中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [307]
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期刊论文 [853]
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Biochemis... [11]
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Structurally diverse terpenoids and their DRAK2 inhibitory activities: A follow-up study on the vulnerable conifer Pseudotsuga forrestii
期刊论文
OAI收割
JOURNAL OF MOLECULAR STRUCTURE, 2024, 卷号: 1305, 页码: 13
作者:
Zhou, Peng-Jun
;
Huang, Ting
;
Ma, Guang-Lei
;
Zhao, Ze-Yu
;
Jiang, Zhe-Lu
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/05/07
Pseudotsuga forrestii
Rare and endangered plants (REPs)
Triterpene-monoterpene hybrids
GLMDs
DRAK2 inhibition
Molecular docking
A strategy to boost xanthine oxidase and angiotensin converting enzyme inhibitory activities of peptides via molecular docking and module substitution
期刊论文
OAI收割
FOOD CHEMISTRY, 2024, 卷号: 442, 页码: 9
作者:
Meng, Pengfei
;
Wang, Yanxin
;
Huang, Yumeng
;
Liu, Tong
;
Ma, Mingxia
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/07
Peptide
Activity boosting strategy
Molecular docking
Module substitution
Xanthine oxidase inhibitory
Angiotensin-converting enzyme inhibitory
Synaptotagmin 7 docks synaptic vesicles to support facilitation and Doc2α-triggered asynchronous release
期刊论文
OAI收割
ELIFE, 2024, 卷号: 12, 页码: 35
作者:
Wu, Zhenyong
;
Kusick, Grant F.
;
Berns, Manon M. M.
;
Raychaudhuri, Sumana
;
Itoh, Kie
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/07
asynchronous release
short-term plasticity
synaptotagmin
zap-and-freeze
iGluSnFR
synaptic vesicle docking
Mouse
Atranorin inhibits Zika virus infection in human glioblastoma cell line SNB-19 via targeting Zika virus envelope protein
期刊论文
OAI收割
PHYTOMEDICINE, 2024, 卷号: 125, 页码: 11
作者:
Huang, Guan-gen
;
Wang, Hao-yu
;
Wang, Xiao-han
;
Yang, Tao
;
Zhang, Xiao-meng
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Zika virus
SNB-19 cells
Atranorin
Envelope protein
Entry stage
Antiviral drugs
Discovery of a CB2 and 5-HT1A receptor dual agonist for the treatment of depression and anxiety
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 20
作者:
Yang, Wenjiao
;
Gong, Xudong
;
Sun, Haiguo
;
Wu, Chunhui
;
Suo, Jin
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/03/06
CB2R agonist
5-HT1AR agonist
CB1R antagonist
Antidepressant
Anxiolytic
New chromone derivatives bearing thiazolidine-2,4-dione moiety as potent PTP1B inhibitors: Synthesis and biological activity evaluation
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 143, 页码: 9
作者:
Zheng, Yingying
;
Lu, Li
;
Li, Mengyue
;
Xu, Dehua
;
Zhang, Laishun
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/01/26
Chromone
Thiazolidine-2
4-dione
Protein tyrosine phosphatase 1B
Inhibitors
Polymeric membrane potentiometric antibiotic sensors using computer-aided screening of supramolecular macrocyclic carriers
期刊论文
OAI收割
ANALYST, 2024, 页码: 8
作者:
Liu, Aohua
;
Liu, Zhe
;
Liang, Rongning
;
Qin, Wei
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/07
Design and synthesis of cantharidin derivative DCZ5418 as a TRIP13 inhibitor with anti-multiple myeloma activity
in
vitro
and
in
vivo
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 98, 页码: 7
作者:
Dong, Sanfeng
;
Hu, Ke
;
Shi, Yulong
;
Wang, Guanli
;
Yu, Dandan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/02/19
Multiple myeloma
TRIP13 inhibitor
Cantharidin
DCZ5418
DCZ0415
Cryptotanshinone regulates gut microbiota and PI3K-AKT pathway in rats to alleviate CUMS induced depressive symptoms
期刊论文
OAI收割
BIOMEDICINE & PHARMACOTHERAPY, 2023, 卷号: 169, 页码: 11
作者:
Bian, Li-hua
;
Wang, Si-qi
;
Li, Wen-jing
;
Li, Jie
;
Yin, Yi
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/01/18
Depression
Cryptotanshinone
16 S rDNA
Transcriptomics
PI3K-AKT pathway
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:
Zhang, Jingyu
;
Duan, Haiting
;
Gui, Renzhao
;
Wu, Mingfei
;
Shen, Liteng
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/12/19
Acute myeloid leukemia
Bromodomain-containing protein 9
Proteolysis-targeting chimera
Orally bioavailable
Docking