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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [73]
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OAI收割 [73]
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期刊论文 [71]
会议论文 [2]
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2024 [2]
2023 [3]
2022 [5]
2021 [3]
2020 [4]
2019 [2]
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专题:上海药物研究所
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Novel imidazo[1,2,4] triazole derivatives: Synthesis, fluorescence, bioactivity for SHP1
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 15
作者:
Yan, Xue
;
Zhang, Chun
;
Gao, Li-Xin
;
Liu, Min -Min
;
Yang, Yu-Ting
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/02/27
Imidazo[124] triazole derivatives
Fluorescence property
SHP1
Bioactivity
Cellular imaging
SIBP-03, a novel anti-HER3 antibody, exerts antitumor effects and synergizes with EGFR- and HER2-targeted drugs
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 10
作者:
Li, Wen-jing
;
Xie, Cheng-ying
;
Zhu, Xi
;
Tang, Jiao
;
Wang, Lei
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2024/02/19
SIBP-03
HER3
HER3-targeted therapy
neuregulin 1
EGFR
HER2
Glimepiride, a novel soluble epoxide hydrolase inhibitor, protects against heart failure via increasing epoxyeicosatrienoic acids
期刊论文
OAI收割
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 2023, 卷号: 185, 页码: 13-25
作者:
Zhao, Chengcheng
;
Jiang, Xiangrui
;
Peng, Liyuan
;
Zhang, Yan
;
Li, Huihui
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/01/16
Heart failure
Hypertrophy
Epoxyeicosatrienoic acids
Soluble epoxide hydrolase
Human serum albumin-based supramolecular host-guest boronate probe for enhanced peroxynitrite sensing
期刊论文
OAI收割
ORGANIC & BIOMOLECULAR CHEMISTRY, 2023, 卷号: 21, 期号: 22, 页码: 4661-4666
作者:
Tian Jr, He
;
Guo, Chen
;
Hu, Xi-Le
;
Wang, Jing-Bo
;
Zang, Yi
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/10/17
Root-Extracted lignanamides from Limonium gmelinii (Willd.) Kuntze with a potential PTP1B inhibitory activity by regulating PI3K/AKT signaling pathway
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 132, 页码: 9
作者:
Tuohongerbieke, Amanguli
;
Liu, Liu
;
Li, Jun
;
Xin, Xuelei
;
Aisa, Haji Akber
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/10/17
Limonium gmelinii (Willd
) Kuntze
Plumbaginaceae
Lignanamides
Protein tyrosine phosphatase 1B inhibitors
PI3K
AKT Signaling Pathway
Design, synthesis, and biological evaluation of Wee1 kinase degraders
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 243, 页码: 21
作者:
Zhu, Shulei
;
Liu, Jieyu
;
Xiao, Donghuai
;
Wang, Peipei
;
Ma, Jingkun
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2022/11/11
CRBN
Wee1
PROTAC
Degradation
Predicting In Vitro and In Vivo Anti-SARS-CoV-2 Activities of Antivirals by Intracellular Bioavailability and Biochemical Activity
期刊论文
OAI收割
ACS OMEGA, 2022, 页码: 13
作者:
Zhang, Jinwen
;
He, Mingfeng
;
Xie, Qian
;
Su, Ailing
;
Yang, Kuangyang
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/04/10
Strategies of engineering nanomedicines for tumor retention
期刊论文
OAI收割
JOURNAL OF CONTROLLED RELEASE, 2022, 卷号: 346, 页码: 193-211
作者:
Qian, Xindi
;
Xu, Xiaoxuan
;
Wu, Yao
;
Wang, Jiaoying
;
Li, Jie
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2022/08/16
Nanomedicines
Tumor retention
Drug delivery
Size-enlargement
Morphology changes
Quantitative Proteomics Analysis Expands the Roles of Lysine beta-Hydroxybutyrylation Pathway in Response to Environmental beta-Hydroxybutyrate
期刊论文
OAI收割
OXIDATIVE MEDICINE AND CELLULAR LONGEVITY, 2022, 卷号: 2022, 页码: 15
作者:
Hou, Wanting
;
Liu, Guobin
;
Ren, Xuelian
;
Liu, Xianming
;
He, Lei
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2022/06/15
SAF-248,a novel PI3Kδ-selective inhibitor,potently suppresses the growth of diffuse large B-cell lymphoma
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 卷号: 43, 期号: 1, 页码: 209
作者:
Zhang Xi
;
Duan Yuting
;
Wang Yi
;
Zhao Xingdong
;
Sun Yiming
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/05/22
PI3K6
PI3K/AKT/mTOR
diffuse large B-cell lymphoma
resistance
combination therapy