中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [45]
上海生物化学与细胞生... [5]
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期刊论文 [71]
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HDAC inhibitor GCJ-490A modulates tumor microenvironment and synergizes with PD-1 antibody against breast and lung cancers in syngeneic murine models
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 13
作者:
Zhang, Wen-xin
;
He, Ting
;
Fang, Kun
;
Gao, Ying-lei
;
Sun, Yi-ming
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Mechanism of hydroxamic acid group metabolism to carboxylic acid: Oxidation versus hydrolysis
期刊论文
OAI收割
DRUG METABOLISM AND DISPOSITION, 2025, 卷号: 53, 期号: 10, 页码: 11
作者:
Huang, Xiyue
;
Zhou, Lei
;
Chen, Huixian
;
Sun, Xiaowei
;
Cao, Mengyi
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Discovery of a potential hematologic malignancies therapy: Selective and potent HDAC7 PROTAC degrader targeting non-enzymatic function
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 3, 页码: 1659-1679
作者:
Jin, Yuheng
;
Qi, Xuxin
;
Yu, Xiaoli
;
Cheng, Xirui
;
Chen, Boya
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IHCH9033, a novel class I HDAC inhibitor, synergizes with FLT3 inhibitor and rescues quizartinib resistance in FLT3-ITD AML via enhancing DNA damage response
期刊论文
OAI收割
EXPERIMENTAL HEMATOLOGY & ONCOLOGY, 2025, 卷号: 14, 期号: 1, 页码: 19
作者:
Yao, Mingyue
;
Yan, Wenzhong
;
Wang, Yafang
;
Zhao, Yu
;
Xu, Xiaowei
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Design, Synthesis, and Biological Evaluation of HDAC Inhibitors Containing Natural Product-Inspired
N
-Linked 2-Acetylpyrrole Cap
期刊论文
OAI收割
MOLECULES, 2024, 卷号: 29, 期号: 19, 页码: 26
作者:
Zhang, Han
;
Shen, Qianqian
;
Hu, Zhu
;
Wu, Pei-Qian
;
Chen, Yi
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NIR-II fluorescence-guided liver cancer surgery by a small molecular HDAC6 targeting probe
期刊论文
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EBIOMEDICINE, 2023, 卷号: 98, 页码: 18
作者:
Wang, Bo
;
Tang, Chu
;
Lin, En
;
Jia, Xiaohua
;
Xie, Ganyuan
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The intrinsic effects of using rhenium gaskets in hydrothermal diamond anvil cell experiments on background fluorescence, contamination, and redox control
期刊论文
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CHEMICAL GEOLOGY, CHEMICAL GEOLOGY, 2023, 2023, 卷号: 632, 632, 页码: 14, 14
作者:
Cheng, Nanfei
;
Chou, I. -Ming
;
Wan, Ye
;
Wang, Ruoheng
;
Zhang, Haiyan
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Hedgehog pathway orchestrates the interplay of histone modifications and tailors combination epigenetic therapies in breast cancer
期刊论文
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ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 6, 页码: 2601-2612
作者:
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The HDAC inhibitor GCJ-490A suppresses c-Met expression through IKK? and overcomes gefitinib resistance in non-small cell lung cancer
期刊论文
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CANCER BIOLOGY & MEDICINE, 2022, 卷号: 19, 期号: 8, 页码: 1172-1192
作者:
He, Ting
;
Gao, Yinglei
;
Fang, Yanfen
;
Zhang, Yangming
;
Zhang, Shuwei
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A novel aromatic amide derivative SY-65 co-targeted tubulin and histone deacetylase 1 with potent anticancer activity in vitro and in vivo
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2022, 卷号: 201, 页码: 115070
作者:
Li, Yin-Ru
;
Liu, Fang-Fang
;
Liu, Wen-Bo
;
Zhang, Yi-Fan
;
Tian, Xin-Yi
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