中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [41]
昆明植物研究所 [9]
中国科学院大学 [3]
西双版纳热带植物园 [2]
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期刊论文 [62]
学位论文 [4]
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Discovery of betulinic acid derivatives as gut-restricted TGR5 agonists: Balancing the potency and physicochemical properties
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 144, 页码: 18
作者:
Zhuo, Ning
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/03/25
Type 2 Diabetes
TGR5 agonist
Betulinic acid
Gut-restricted
Gallbladder-filling effects
Kinetophores
New chromone derivatives bearing thiazolidine-2,4-dione moiety as potent PTP1B inhibitors: Synthesis and biological activity evaluation
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 143, 页码: 9
作者:
Zheng, Yingying
;
Lu, Li
;
Li, Mengyue
;
Xu, Dehua
;
Zhang, Laishun
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/01/26
Chromone
Thiazolidine-2
4-dione
Protein tyrosine phosphatase 1B
Inhibitors
Anxiolytic effect of antidiabetic metformin is mediated by AMPK activation in mPFC inhibitory neurons
期刊论文
OAI收割
MOLECULAR PSYCHIATRY, 2023, 页码: 11
作者:
Zhang, Yong-mei
;
Zong, Hai-chao
;
Qi, Ying-bei
;
Chang, Liu-liu
;
Gao, Ya-nan
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/12/08
Diversity-oriented synthesis of marine polybrominated diphenyl ethers as potential KCNQ potassium channel activators
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 126, 页码: 105909
作者:
Liu, Lai-Xin
;
Gu, Ru-Rong
;
Jin, Yang
;
Chen, Xue-Qin
;
Li, Xu-Wen
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/03/21
Marine Natural product
Polybrominated diphenyl ethers
KCNQ potassium channel
Tinospora cordifolia (Willd.) Miers: Protection mechanisms and strategies against oxidative stress-related diseases
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2022, 卷号: 283, 页码: 114540
作者:
Arunachalm,Karuppusamy
;
Yang,Xuefei
;
San,Thae Thae
  |  
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2022/04/02
Tinospora cordifolia
Traditional medicine
Antioxidant
Reactive oxygen species
Immunomodulatory effect
COVID-19
CLERODANE FURANO-DITERPENE
INDIAN MEDICINAL-PLANTS
IN-VITRO ANTIOXIDANT
EX HOOK F
FREE-RADICALS
LIPID-PEROXIDATION
ETHANOLIC EXTRACT
AYURVEDIC FORMULATION
ALCOHOLIC EXTRACT
CARDIOPROTECTIVE ACTIVITY
Identification of Betulinic Acid Derivatives as Potent TGR5 Agonists with Antidiabetic Effects via Humanized TGR5(H88Y) Mutant Mice
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12181-12199
作者:
Yun, Ying
;
Zhang, Chenlu
;
Guo, Shimeng
;
Liang, Xiaoying
;
Lan, Yuan
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2021/11/04
滇牡丹降血糖活性成分的比较分析和挖掘
学位论文
OAI收割
2021
作者:
黄骞
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/03/20
A novel GPR120-selective agonist promotes insulin secretion and improves chronic inflammation
期刊论文
OAI收割
LIFE SCIENCES, 2021, 卷号: 269, 页码: 8
作者:
Yang, Liu
;
Lei, Xian-Tao
;
Huang, Qi
;
Wang, Ting
;
Sun, Hong-Bin
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2021/05/24
GPR120 agonist
Insulin secretion
Anti-inflammation
Insulin resistance
Type 2 diabetes mellitus
Diarylheptanoid-flavanone Hybrids as Multiple-target Antidiabetic Agents from Alpinia katsumadai
期刊论文
OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2021, 卷号: 39, 期号: 11, 页码: 3051-3063
作者:
He,Xiao-Feng
;
Chen,Ji-Jun
;
Li,Tian-Ze
;
Hu,Jing
;
Huang,Xiao-Yan
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2022/04/02
Alpinia katsumadai
Katsumadainols B-1-B-15
Natural products
Structure elucidation
Biological activity
TYROSINE-PHOSPHATASE 1B
GLYCOGEN-PHOSPHORYLASE
ALPHA-GLUCOSIDASE
ABSOLUTE-CONFIGURATION
STRUCTURE ELUCIDATION
DUAL INHIBITION
SEEDS
CONSTITUENT
DERIVATIVES
CHALCONE
Chemical profiling and antidiabetic potency of Paeonia delavayi: Comparison between different parts and constituents
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2021, 卷号: 198, 页码: 113998
作者:
Huang,Qian
;
Chen,Ji-Jun
;
Pan,Yang
;
He,Xiao-Feng
;
Wang,Yuan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2022/04/02
Paeonia delavayi
Chemical comparison
LCMS analyses
Antidiabetic effects
PTP1B/TCPTP selective inhibitors
LIQUID-CHROMATOGRAPHY
MULTIPLE CONSTITUENTS
RAPID IDENTIFICATION
GLYCOSIDES
ROOT
DERIVATIVES
TARGETS
CAPSULE
L.