中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共44条,第1-10条 帮助

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Tumor-targeted PROTAC prodrug nanoplatform enables precise protein degradation and combination cancer therapy 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 12
作者:  
Zou, Zhi-feng;  Yang, Lei;  Nie, Hui-jun;  Gao, Jing;  Lei, Shu-min
  |  收藏  |  浏览/下载:0/0  |  提交时间:2024/05/22
Discovery of potent PROTAC degraders of Pin1 for the treatment of acute myeloid leukemia 期刊论文  OAI收割
CHEMICAL SCIENCE, 2024, 卷号: 15, 期号: 13, 页码: 5027-5035
作者:  
Shi, Yunkai;  Liu, Minmin;  Li, Mengna;  Mao, Yiwen;  Ma, Jingkun
  |  收藏  |  浏览/下载:5/0  |  提交时间:2024/05/07
Uncovering PROTAC Sensitivity and Efficacy by Multidimensional Proteome Profiling: A Case for STAT3 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 6, 页码: 4804-4818
作者:  
Suo, Yuying;  Du, Daohai;  Chen, Chao;  Zhu, Hongwen;  Wang, Xiongjun
  |  收藏  |  浏览/下载:3/0  |  提交时间:2024/05/07
PROTAC Prodrug-Integrated Nanosensitizer for Potentiating Radiation Therapy of Cancer 期刊论文  OAI收割
ADVANCED MATERIALS, 2024, 页码: 12
作者:  
Zhang, Shunan;  Lai, Yi;  Pan, Jiaxing;  Saeed, Madiha;  Li, Shiqin
  |  收藏  |  浏览/下载:17/0  |  提交时间:2024/04/09
Discovery of Novel PROTAC Degraders of p300/CBP as Potential Therapeutics for Hepatocellular Carcinoma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 4, 页码: 2466-2486
作者:  
Chang, Qi;  Li, Jiayi;  Deng, Yue;  Zhou, Ruilin;  Wang, Bingwei
  |  收藏  |  浏览/下载:18/0  |  提交时间:2024/03/25
Discovery of a PROTAC degrader for METTL3-METTL14 complex 期刊论文  OAI收割
CELL CHEMICAL BIOLOGY, 2024, 卷号: 31, 期号: 1, 页码: 25
作者:  
Du, Wenhao;  Huang, Yuting;  Chen, Xiaoai;  Deng, Yue;  Sun, Yaoliang
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/07
Design, Synthesis, and Biological Evaluation of Potent and Selective PROTAC Degraders of Oncogenic KRASG12D 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1147-1167
作者:  
Zhou, Chuan;  Fan, Zisheng;  Gu, Yuejiao;  Ge, Zhiming;  Tao, Zhaofan
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/02/27
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:  
Zhang, Jingyu;  Duan, Haiting;  Gui, Renzhao;  Wu, Mingfei;  Shen, Liteng
  |  收藏  |  浏览/下载:12/0  |  提交时间:2023/12/19
The new direction of drug development: Degradation of undruggable targets through targeting chimera technology 期刊论文  OAI收割
MEDICINAL RESEARCH REVIEWS, 2023, 页码: 54
作者:  
Liang, Xuewu;  Ren, Hairu;  Han, Fengyang;  Liang, Renwen;  Zhao, Jiayan
  |  收藏  |  浏览/下载:25/0  |  提交时间:2024/01/16
HDAC3 and HDAC8 PROTAC dual degrader reveals roles of histone acetylation in gene regulation 期刊论文  OAI收割
CELL CHEMICAL BIOLOGY, 2023, 卷号: 30, 期号: 11, 页码: 1421-+
作者:  
  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/01/16