中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [8]
中国科学院大学 [2]
兰州化学物理研究所 [1]
采集方式
OAI收割 [9]
iSwitch采集 [2]
内容类型
期刊论文 [11]
发表日期
2016 [1]
2013 [1]
2010 [1]
2009 [1]
2007 [1]
2006 [2]
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学科主题
Research &... [1]
分析化学与药物化学 [1]
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Characterization of TPN729 metabolites in humans using ultra-performance liquid chromatography/quadrupole time-of-flight mass spectrometry
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2016, 卷号: 117, 页码: 217-226
作者:
Zhu, Yunting
;
Li, Liang
;
Deng, Pan
;
Chen, Xiaoyan
;
Zhong, Dafang
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
TPN729
UPLC/Q-TOF MS
Metabolite identification
Metabolic pathways
Human
Sildenafil
Magnetic molecularly imprinted polymer for the selective extraction of sildenafil, vardenafil and their analogs from herbal medicines
期刊论文
OAI收割
Talanta, 2013, 卷号: 115, 页码: 482-489
作者:
Chen FF(陈方方)
;
Jie XY(解笑瑜)
;
Shi YP(师彦平)
;
Shi YP(师彦平)
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2013/12/11
Magnetic molecularly imprinted polymers
Herbal medicines
Phosphodiesterase type-5 inhibitors
Sildenafil
Solid phase extraction
Synthesis and phosphodiesterase type-5 inhibitory activity of sildenafil analogues possessing a guanidine group in the phenyl ring
期刊论文
OAI收割
Journal of China Pharmaceutical University, 2010, 卷号: 41, 期号: 2, 页码: 112-117
作者:
Shi J(石静)
;
Liu Z(刘正)
;
Wang Z(王 震)
;
Tian GH(田广辉)
;
Yang XJ(杨小军)
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
sildenafil analogues
guanidine group
PDE5 inhibitor
2-Phenylquinazolin-4(3H)-one, a class of potent PDE5 inhibitors with high selectivity versus PDE6
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 卷号: 19, 期号: 10, 页码: 2777-2779
作者:
Duan, Hongliang
;
Zheng, Jin
;
Lai, Qinglin
;
Liu, Zheng
;
Tian, Guanghui
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
2-Phenylquinazolin-4(3H)-one
PDE5 Inhibitor
Selectivity versus PDE6
Sildenafil
Erectile dysfunction
synthesisandevaluationofpde5inhibitoryactivityofnovelpyrido2151pyrazolo43dpyrimidin4onederivatives
期刊论文
OAI收割
chinesejournalofchemistry, 2007, 卷号: 25, 期号: 2, 页码: 241
作者:
GuangHui Tian
;
GuangXin Xia
;
WeiXi Jin
;
XinJian Chen
;
ShunAn Lai
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/07/01
ERECTILE DYSFUNCTION
RECEPTOR ANTAGONISTS
SILDENAFIL ANALOGS
POTENT
PHOSPHODIESTERASE
Bosentan, sildenafil, and their combination in the monocrotaline model of pulmonary hypertension in rats
期刊论文
OAI收割
EXPERIMENTAL BIOLOGY AND MEDICINE, 2006, 卷号: 231, 期号: 6, 页码: 967-973
作者:
Clozel, M
;
Hess, P
;
Rey, M
;
Iglarz, M
;
Binkert, C
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
bosentan
endothelin
nitric oxide
pulmonary hypertension
sildenafil
Design and synthesis of pyrido[1,2-e]purin-4(3h)-one derivatives as potential pde 5 inhibitors
期刊论文
iSwitch采集
Chinese chemical letters, 2005, 卷号: 16, 期号: 10, 页码: 1283-1286
作者:
Xia, GX
;
Li, JF
;
Lai, SA
;
Peng, AM
;
Zhang, SJ
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/05/10
Pyrido[1,2-e]purin-4(3h)-one
Pde5 inhibitor
Sildenafil
Erectile dysfunction (ed)
Design and synthesis of pyrido[1,2-e]purin-4(3H)-one derivatives as potential PDE 5 inhibitors
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2005, 卷号: 16, 期号: 10, 页码: 1283-1286
作者:
Xia, GX
;
Li, JF
;
Lai, SA
;
Peng, AM
;
Zhang, SJ
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
pyrido[1,2-e]purin-4(3H)-one
PDE5 inhibitor
sildenafil
erectile dysfunction (ED)
Synthesis and phosphodiesterase 5 inhibitory activity of novel pyrido[1,2-e]purin-4(3h)-one derivatives
期刊论文
iSwitch采集
Bioorganic & medicinal chemistry letters, 2005, 卷号: 15, 期号: 11, 页码: 2790-2794
作者:
Xia, GX
;
Li, JF
;
Peng, AM
;
Lai, SN
;
Zhang, SJ
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/05/10
Pyrido[1,2-e]purin-4(3h)-one
Pde5 inhibitor
Sildenafil
Erectile dysfunction