中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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A Computational and Chemical Design Strategy for Manipulating Glycan-Protein Recognition
期刊论文
OAI收割
ADVANCED SCIENCE, 2024, 页码: 14
作者:
Zhu, Qiang
;
Geng, Didi
;
Li, Jingchao
;
Zhang, Jinqiu
;
Sun, Haofan
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/22
CH-pi interaction
glycan-protein recognition
glycoproteomics
PhoSL
core fucose
Distinct roles of the extracellular surface residues of glucagon-like peptide-1 receptor in B-arrestin 1/2 signaling
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACOLOGY, 2024, 卷号: 968, 页码: 17
作者:
Lei, Saifei
;
Meng, Qian
;
Liu, Yanyun
;
Liu, Qiaofeng
;
Dai, Antao
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/05/22
GLP-1R
B-arrestin 1/2
Biased agonism
Bioluminescence resonance energy transfer
Proteomics profiling
Nanobodies as negative allosteric modulators for human calcium sensing receptor
期刊论文
OAI收割
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2024, 卷号: 695, 页码: 9
作者:
Cui, Qianqian
;
Wang, Lu
;
Wang, Haonan
;
Chen, Xiaochen
;
Han, Li
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/04/09
G-protein-coupled receptor
Extracellular calcium sensing receptor
Nanobody
Cryo-electron microscope
Systemic Ca 2+homoeostasis
The emergence of machine learning force fields in drug design
期刊论文
OAI收割
MEDICINAL RESEARCH REVIEWS, 2024, 页码: 36
作者:
Chen, Mingan
;
Jiang, Xinyu
;
Zhang, Lehan
;
Chen, Xiaoxu
;
Wen, Yiming
  |  
收藏
  |  
浏览/下载:16/0
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提交时间:2024/02/19
computational chemistry
drug design
force field
machine learning
molecular modeling
Exploring the mechanism of the PTP1B inhibitors by molecular dynamics and experimental study
期刊论文
OAI收割
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2023, 卷号: 125, 页码: 12
作者:
Zhao, Tian-Tian
;
Hu, Hao-Jie
;
Gao, Li-Xin
;
Zhou, Yu-Bo
;
Zhu, Yun-Long
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Protein tyrosine phosphatases inhibitors
PTP1B inhibitors
Mechanism study
Molecular dynamics
Structural insights into the interaction of three Y- shaped ligands with PI3Kα
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2023, 卷号: 120, 期号: 34, 页码: 9
作者:
Zhou, Qingtong
;
Liu, Xiao
;
Neri, Dario
;
Li, Wenxin
;
Favalli, Nicholas
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收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/12/08
phosphoinositide 3-kinase
drug target
ligand
binding pocket
chemical scaffold
Structural analysis of the dual agonism at GLP-1R and GCGR
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2023, 卷号: 120, 期号: 33, 页码: 12
作者:
Li, Yang
;
Zhou, Qingtong
;
Dai, Antao
;
Zhao, Fenghui
;
Chang, Rulue
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/07
glucagon-like peptide-1 receptor
glucagon receptor
cryo-electron microscopy
dual agonism
Fibroblast Activation Protein Targeting Probe with Gly-Pro Sequence for PET of Glioblastoma
期刊论文
OAI收割
MOLECULAR PHARMACEUTICS, 2023, 卷号: 20, 期号: 8, 页码: 4120-4128
作者:
Lai, Chaoquan
;
Cao, Rui
;
Li, Renda
;
He, Chunfeng
;
Wang, Xiao
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/10/17
glioblastoma
fibroblast activation protein
FAPI
PET imaging
Preferred microenvironments of halogen bonds and hydrogen bonds revealed using statistics and QM/MM calculation studies
期刊论文
OAI收割
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2023, 卷号: 25, 期号: 26, 页码: 17692-17699
作者:
Zhou, Liping
;
Li, Jintian
;
Shi, Yulong
;
Wu, Leyun
;
Zhu, Weiliang
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2023/10/17
Cryo-EM structure of the human chemerin receptor 1-Gi protein complex bound to the C-terminal nonapeptide of chemerin
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2023, 卷号: 120, 期号: 11, 页码: 8
作者:
Wang, Junlin
;
Chen, Geng
;
Liao, Qiwen
;
Lyu, Wenping
;
Liu, Aijun
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/04/09
GPCRs
chemerin
adipokine
innate immunity
cryo-EM