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Chinese Academy of Sciences Institutional Repositories Grid
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Selective FRET nano probe based on carbon dots and naphthalimide-isatin for the ratiometric detection of peroxynitrite in drug-induced liver injury
期刊论文
OAI收割
CHEMICAL SCIENCE, 2024, 卷号: 15, 期号: 2, 页码: 757-764
作者:
Wu, Yueci
;
Sun, Lu-Lu
;
Han, Hai-Hao
;
He, Xiao-Peng
;
Cao, Weiguo
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/01/26
Discovery of novel triazine derivatives as potent retinoic acid receptor-related orphan receptor gamma t (ROR gamma t) inverse agonists
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 256, 页码: 18
作者:
Lu, Lixue
;
Chen, Song
;
Yu, Mingcheng
;
Zhou, Ronghui
;
Guo, Siqi
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/10/17
ROR gamma t
Triazines
Inverse agonist
Psoriasis
Autoimmune diseases
Optimization of carbazole carboxamide RORγt agonists: Challenges in improving the metabolic stability and maintaining the agonistic activity
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 251, 页码: 115213
作者:
Sun, Nannan
;
Yu, Mingcheng
;
Jiang, Zhengyuan
;
Yang, Feng
;
Lu, Lixue
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/03/27
ROR?t agonists
Carbazole carboxamide
Agonistic activity
Metabolic stability
Co-crystallization
Molecular docking
Discovery and mechanism of action of Thonzonium bromide from an FDA-approved drug library with potent and broad-spectrum inhibitory activity against main proteases of human coronaviruses
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 130, 页码: 11
作者:
Wang, Ruyu
;
Zhai, Guanglei
;
Zhu, Guanghao
;
Wang, Mengge
;
Gong, Xiaoyi
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/04/10
SARS-CoV-23CLpro
Thonzonium bromide
Mechanism of action
Broad-spectrum inhibitor
Accurate photoactivation monitoring via the construction of an intramolecular synergistic counteracting mechanism of FRET and IFE
期刊论文
OAI收割
CHEMICAL COMMUNICATIONS, 2023, 卷号: 59, 期号: 37, 页码: 5599
作者:
Ma, Siyue
;
Wang, Yihan
;
Wang, Chao
;
Wang, Linlin
;
Miao, Qing
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2023/12/01
Recent progress in assays for GPCR drug discovery
期刊论文
OAI收割
AMERICAN JOURNAL OF PHYSIOLOGY-CELL PHYSIOLOGY, 2022, 卷号: 323, 期号: 2, 页码: C583-C594
作者:
Guo, Shimeng
;
Zhao, Tingting
;
Yun, Ying
;
Xie, Xin
  |  
收藏
  |  
浏览/下载:10/0
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提交时间:2023/04/10
biased signaling
GPCR
high -throughput screening assays
humanized mouse model
protein
protein interaction
Forster and nanometal surface-energy transfer in CsPbCl3/Yb3+ quantum-cutting multilayer structures
期刊论文
OAI收割
Physical Chemistry Chemical Physics, 2022, 卷号: 24, 期号: 48, 页码: 29902-29908
作者:
C. X. Liu
;
J. S. Zhang
;
Y. Y. Chen
;
L. J. Wang
;
Y. Song and L. J. Wang
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2023/06/14
Manipulating the Injected Energy Flux via Host-Sensitized Nanostructure for Improving Multiphoton Upconversion Luminescence of Tm3+
期刊论文
OAI收割
Nano Letters, 2022, 页码: 9
作者:
X. Y. Xie
;
Q. Q. Li
;
H. R. Chen
;
W. Wang
;
F. X. Wu
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2023/06/14
A homogeneous time-resolved fluorometric energy transfer assay for the binding assessment of FcRn with IgG antibodies
期刊论文
OAI收割
JOURNAL OF IMMUNOLOGICAL METHODS, 2021, 卷号: 499, 页码: 6
作者:
Song, Yakai
;
Deng, Xiaojie
;
Shi, Wei
;
Tang, Feng
;
Huang, Wei
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/01/04
FcRn
TR-FRET
mAb
ADC
Pharmacokinetics
Botulinum toxin as an ultrasensitive reporter for bacterial and SARS-CoV-2 nucleic acid diagnostics
期刊论文
OAI收割
BIOSENSORS & BIOELECTRONICS, 2021, 卷号: 176, 页码: 8
作者:
Song, Fengge
;
Shen, Yuanyuan
;
Wei, Yangdao
;
Yang, Chunrong
;
Ge, Xiaolin
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2021/04/14
Bacterial diagnostic
SARS-CoV-2
Botulinum toxin
Fluorescence resonance energy transfer
Colorimetric detection
Biosensors