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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [12]
寒区旱区环境与工程研... [1]
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期刊论文 [13]
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2023 [1]
2019 [1]
2018 [3]
2017 [1]
2016 [4]
2015 [2]
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Structural Optimization of Fibroblast Growth Factor Receptor Inhibitors for Treating Solid Tumors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 5, 页码: 3226-3249
作者:
Li, Chunpu
;
Dai, Yang
;
Kong, Xiangtai
;
Wang, Bao
;
Peng, Xia
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/03/27
Recyclable and Stable alpha-Methylproline-Derived Chiral Ligands for the Chemical Dynamic Kinetic Resolution of free C,N-Unprotected alpha-Amino Acids
期刊论文
OAI收割
MOLECULES, 2019, 卷号: 24, 期号: 12, 页码: 19
作者:
Shu, Shuangjie
;
Zhao, Liang
;
Zhou, Shengbin
;
Wu, Chenglin
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/07/01
quaternary carbon
dynamic kinetic resolution
unprotected alpha-amino acids
Schiff base intermediates
ligands
Discovery of thiophene-containing biaryl amide derivatives as novel glucagon receptor antagonists
期刊论文
OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2018, 卷号: 92, 期号: 1, 页码: 1241-1254
作者:
Li, Jia
;
Feng, Yang
;
Li, Huihui
;
Shu, Shuangjie
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2019/01/08
biaryl amide
glucagon receptor antagonist
molecular simulation
A novel series of 4-methyl substituted pyrazole derivatives as potent glucagon receptor antagonists: Design, synthesis and evaluation of biological activities
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1896-1908
作者:
Shu, Shuangjie
;
Dai, Antao
;
Wang, Jiang
;
Wang, Bin
;
Feng, Yang
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
Pyrazole derivatives
Glucagon receptor antagonist
Docking study
Binding pocket
Cobalt-catalyzed C(sp(3))-H/C(sp(2))-H oxidative coupling between alkanes and benzamides
期刊论文
OAI收割
RSC ADVANCES, 2018, 卷号: 8, 期号: 24, 页码: 13454-13458
作者:
Li, Shuangjie
;
Wang, Bao
;
Dong, Guangyu
;
Li, Chunpu
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2019/01/08
Palladium-Catalyzed Ortho-Alkoxylation of N-Benzoyl alpha-Amino Acid Derivatives at Room Temperature
期刊论文
OAI收割
JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 82, 期号: 1, 页码: 126-134
作者:
Li, Shuangjie
;
Zhu, Wei
;
Gao, Feng
;
Li, Chunpu
;
Wang, Jiang
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
Nickel-Catalyzed ortho-C-H Thiolation of N-Benzoyl alpha-Amino Acid Derivatives
期刊论文
OAI收割
JOURNAL OF ORGANIC CHEMISTRY, 2016, 卷号: 81, 期号: 19, 页码: 9122-9130
作者:
Gao, Feng
;
Zhu, Wei
;
Zhang, Dengyou
;
Li, Shuangjie
;
Wang, Jiang
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
Design, synthesis, structure-activity relationships, and docking studies of pyrazole-containing derivatives as a novel series of potent glucagon receptor antagonists
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 12, 页码: 2852-2863
作者:
Shu, Shuangjie
;
Cai, Xiaoqing
;
Li, Jia
;
Feng, Yang
;
Dai, Antao
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
Glucagon receptor
Antagonist
Molecular docking
Pyrazole
Type 2 diabetes mellitus
Advanced asymmetric synthesis of (1R,2S)-1-amino-2-vinylcyclopropanecarboxylic acid by alkylation/cyclization of newly designed axially chiral Ni(II) complex of glycine Schiff base
期刊论文
OAI收割
AMINO ACIDS, 2016, 卷号: 48, 期号: 4, 页码: 973-986
作者:
Kawashima, Aki
;
Shu, Shuangjie
;
Takeda, Ryosuke
;
Kawamura, Akie
;
Sato, Tatsunori
  |  
收藏
  |  
浏览/下载:177/0
  |  
提交时间:2019/01/08
Anti-viral (HCV) activity
Asymmetric synthesis
Amino acids
Chirality
Schiff bases
Application of Sulfonyl in Drug Design
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2016, 卷号: 36, 期号: 3, 页码: 490-501
作者:
Zhao Fei
;
Wang Jiang
;
Ding Xiao
;
Shu Shuangjie
;
Liu Hong
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
sulfonyl
drug design
lead optimization