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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
合肥物质科学研究院 [29]
上海药物研究所 [1]
西北高原生物研究所 [1]
大连化学物理研究所 [1]
地球化学研究所 [1]
采集方式
OAI收割 [33]
内容类型
期刊论文 [33]
发表日期
2023 [2]
2022 [2]
2018 [6]
2017 [13]
2016 [8]
2015 [2]
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学科主题
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共33条,第1-10条
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A rapid extraction process monitoring of Swertia mussotii Franch. With near infrared spectroscopy
期刊论文
OAI收割
SPECTROCHIMICA ACTA PART A-MOLECULAR AND BIOMOLECULAR SPECTROSCOPY, 2023, 卷号: 295
作者:
Zhang, Mengqi
;
Zhao, Bing
;
Li, Lian
;
Nie, Lei
;
Li, Peipei
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/12/01
Hydrological niche regulation induced by different resistance strategies facilitates coexistence of P. longipes and L. communis under drought stress
期刊论文
OAI收割
Physiologia Plantarum, 2023, 卷号: 175, 期号: 6
作者:
Kai Yao
;
Aoli Zhang
;
Bo Rang
;
Junting Yang
;
Yingliang Liu
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2024/04/08
A spiropyran with low pK(a) for tracking DNA G-quadruplexes and revealing the dissipation of Delta Psi m with senescence using an in-situ switching strategy
期刊论文
OAI收割
SENSORS AND ACTUATORS B-CHEMICAL, 2022, 卷号: 359
作者:
Tian, Xinrong
;
Li, Jin
;
Zhang, Yanhui
;
Gao, Ying
;
Afzal, Muhammad Wasim
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2022/12/22
Fluorescent probes
G-quadruplexes
Membrane potential of mitochondria
Senescence
Senescent cells
Inhibition of the deubiquitinating enzyme USP47 as a novel targeted therapy for hematologic malignancies expressing mutant EZH2
期刊论文
OAI收割
LEUKEMIA, 2022
作者:
Yang, Jing
  |  
收藏
  |  
浏览/下载:86/0
  |  
提交时间:2022/02/14
Discovery of (E)-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)propanamide (CHMFL-ABL-121) as a highly potent ABL kinase inhibitor capable of overcoming a variety of ABL mutants including T315I for chronic myeloid leukemia
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 160, 页码: 61-81
作者:
Liu, Xuesong
;
Wang, Beilei
;
Chen, Cheng
;
Jiang, Zongru
;
Hu, Chen
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/01/11
ABL kinase
Kinase inhibitor
ABL mutant
CML
Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 896-916
作者:
Wang, Beilei
;
Wu, Jiaxin
;
Wu, Yun
;
Chen, Cheng
;
Zou, Fengming
  |  
收藏
  |  
浏览/下载:77/0
  |  
提交时间:2019/12/25
CDK9
Kinase inhibitor
Structure-activity relationship
Leukemia
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3K delta) inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 页码: 831-846
作者:
Liang, Xiaofei
;
Li, Feng
;
Chen, Cheng
;
Jiang, Zongru
;
Wang, Aoli
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2019/12/10
PI3K delta
Kinase inhibitor
Acute myeloid leukemia
Structure-activity relationship
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:
Xue, Yu
;
Song, Peiran
;
Song, Zilan
;
Wang, Aoli
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2019/08/23
Discovery of 4,7-Diamino-5-(4-phenoxyphenyl)-6-methylene-pyrinnido[5,4-b]pyrrolizines as Novel Bruton's Tyrosine Kinase Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 10, 页码: 4608-4627
作者:
Xue, Yu
;
Song, Peiran
;
Song, Zilan
;
Wang, Aoli
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2019/01/08
Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFR alpha kinase inhibitor for PDGFR alpha driving chronic eosinophilic leukemia
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 期号: 无, 页码: 366-384
作者:
Wang, Qiang
;
Liu, Feiyang
;
Qi, Shuang
;
Qi, Ziping
;
Yan, Xiao-E.
  |  
收藏
  |  
浏览/下载:75/0
  |  
提交时间:2019/06/10
PDGFR kinase
Type II inhibitor
Kinase inhibitor
CEL