;  Wu, Chenglin
  |  收藏  |  浏览/下载:28/0  |  提交时间:2022/08/16
RBD conjugate vaccine with a built-in TLR1/2 agonist is highly immunogenic against SARS-CoV-2 and variants of concern 期刊论文  OAI收割
CHEMICAL COMMUNICATIONS, 2022, 卷号: 58, 期号: 13, 页码: 2120-2123
作者:  
Zhou, Shi-Hao;  Zhang, Ru-Yan;  Zhang, Hai-Wei;  Liu, Yan-Ling;  Wen, Yu
  |  收藏  |  浏览/下载:24/0  |  提交时间:2022/06/15
Computational and Structure-Based Development of High Potent Cell-Active Covalent Inhibitor Targeting the Peptidyl-Prolyl Isomerase NIMA-Interacting-1 (Pin1) 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 3, 页码: 2174-2190
作者:  
Liu, Liping;  Zhu, Rui;  Li, Jiacheng;  Pei, Yuan;  Wang, Shuangshuang
  |  收藏  |  浏览/下载:27/0  |  提交时间:2022/08/16
Self-Adjuvanting Lipoprotein Conjugate alpha GalCer-RBD Induces Potent Immunity against SARS-CoV-2 and its Variants of Concern 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 3, 页码: 2558-2570
作者:  
Wang, Jian;  Wen, Yu;  Zhou, Shi-Hao;  Zhang, Hai-Wei;  Peng, Xiao-Qian
  |  收藏  |  浏览/下载:30/0  |  提交时间:2022/08/16
Dehydroberberine Analogue Nanoassemblies for Inducing and Self-Reporting Mitochondrial Dysfunction in Tumor Cells 期刊论文  OAI收割
ACS applied bio materials, 2021, 卷号: 4, 期号: 3, 页码: 2033-2043
作者:  
Zhang, Rui;  An, Ruibing;  Gu, Zhanni;  Sun, Haifeng;  Ye, Deju
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/03/15
Design, synthesis, and biological evaluation of tetrahydroisoquinolines derivatives as novel, selective PDE4 inhibitors for antipsoriasis treatment 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 211, 页码: 20
作者:  
Zhang, Rui;  Li, Heng;  Zhang, Xianglei;  Li, Jian;  Su, Haixia
  |  收藏  |  浏览/下载:31/0  |  提交时间:2021/05/24