中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
高能物理研究所 [4]
上海药物研究所 [3]
昆明植物研究所 [2]
海洋研究所 [1]
采集方式
OAI收割 [9]
iSwitch采集 [1]
内容类型
期刊论文 [10]
发表日期
2021 [2]
2019 [1]
2017 [2]
2016 [3]
2012 [2]
学科主题
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Chemical profiling and antidiabetic potency of Paeonia delavayi: Comparison between different parts and constituents
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2021, 卷号: 198, 页码: 113998
作者:
Huang,Qian
;
Chen,Ji-Jun
;
Pan,Yang
;
He,Xiao-Feng
;
Wang,Yuan
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2022/04/02
Paeonia delavayi
Chemical comparison
LCMS analyses
Antidiabetic effects
PTP1B/TCPTP selective inhibitors
LIQUID-CHROMATOGRAPHY
MULTIPLE CONSTITUENTS
RAPID IDENTIFICATION
GLYCOSIDES
ROOT
DERIVATIVES
TARGETS
CAPSULE
L.
Diarylheptanoid-chalcone hybrids with PTP1B and alpha-glucosidase dual inhibition from Alpinia katsumadai
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 108, 页码: 104683
作者:
He,Xiao-Feng
;
Chen,Ji-Jun
;
Li,Tian-Ze
;
Hu,Jing
;
Zhang,Xue-Mei
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2022/04/02
Alpinia katsumadai
Katsumadainols A(1)-A(16)
PTP1B/TCPTP selective inhibitors
alpha-glucosidase inhibitors
Antidiabetic effects
THEORETICAL CALCULATION
ABSOLUTE-CONFIGURATION
SEEDS
BLEPHAROCALYXINS
ADDUCT
MOIETY
Identification and characterization of potent and selective inhibitors targeting protein tyrosine phosphatase 1B (PTP1B)
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 16, 页码: 2358-2363
作者:
Jin, Jia
;
Ye, Xiaoqing
;
Boateng, Derrick
;
Dai, Kaili
;
Ye, Fei
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/03/21
PTP1B
TCPTP
Type 2 diabetes
Selective inhibitors
Dihydropyridine thione
Synthesis, crystal structure and ptps inhibition of a zinc(ii) complex with n-(4-hydroxybenzyl)-l-serine
期刊论文
iSwitch采集
Chinese journal of structural chemistry, 2017, 卷号: 36, 期号: 2, 页码: 316-323
作者:
Li Yan-Hong
;
Lu Li-Ping
;
Zhu Miao-Li
;
Yuan Cai-Xia
;
Feng Si-Si
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/04/23
Zinc(ii) complex
N-(4-hydroxybenzyl)-l-serine
Crystal structure
Inhibitory activity
Ptp1b
Tcptp
Synthesis, Crystal Structure and PTPs Inhibition of a Zinc(II) Complex with N-(4-hydroxybenzyl)-L-serine
期刊论文
OAI收割
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY结构化学, 2017, 卷号: 36, 期号: 2, 页码: 316-323
作者:
Zhu, ML
;
Yuan, CX
;
Feng, SS
;
Gao ZQ(高增强)
;
Gao, ZQ
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/08/27
zinc(II) complex
N-(4-hydroxybenzyl)-L-serine
crystal structure
inhibitory activity
PTP1B
TCPTP
The design strategy of selective PTP1B inhibitors over TCPTP
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 16, 页码: 3343-3352
作者:
Li, XiangQian
;
Wang, LiJun
;
Shi, DaYong
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2016/12/05
Selectivity
PTP1B inhibitor
TCPTP
Diabetes
Design strategy
A Copper(II) Complex Based on N-(4-hydroxybenzyl)-L-serine: Synthesis, Crystal Structure and Inhibitory Activity on PTP1B and TCPTP
期刊论文
OAI收割
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY, 2016, 卷号: 35, 期号: 11, 页码: 1686-1693
作者:
Li, YH
;
Lu, LP
;
Zhu, ML
;
Yuan, CX
;
Feng, SS
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2017/07/24
copper(II) complex
N-(4-hydroxybenzyl)-L-serine
crystal structure
inhibitor
PTP1B
TCPTP
Synthesis, Crystal Structure and Protein Tyrosine Phosphatase Inhibition of a Copper(II) Complex with N-(2-Pyridylmethyl)-L-serine
期刊论文
OAI收割
CHEMICAL JOURNAL OF CHINESE UNIVERSITIES-CHINESE, 2016, 卷号: 37, 期号: 12, 页码: 2138-2143
作者:
Li, YH
;
Yuan, CX
;
Lu, LP
;
Zhu, ML
;
Fu, XQ
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2017/07/24
Copper(II) complex
N-(2-Pyridylmethyl)-L-serine
Inhibitor
PTP1B
TCPTP
DESIGN, SYNTHESIS AND BIOLOGICAL ACTIVITY EVALUATION OF 2-MERCAPTO-4(3H)-QUINAZOLINONE DERIVATIVES AS NOVEL INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE 1B
期刊论文
OAI收割
HETEROCYCLES, 2012, 卷号: 85, 期号: 8, 页码: 1897-1911
作者:
Li, Hui
;
Wang, Jin-Ping
;
Yang, Fan
;
Liu, Ting
;
Qiu, Wen-Wei
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
PTP1B
TCPTP
Quinazolinone
Inhibition
Synthesis
SYNTHESIS AND BIOLOGICAL EVALUATION OF OLEANOLIC ACID DERIVATIVES AS NOVEL INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE 1B
期刊论文
OAI收割
HETEROCYCLES, 2012, 卷号: 85, 期号: 5, 页码: 1117-1139
作者:
Li, Hui
;
Zou, Hui
;
Gao, Lixin
;
Liu, Ting
;
Yang, Fan
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
PTP1B
TCPTP
Inhibition