中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [8]
合肥物质科学研究院 [2]
烟台海岸带研究所 [1]
采集方式
OAI收割 [11]
内容类型
期刊论文 [11]
发表日期
2022 [1]
2018 [4]
2015 [4]
2013 [1]
2012 [1]
学科主题
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Genome-wide gain-of-function screening identifies EZH2 mediating resistance to PI3K alpha inhibitors in oesophageal squamous cell carcinoma
期刊论文
OAI收割
CLINICAL AND TRANSLATIONAL MEDICINE, 2022, 卷号: 12, 期号: 5, 页码: 17
作者:
Xing, Hui
;
Gao, Mengshi
;
Wang, Yuxiang
;
Zhang, Xu
;
Shi, Jiajie
  |  
收藏
  |  
浏览/下载:61/0
  |  
提交时间:2022/08/16
CDKNIA
cell cycle
CRISPR-SAM
CYH33
ESCC
EZH2
PI3K alpha inhibitor
resistance
Serum and glucocorticoid inducible protein kinases (SGKs): a potential target for cancer intervention
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2018, 卷号: 8, 期号: 5, 页码: 767-771
作者:
Basnet, Rajesh
;
Gong, Grace Qun
;
Li, Chenyao
;
Wang, Ming-Wei
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2019/01/08
SGK
AKT
PI3K
Cancer
Signalling: Kinase
Inhibitor
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3K delta) inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 页码: 831-846
作者:
Liang, Xiaofei
;
Li, Feng
;
Chen, Cheng
;
Jiang, Zongru
;
Wang, Aoli
  |  
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2019/12/10
PI3K delta
Kinase inhibitor
Acute myeloid leukemia
Structure-activity relationship
PI3K signaling pathways modulated white spot syndrome virus (WSSV) replication in Procambarus clarkii
期刊论文
OAI收割
FISH & SHELLFISH IMMUNOLOGY, 2018, 卷号: 76, 页码: 279-286
作者:
Zhang, Huijing
;
Yao, Xuemei
;
Ding, Yunfei
;
Xu, Zheng
;
Liang, Rongning
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/07/08
PI3K
WSSV replication
Apoptosis
Bax
Bax inhibitor-1
Lectin
Toll
Procambarus clarkii
serumandglucocorticoidinducibleproteinkinasessgksapotentialtargetforcancerintervention
期刊论文
OAI收割
actapharmaceuticasinicab, 2018, 卷号: 000, 期号: 005, 页码: 767
作者:
Basnet Rajesh
;
Gong Grace Qun
;
Li Chenyao
;
Wang Mingwei
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2020/07/01
SGK
AKT
PI3K
Cancer
Signalling
Kinase
Inhibitor
PI3K isoform-selective inhibitors: next-generation targeted cancer therapies
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2015, 卷号: 36, 期号: 10, 页码: 1170-1176
作者:
Wang, Xiang
;
Ding, Jian
;
Meng, Ling-hua
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2019/01/08
PI3K isoforms
isoform-selective inhibitor
CAL101
precise cancer therapy
biomarker
Targeting PI3K: Emerging Therapy for Chronic Lymphocytic Leukemia and Beyond
期刊论文
OAI收割
MEDICINAL RESEARCH REVIEWS, 2015, 卷号: 35, 期号: 4, 页码: 720-752
作者:
Wei, Manman
;
Wang, Xiang
;
Song, Zilan
;
Jiao, Mingkun
;
Ding, Jian
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
chronic lymphocytic leukemia
PI3K
inhibitor
molecularly targeted therapy
idelalisib
Design, synthesis and biological evaluation of acylhydrazone derivatives as PI3K inhibitors
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 1, 页码: 118-120
作者:
Gao, Guo-Rui
;
Liu, Jia-Li
;
Mei, De-Sheng
;
Ding, Jian
;
Meng, Ling-Hua
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
PI3K
Inhibitor
Aclhydrazone
designsynthesisandbiologicalevaluationofacylhydrazonederivativesaspi3kinhibitors
期刊论文
OAI收割
chinesechemicalletters, 2015, 卷号: 26, 期号: 1, 页码: 118
作者:
Gao Guorui
;
Liu Jiali
;
Mei Desheng
;
Ding Jian
;
Meng Linghua
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2020/07/01
PI3-KINASE P110-ALPHA INHIBITORS
3-KINASE
PATHWAY
PI3K
Inhibitor
Aclhydrazone
A pharmacological model reveals biased dependency on PI3K isoforms for tumor cell growth
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2013, 卷号: 34, 期号: 9, 页码: 1201-1207
作者:
Wang, Xiang
;
Li, Jia-peng
;
Yang, Yan
;
Ding, Jian
;
Meng, Ling-hua
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
anticancer drug
PI3K inhibitor
drug selectivity
WJD008
prostate cancer
B cell type leukemia
screening model