中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [14]
采集方式
OAI收割 [14]
内容类型
期刊论文 [14]
发表日期
2023 [1]
2022 [2]
2020 [1]
2019 [2]
2018 [1]
2017 [2]
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专题:上海药物研究所
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Five New Diarylbutyrolactones and Sesquilignans from Saussurea medusa and Their Inhibitory Effects on LPS-induced NO Production
期刊论文
OAI收割
PLANTA MEDICA, 2023, 页码: 11
作者:
Cao, Jing-Ya
;
Wang, Zhi-Yao
;
Stewart, Alan J. J.
;
Dong, Qi
;
Zhao, Ye
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/04/10
Saussurea medusa
Asteraceae
diarylbutyrolactone lignan
sesquilignan
anti-inflammatory activity
molecular docking
Megastigmane sesquiterpenoids from Saussurea medusa and their anti-inflammatory activities
期刊论文
OAI收割
NATURAL PRODUCT RESEARCH, 2022, 页码: 9
作者:
Cao, Jing-Ya
;
Dong, Qi
;
Wang, Zhi-Yao
;
Zhao, Ye
;
Ren, Yu
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/04/10
Saussurea medusa
megastigmane
sesquiterpenoid
anti-inflammatory activity
iNOS enzyme
Safety, tolerability, and pharmacokinetics of VV116, an oral nucleoside analog against SARS-CoV-2, in Chinese healthy subjects
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 9
作者:
Qian, Hong-jie
;
Wang, Yu
;
Zhang, Meng-qi
;
Xie, Yuan-chao
;
Wu, Qing-qing
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/06/15
VV116
nucleoside analog
SARS-CoV-2
safety
pharmacokinetics
healthy subjects
The artemisinin analog SM934 alleviates dry eye disease in rodent models by regulating TLR4/NF-kappa B/NLRP3 signaling
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:
Yang, Fang-ming
;
Fan, Di
;
Yang, Xiao-qian
;
Zhu, Feng-hua
;
Shao, Mei-juan
  |  
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2020/12/24
dry eye disease
artemisinin derivative
beta-aminoarteether maleate
inflammation
macrophages
TLR4
inflammasome
Structure-Based Discovery and Development of a Series of Potent and Selective Bromodomain and Extra-Terminal Protein Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 18, 页码: 8642-8663
作者:
Hu, Jianping
;
Tian, Chang-Qing
;
Damaneh, Mohammadali Soleimani
;
Li, Yanlian
;
Cao, Danyan
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2020/07/01
Enhanced Delivery of Imatinib into Vaginal Mucosa via a New Positively Charged Nanocrystal-Loaded in Situ Hydrogel Formulation for Treatment of Cervical Cancer
期刊论文
OAI收割
PHARMACEUTICS, 2019, 卷号: 11, 期号: 1, 页码: 16
作者:
Ci, Li-qian
;
Huang, Zhi-gang
;
Lv, Feng-mei
;
Wang, Jun
;
Feng, Ling-lin
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2020/07/01
mucoadhesiveness
cervicovaginal tumors
cationic functionalization
imatinib
nanocrystals
in situ hydrogel
Green Quantification Strategy Combined with Chemometric Analysis for Triglycerides in Seeds Used in Traditional Chinese Medicine
期刊论文
OAI收割
PLANTA MEDICA, 2018, 卷号: 84, 期号: 6-7, 页码: 457-464
作者:
Hou, Jin-Jun
;
Guo, Ji-ling
;
Cao, Chun-Mei
;
Yao, Shuai
;
Long, Hua-li
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
triglycerides
single standard to determine multicomponents
Coix lacryma-jobi var. ma-yuen
Poaceae
triolein
core-shell
chemometrics
Design, Synthesis, and Biological Evaluation of the First c-Met/HDAC Inhibitors Based on Pyridazinone Derivatives
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 8, 期号: 8, 页码: 830-834
作者:
Lu, Dong
;
Yan, Juan
;
Wang, Lang
;
Liu, Hongchun
;
Zeng, Limin
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2019/01/08
Dual c-Met/HDAC inhibitor
hybrid
designed multiple ligand (DML)
Pyrazolopyrimidines as Potent Stimulators for Transient Receptor Potential Canonical 3/6/7 Channels
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 11, 页码: 4680-4692
作者:
Qu, Chunrong
;
Ding, Mingmin
;
Zhu, Yingmin
;
Lu, Yungang
;
Du, Juan
  |  
收藏
  |  
浏览/下载:89/0
  |  
提交时间:2019/01/08
Bacillus as a potential diagnostic marker for yellow tongue coating
期刊论文
OAI收割
SCIENTIFIC REPORTS, 2016, 卷号: 6
作者:
Ye, Juan
;
Cai, Xueting
;
Yang, Jie
;
Sun, Xiaoyan
;
Hu, Chunping
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/01/08