中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [82]
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OAI收割 [82]
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期刊论文 [79]
会议论文 [2]
专利 [1]
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2024 [1]
2023 [10]
2022 [7]
2021 [9]
2020 [14]
2019 [5]
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专题:上海药物研究所
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Novel imidazo[1,2,4] triazole derivatives: Synthesis, fluorescence, bioactivity for SHP1
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 15
作者:
Yan, Xue
;
Zhang, Chun
;
Gao, Li-Xin
;
Liu, Min -Min
;
Yang, Yu-Ting
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/02/27
Imidazo[124] triazole derivatives
Fluorescence property
SHP1
Bioactivity
Cellular imaging
Exploring the mechanism of the PTP1B inhibitors by molecular dynamics and experimental study
期刊论文
OAI收割
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2023, 卷号: 125, 页码: 12
作者:
Zhao, Tian-Tian
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/10/17
Protein tyrosine phosphatases inhibitors
PTP1B inhibitors
Mechanism study
Molecular dynamics
Five undescribed abietane-type diterpenes of Callicarpa macrophylla
期刊论文
OAI收割
FITOTERAPIA, 2023, 卷号: 170, 页码: 10
作者:
Du, Gao-Xiang
;
Chen, Tong
;
Wang, Ge
;
Liu, Ying-Bo
;
Zheng, Liu
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/10/17
Callicarpa macrophylla
Verbenaceae
Abietane-type diterpenoids
PCSK9
Macrophypene F -J
Discovery of ARD-1676 as a Highly Potent and Orally Efficacious AR PROTAC Degrader with a Broad Activity against AR Mutants for the Treatment of AR plus Human Prostate Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 18, 页码: 13280-13303
作者:
Xiang, Weiguo
;
Zhao, Lijie
;
Han, Xin
;
Xu, Tianfeng
;
Kregel, Steven
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/12/08
A pectic polysaccharide isolated from Achyranthes bidentata is metabolized by human gut Bacteroides spp.
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2023, 卷号: 248, 页码: 14
作者:
Wen, Chang
;
Li, Tingting
;
Wang, Binqiang
;
Jin, Can
;
Li, Saijuan
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/10/17
Achyranthes bidentata
Polysaccharides
Gut microbiota
PULs
SCFAs
Photophysical Exploration of Alectinib and Rilpivirine: Insights from Theory and Experiment
期刊论文
OAI收割
MOLECULES, 2023, 卷号: 28, 期号: 16, 页码: 16
作者:
Zhang, Chun
;
Yang, Yuting
;
Gan, Suya
;
Ren, Aimin
;
Zhou, Yu-Bo
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/10/17
fluorescence imaging
Alectinib
Rilpivirine
quantum chemistry
Design, Synthesis and Evaluation of Fluorescent Properties of Benzothiazole Derivatives
期刊论文
OAI收割
CHEMPHYSCHEM, 2023, 页码: 13
作者:
Sun, Yi-Tao
;
Zhang, Chun
;
Gao, Li-Xin
;
Liu, Min-Min
;
Yang, Yuting
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/10/17
Chloroquine enhances the efficacy of chemotherapy drugs against acute myeloid leukemia by inactivating the autophagy pathway
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 11
作者:
Wang, Han-lin
;
Li, Jia-nan
;
Kan, Wei-juan
;
Xu, Gao-ya
;
Luo, Guang-hao
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/10/17
acute myeloid leukemia
cytarabine
daunorubicin
idarubicin
drug resistant
multi-omics
autophagy
chloroquine phosphate
Comparative Characterization of the Ginsenosides from Six Panax Herbal Extracts and Their In Vitro Rat Gut Microbial Metabolites by Advanced Liquid Chromatography-Mass Spectrometry Approaches
期刊论文
OAI收割
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2023, 卷号: 71, 期号: 24, 页码: 9391-9403
作者:
Mi, Yue-Guang
;
Xu, Xiao-Yan
;
Hong, Li-Li
;
Jiang, Mei-Ting
;
Chen, Bo-Xue
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/10/17
Panax
multicomponent characterization
quantitative assay
gut microbiota
in vitro biotransformation
liquid chromatography-massspectrometry
A study on optical properties of various hot drug molecules by 2020
期刊论文
OAI收割
NEW JOURNAL OF CHEMISTRY, 2023, 卷号: 47, 期号: 21, 页码: 10046-10060
作者:
Zhang, Chun
;
Yang, Yuting
;
Yan, Xue
;
Sun, Yi-Tao
;
Shao, Andong
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/10/17