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Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [10]
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期刊论文 [19]
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Structural basis of peptidomimetic agonism revealed by small-molecule GLP-1R agonists Boc5 and WB4-24
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 卷号: 119, 期号: 20, 页码: 10
作者:
Cong, Zhaotong
;
Zhou, Qingtong
;
Li, Yang
;
Chen, Li-Nan
;
Zhang, Zi-Chen
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2022/09/30
glucagon-like peptide-1 receptor
type 2 diabetes mellitus
cryoelectron microscopy
peptidomimetic agonism
Signaling profiles in HEK 293T cells co-expressing GLP-1 and GIP receptors
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 8
作者:
Wang, Yu-zhe
;
Yang, De-hua
;
Wang, Ming-wei
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2021/11/04
glucagon-like peptide-1 receptor
glucose-dependent insulinotropic peptide receptor
peptide 19
LY3298176
heteromerization
type 2 diabetes
Inositol polyphosphate multikinase IPMK-1 regulates development through IP3/calcium signaling in Caenorhabditis elegans
期刊论文
OAI收割
CELL CALCIUM, 2021, 卷号: 93, 页码: 102327
作者:
Yang,Zhong-Lin
;
Chen,Jian-Ning
;
Lu,Yu-Yang
;
Lu,Min
;
Wan,Qin-Li
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2022/04/02
Inositol polyphosphates
Inositol polyphosphate multikinase
Type I inositol 5-phosphatase
Development
Calcium signaling
Defecation rhythm
C. elegans
C-ELEGANS
PHOSPHOLIPASE-C
CALCIUM
1,4,5-TRISPHOSPHATE
CALCINEURIN
KINASE
IDENTIFICATION
TRISPHOSPHATE
METABOLISM
RECEPTOR
Systematic characterization of AT1 receptor antagonists with label-free dynamic mass redistribution assays
期刊论文
OAI收割
JOURNAL OF PHARMACOLOGICAL AND TOXICOLOGICAL METHODS, 2020, 卷号: 102
作者:
Qu, Lala
;
Wang, Jixia
;
Hou, Tao
;
Zhou, Han
;
Wang, Zhiwei
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/11/25
Angiotensin II type 1 receptor
Antagonist
Binding property
Dynamic mass redistribution assay
Functional, signalling and transcriptional differences of three distinct type I IFNs in a perciform fish, the mandarin fish Siniperca chuatsi
期刊论文
OAI收割
DEVELOPMENTAL AND COMPARATIVE IMMUNOLOGY, 2018, 卷号: 84, 期号: 1, 页码: 94-108
作者:
Laghari, Zubair Ahmed
;
Chen, Shan Nan
;
Li, Li
;
Huang, Bei
;
Gan, Zhen
  |  
收藏
  |  
浏览/下载:105/0
  |  
提交时间:2019/07/03
Type I IFN
Cytokine receptor family B
CRFB
STAT1
STAT2
IRF3
IRF7
Teleost fish
Single-molecule force spectroscopy study of interactions between angiotensin II type 1 receptor and different biased ligands in living cells
期刊论文
OAI收割
ANALYTICAL AND BIOANALYTICAL CHEMISTRY, 2018, 卷号: 410, 期号: 14, 页码: 3275-3284
作者:
Li, Wenhui
;
Xu, Jiachao
;
Kou, Xiaolong
;
Zhao, Rong
;
Zhou, Wei
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2019/04/09
Angiotensin Ii Type 1 Receptor
Biased Ligands
Atomic Force Microscopy
Single-molecule Force Spectroscopy
Energy Landscape
An activity-based probe reveals dynamic protein-protein interactions mediating IGF-1R transactivation by the GABA(B) receptor
期刊论文
OAI收割
BIOCHEMICAL JOURNAL, 2012, 卷号: 443, 页码: 627-634
作者:
Lin, Xin
;
Li, Xin
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2019/01/08
activity-based probe
gamma-aminobutyric acid B receptor (GABA(B) receptor)
dynamic protein-protein interaction
insulin-like growth factor type I receptor (IGF-1R)
transactivation
Microarray analysis of responsible genes in increased growth rate in the subline of HL60 (HL60RG) cells
期刊论文
OAI收割
MUTATION RESEARCH-FUNDAMENTAL AND MOLECULAR MECHANISMS OF MUTAGENESIS, 2012, 卷号: 731, 期号: 1-2, 页码: 20-26
作者:
Luan, Yang
;
Kogi, Mieko
;
Rajaguru, Palanisamy
;
Ren, Jin
;
Yamaguchi, Teruhide
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
Microarray analysis
HL60 cells
HL60RG cell
Type II tumor necrosis factor-alpha receptor (TNFRSF1B)
TNFRSF8
A continued saga of Boc5, the first non-peptidic glucagon-like peptide-1 receptor agonist with in vivo activities
期刊论文
OAI收割
acta pharmacologica sinica, 2012, 卷号: 33, 期号: 2, 页码: 148-154
作者:
He, Min
;
Guan, Ni
;
Gao, Wei-wei
;
Liu, Qing
;
Wu, Xiao-yan
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2015/11/13
type 2 diabetes
glucagon-like peptide-1
non-peptidic agonist
Boc5
G-protein coupled receptor
A continued saga of Boc5, the first non-peptidic glucagon-like peptide-1 receptor agonist with in vivo activities
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 2, 页码: 148-154
作者:
He, Min
;
Guan, Ni
;
Gao, Wei-wei
;
Liu, Qing
;
Wu, Xiao-yan
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
type 2 diabetes
glucagon-like peptide-1
non-peptidic agonist
Boc5
G-protein coupled receptor