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CAS IR Grid
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化学研究所 [30]
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期刊论文 [150]
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Discovery of novel GluN1/GluN3A NMDA receptor inhibitors using a deep learning-based method
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 8
作者:
Wang, Shi-hang
;
Zeng, Yue
;
Yang, Hao
;
Tian, Si-yuan
;
Zhou, Yong-qi
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2025/07/25
N
-methyl-
D
-aspartate receptors
GluN1/GluN3A
ligand-based virtual screening
scaffold hopping
deep learning
GeminiMol
Biodegradable cellulose scaffolds embedding kartogenin-loaded microspheres for cartilage regeneration
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2025, 卷号: 306, 页码: 11
作者:
Yu, Xinding
;
Wang, Jian
;
Zhou, Shenglai
;
Pan, Peng
;
Chen, Tiantian
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/04/27
Cartilage defect
Microspheres
Composite scaffold
Novel 5-alkenylthiothiazolidinone scaffold discovery as Multi-Chitinases inhibitors to arrest the molting of Asian corn borer
期刊论文
OAI收割
JOURNAL OF MOLECULAR STRUCTURE, 2025, 卷号: 1321, 页码: 11
作者:
Shi, Dongmei
;
Ji, Xinge
;
Zou, Renxuan
;
Jiang, Zhiyang
;
Duan, Yangwei
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2024/10/21
5-alkenylthiothiazolidinone scaffold
Multichitinase inhibitor
Amide bond
Asian corn borer
insect growth regulator
3D chitosan scaffolds loaded with ZnO nanoparticles for bone tissue engineering
期刊论文
OAI收割
COLLOIDS AND SURFACES B-BIOINTERFACES, 2025, 卷号: 245, 页码: 9
作者:
Tang, Wenmin
;
Pan, Peng
;
Chen, Tiantian
;
Wang, Jian
;
Cui, Xiangnan
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/04/27
Zinc oxide nanoparticles
Chitosan
Tissue engineering scaffold
Bone repair
3D chitosan scaffolds loaded with ZnO nanoparticles for bone tissue engineering
期刊论文
OAI收割
COLLOIDS AND SURFACES B-BIOINTERFACES, 2025, 卷号: 245, 页码: 9
作者:
Tang, Wenmin
;
Pan, Peng
;
Chen, Tiantian
;
Wang, Jian
;
Cui, Xiangnan
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/04/27
Zinc oxide nanoparticles
Chitosan
Tissue engineering scaffold
Bone repair
The application of nanodiscs in membrane protein drug discovery & development and drug delivery
期刊论文
OAI收割
FRONTIERS IN CHEMISTRY, 2024, 卷号: 12
作者:
Dong, Yingkui
;
Tang, Huan
;
Dai, Han
;
Zhao, Hongxin
;
Wang, Junfeng
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2024/11/20
nanodisc (ND)
membrane protein
drug discovery & development
drug delievery
membrane scaffold protein (MSP)
Discovery and characterization of novel potent non-covalent small molecule inhibitors targeting papain-like protease from SARS-CoV-2
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 7, 页码: 3286-3290
作者:
Zheng, Miao
;
Feng, Bo
;
Zhang, Yumin
;
Liu, Xin
;
Zhao, Na
  |  
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2024/08/22
Non-covalent PLpro inhibitors
Antiviral activity
Structural-based drug design
Imidazo[4,5-b]pyridine scaffold
Discovery of a 1,6-naphthyridin-4-one-based AXL inhibitor with improved pharmacokinetics and enhanced in vivo antitumor efficacy
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 17
作者:
Lan, Yaohan
;
Peng, Xia
;
Ji, Yinchun
;
Su, Yi
;
Duan, Wenhu
  |  
收藏
  |  
浏览/下载:73/0
  |  
提交时间:2024/02/27
AXL inhibitor
In vivo antitumor efficacy
6-Naphthyridin-4-one derivatives
Scaffold hopping
Structure-based drug design
Physically cross-linked chitosan gel with tunable mechanics and biodegradability for tissue engineering scaffold
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2024, 卷号: 257, 页码: 12
作者:
Pan, Peng
;
Wang, Jian
;
Wang, Xi
;
Kang, Ye
;
Yu, Xinding
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/04/27
Physical chitosan gel
Water content
Tissue engineering scaffold
Physically cross-linked chitosan gel with tunable mechanics and biodegradability for tissue engineering scaffold
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2024, 卷号: 257, 页码: 12
作者:
Pan, Peng
;
Wang, Jian
;
Wang, Xi
;
Kang, Ye
;
Yu, Xinding
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/04/27
Physical chitosan gel
Water content
Tissue engineering scaffold