中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共79条,第1-10条 帮助

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Discovery of peptidomimetic spiropyrrolidine derivatives as novel 3CLpro inhibitors against SARS-CoV-2 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 281, 页码: 22
作者:  
Guma, Samuel Desta;  Zhou, Zhaoyin;  Song, Kang;  Yang, Feipu;  Suo, Jin
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/12/11
F-CPI: A Multimodal Deep Learning Approach for Predicting Compound Bioactivity Changes Induced by Fluorine Substitution 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 13
作者:  
Zhang, Qian;  Yin, Wenhai;  Chen, Xinyao;  Zhou, Aimin;  Zhang, Guixu
  |  收藏  |  浏览/下载:6/0  |  提交时间:2025/02/28
Direct Reductive N-alkylation of Amines with Carboxylic Esters 期刊论文  OAI收割
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2024, 页码: 7
作者:  
Zhang, Yuxuan;  Bonku, Emmanuel Mintah;  Yang, Xingbang;  Zhu, Fuqiang
  |  收藏  |  浏览/下载:7/0  |  提交时间:2025/01/14
Design, synthesis, and evaluation of novel oxyacanthine derivatives for anti-SARS-CoV-2 activity 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 113, 页码: 5
作者:  
Lu, Jie;  Cheng, Yan;  Zhang, Yumin;  Wang, Yi;  Xia, Bingqing
  |  收藏  |  浏览/下载:4/0  |  提交时间:2025/02/28
Discovery of the potent covalent inhibitor with an acrylate warhead for SARS-CoV-2 3CL protease 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 112, 页码: 5
作者:  
Shen, Wen;  Chen, Xinyao;  Zhou, Liping;  Cheng, Yan;  Zhang, Yan
  |  收藏  |  浏览/下载:22/0  |  提交时间:2024/10/21
Identification of Dihydrobenzofuran Neolignans as Novel PDE4 Inhibitors and Evaluation of Antiatopic Dermatitis Efficacy in DNCB-Induced Mice Model 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 6, 页码: 4855-4869
作者:  
Gu, Chenming;  Liu, Jiayuan;  Qian, Fei;  Yu, Wenchao;  Huang, Doudou
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/05/07
TPN10475 Constrains Effector T Lymphocytes Activation and Attenuates Experimental Autoimmune Encephalomyelitis Pathogenesis by Facilitating TGF-β Signal Transduction 期刊论文  OAI收割
JOURNAL OF NEUROIMMUNE PHARMACOLOGY, 2024, 卷号: 19, 期号: 1, 页码: 16
作者:  
Wang, Chun;  Jiang, Xiangrui;  Lv, Jie;  Zhuang, Wei;  Xie, Ling
  |  收藏  |  浏览/下载:34/0  |  提交时间:2024/04/09
Discovery of a CB2 and 5-HT1A receptor dual agonist for the treatment of depression and anxiety 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 20
作者:  
Yang, Wenjiao;  Gong, Xudong;  Sun, Haiguo;  Wu, Chunhui;  Suo, Jin
  |  收藏  |  浏览/下载:18/0  |  提交时间:2024/03/06
Dual-channel hypergraph convolutional network for predicting herb-disease associations 期刊论文  OAI收割
BRIEFINGS IN BIOINFORMATICS, 2024, 卷号: 25, 期号: 2, 页码: 13
作者:  
Hu, Lun;  Zhang, Menglong;  Hu, Pengwei;  Zhang, Jun;  Niu, Chao
  |  收藏  |  浏览/下载:5/0  |  提交时间:2024/08/22
Glimepiride, a novel soluble epoxide hydrolase inhibitor, protects against heart failure via increasing epoxyeicosatrienoic acids 期刊论文  OAI收割
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 2023, 卷号: 185, 页码: 13-25
作者:  
Zhao, Chengcheng;  Jiang, Xiangrui;  Peng, Liyuan;  Zhang, Yan;  Li, Huihui
  |  收藏  |  浏览/下载:40/0  |  提交时间:2024/01/16