中国科学院机构知识库网格系统: 检索

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	Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia 期刊论文 OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18 作者: Zhang, Jingyu; Duan, Haiting; Gui, Renzhao; Wu, Mingfei; Shen, Liteng \| 收藏 \| 浏览/下载：11/0 \| 提交时间：2023/12/19 Acute myeloid leukemia Bromodomain-containing protein 9 Proteolysis-targeting chimera Orally bioavailable Docking
	Identification of small molecule inhibitors targeting the SMARCA2 bromodomain from a high-throughput screening assay 期刊论文 OAI收割 ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 9, 页码: 1544-1552 作者: Lu, Tian; Hu, Jun-chi; Lu, Wen-chao; Han, Jie; Ding, Hong \| 收藏 \| 浏览/下载：33/0 \| 提交时间：2019/01/08 AlphaScreen high-throughput screening SMARCA2 bromodomain small molecule inhibitor
	Structure-Based Discovery of CF53 as a Potent and Orally Bioavailable Bromodomain and Extra-Terminal (BET) Bromodomain Inhibitor 期刊论文 OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 14, 页码: 6110-6120 作者: Zhao, Yujun; Zhou, Bing; Bai, Longchuan; Liu, Liu; Yang, Chao-Yie \| 收藏 \| 浏览/下载：49/0 \| 提交时间：2019/01/08
	Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups 期刊论文 OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 页码: 156-175 作者: Hu, Jianping; Wang, Yingqing; Li, Yanlian; Cao, Danyan; Xu, Lin \| 收藏 \| 浏览/下载：34/0 \| 提交时间：2019/01/08 BRD4 BI2536 Indoline WPF binders c-Myc PD-L1
	Y08060: A Selective BET Inhibitor for Treatment of Prostate Cancer 期刊论文 OAI收割 ACS MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 9, 期号: 3, 页码: 262-267 作者: Xiang, Quping; Zhang, Yan; Li, Jiaguo; Xue, Xiaoqian; Wang, Chao \| 收藏 \| 浏览/下载：42/0 \| 提交时间：2019/06/20 Bromodomain Brd4 Prostate Cancer Epigenetics
	Nmr-based platform for fragment-based lead discovery used in screening brd4-targeted compounds 期刊论文 iSwitch采集 Acta pharmacologica sinica, 2016, 卷号: 37, 期号: 7, 页码: 984-993 作者: Yu, Jun-lan; Chen, Tian-tian; Zhou, Chen; Lian, Fu-lin; Tang, Xu-long 收藏 \| 浏览/下载：23/0 \| 提交时间：2019/05/09 Fragment-based lead discovery Nmr Bromodomain Brd4 inhibitors
	NMR-based platform for fragment-based lead discovery used in screening BRD4-targeted compounds 期刊论文 OAI收割 ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 7, 页码: 984-993 作者: Yu, Jun-lan; Chen, Tian-tian; Zhou, Chen; Lian, Fu-lin; Tang, Xu-long \| 收藏 \| 浏览/下载：22/0 \| 提交时间：2019/01/08 fragment-based lead discovery NMR bromodomain BRD4 inhibitors
	转录暂停——延伸转变调控小鼠体细胞重编程的机制研究学位论文 OAI收割广州生物院: 中国科学院研究生院, 2015 作者: 许燕 \| 收藏 \| 浏览/下载：20/0 \| 提交时间：2018/12/24 诱导多能干细胞转录调控 RNA聚合酶II 暂停——延伸 P-TEFb KLF4转变