中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [31]
采集方式
OAI收割 [31]
内容类型
期刊论文 [31]
发表日期
2023 [2]
2021 [2]
2020 [1]
2019 [4]
2017 [1]
2016 [2]
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Pharmacolo... [1]
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浏览/检索结果:
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专题:上海药物研究所
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Exploration of novel four-membered-heterocycle constructed peptidyl proteasome inhibitors with improved metabolic stability for cancer treatment
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 138, 页码: 22
作者:
Wang, Hanlin
;
Wu, Zhaoxiao
;
Cao, Yu
;
Gao, Lixin
;
Shao, Jiaan
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/10/17
Metabolic stability
Four-membered heterocycles
Proteasome inhibitors
Multiple myeloma
Privileged heterocycles for DNA-encoded library design and hit-to-lead optimization
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 248, 页码: 26
作者:
Wen, Xin
;
Wu, Xinyuan
;
Jin, Rui
;
Lu, Xiaojie
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/04/10
DNA Encoded library
Drug discovery
Heterocycles
Hit identification
Lead generation
Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel N-Acylhydrazone Derivatives Containing Carbazole and Aromatic Ring/Aromatic Fused Heterocycle
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 9, 页码: 3593-3607
作者:
Li Yingjun
;
Lin Ledi
;
Liu Jihong
;
Gao Lixin
;
Sheng Li
  |  
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2021/12/01
PTP1B inhibitor
carbazole
N-actylhydrazone
synthesis
molecular docking
DNA-encoded C-H functionality via photoredox-mediated hydrogen atom transformation catalysis
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 42, 页码: 4
作者:
Shan, Jinming
;
Ling, Xing
;
Liu, JiaXiang
;
Wang, Xuan
;
Lu, Xiaojie
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2021/08/17
Photoredox
Hydrogen atom transfer
N-Boc saturated heterocycle
DNA Encoded Library (DEL)
NaH Promoted One-Pot Tandem Reactions of 3-(1-Alkynyl) Chromones to Form 2-Nitrogen-Substituted Xanthones
期刊论文
OAI收割
ACS OMEGA, 2020, 卷号: 5, 期号: 22, 页码: 13454-13461
作者:
Duan, Wen-Di
;
Zhang, Yu-Fang
;
Hu, Youhong
  |  
收藏
  |  
浏览/下载:59/0
  |  
提交时间:2020/12/24
Rh(III)-Catalyzed C-H Bond Activation for the Construction of Heterocycles with sp(3)-Carbon Centers
期刊论文
OAI收割
CATALYSTS, 2019, 卷号: 9, 期号: 10, 页码: 29
作者:
Wang, Run
;
Xie, Xiong
;
Liu, Hong
;
Zhou, Yu
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2020/07/01
C-H bond activation
Rhodium(III)-based catalysts
heterocycle with sp(3) carbon centers
chirality
Green and Facile Assembly of Diverse Fused N-Heterocycles Using Gold-Catalyzed Cascade Reactions in Water
期刊论文
OAI收割
MOLECULES, 2019, 卷号: 24, 期号: 5, 页码: 30
作者:
Jia, Xiuwen
;
Li, Pinyi
;
Liu, Xiaoyan
;
Lin, Jiafu
;
Chu, Yiwen
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/07/01
amine nucleophiles
alkynoic acids
cascade reaction
gold catalysis
fused N-heterocycles
One-Pot NBS-Promoted Synthesis of Imidazoles and Thiazoles from Ethylarenes in Water
期刊论文
OAI收割
MOLECULES, 2019, 卷号: 24, 期号: 5, 页码: 13
作者:
Chen, Liang
;
Zhu, Huajian
;
Wang, Jiang
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2020/07/01
NBS
nitrogen-containing heterocycle
water
one-pot
coppercatalyzedselectivechtrifluoromethylationofacrylamideswithtmscf3
期刊论文
OAI收割
chinesechemicalletters, 2019, 卷号: 30, 期号: 5, 页码: 969
作者:
Sun Shangzheng
;
Xu Hui
;
Dai Huixiong
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2020/07/01
C–H trifluoromethylation
Copper
Acrylamides
Heterocycle
LLDT-288, a novel triptolide analogue exhibits potent antitumor activity in vitro and in vivo
期刊论文
OAI收割
BIOMEDICINE & PHARMACOTHERAPY, 2017, 卷号: 93, 页码: 1004-1009
作者:
Xu, Hongtao
;
Fan, Xiaoting
;
Zhang, Guanjun
;
Liu, Xiaoyu
;
Li, Zhihong
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/01/08
Triptolide
Natural products
Drug-resistance
CYP