中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [47]
采集方式
OAI收割 [47]
内容类型
期刊论文 [47]
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2023 [4]
2022 [4]
2021 [2]
2020 [5]
2019 [5]
2018 [5]
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专题:上海药物研究所
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A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:
Yang, Xin-Mei
;
Yang, Yang
;
Yao, Bu-Fan
;
Ye, Pan-Pan
;
Xu, Yan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/11
COVID-19
Simnotrelvir
Safety
Pharmacokinetics
Healthy subjects
Discovery, SAR Study of GST Inhibitors from a Novel Quinazolin-4(1H)-one Focused DNA-Encoded Library
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 15
作者:
Wen, Xin
;
Zhang, Minmin
;
Duan, Zhiqiang
;
Suo, Yanrui
;
Lu, Weiwei
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2023/10/17
Controlled sequential in situ self-assembly and disassembly of a fluorogenic cisplatin prodrug for cancer theranostics
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 1
作者:
Xidan Wen
;
Rui Zhang
;
Yuxuan Hu
;
Luyan Wu
;
He Bai
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/05/22
Intranasal delivery of replicating mRNA encoding hACE2-targeting antibody against SARS-CoV-2 Omicron infection in the hamster
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2023, 卷号: 209, 页码: 9
作者:
Zhang, Ya-Nan
;
Zhang, Hong-Qing
;
Wang, Gui-Feng
;
Zhang, Zhe-Rui
;
Li, Jia-Qi
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/04/10
Omicron
VEEV VRP
Replicable mRNA
Identification and evaluation of a lipid-lowering small compound in preclinical models and in a Phase I trial
期刊论文
OAI收割
CELL METABOLISM, 2022, 卷号: 34, 期号: 5, 页码: 667-+
作者:
Wang, Jiang
;
Zhao, Jing
;
Yan, Cong
;
Xi, Cong
;
Wu, Chenglin
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/08/16
RBD conjugate vaccine with a built-in TLR1/2 agonist is highly immunogenic against SARS-CoV-2 and variants of concern
期刊论文
OAI收割
CHEMICAL COMMUNICATIONS, 2022, 卷号: 58, 期号: 13, 页码: 2120-2123
作者:
Zhou, Shi-Hao
;
Zhang, Ru-Yan
;
Zhang, Hai-Wei
;
Liu, Yan-Ling
;
Wen, Yu
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/06/15
Computational and Structure-Based Development of High Potent Cell-Active Covalent Inhibitor Targeting the Peptidyl-Prolyl Isomerase NIMA-Interacting-1 (Pin1)
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 3, 页码: 2174-2190
作者:
Liu, Liping
;
Zhu, Rui
;
Li, Jiacheng
;
Pei, Yuan
;
Wang, Shuangshuang
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/08/16
Self-Adjuvanting Lipoprotein Conjugate alpha GalCer-RBD Induces Potent Immunity against SARS-CoV-2 and its Variants of Concern
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 3, 页码: 2558-2570
作者:
Wang, Jian
;
Wen, Yu
;
Zhou, Shi-Hao
;
Zhang, Hai-Wei
;
Peng, Xiao-Qian
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/08/16
Dehydroberberine Analogue Nanoassemblies for Inducing and Self-Reporting Mitochondrial Dysfunction in Tumor Cells
期刊论文
OAI收割
ACS applied bio materials, 2021, 卷号: 4, 期号: 3, 页码: 2033-2043
作者:
Zhang, Rui
;
An, Ruibing
;
Gu, Zhanni
;
Sun, Haifeng
;
Ye, Deju
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/03/15
dehydroberberine
fluorescence
mitochondria
self-assembly
self-reporting
Design, synthesis, and biological evaluation of tetrahydroisoquinolines derivatives as novel, selective PDE4 inhibitors for antipsoriasis treatment
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 211, 页码: 20
作者:
Zhang, Rui
;
Li, Heng
;
Zhang, Xianglei
;
Li, Jian
;
Su, Haixia
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/05/24
PDE4 inhibitors
Tetrahydroisoquinoline
Antipsoriasis