中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [459]
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Ent-labdane-type diterpene glycosides obtained from Rubus chingii Hu and their inhibitory effects on PDE5A activity 期刊论文  OAI收割
FITOTERAPIA, 2024, 卷号: 173, 页码: 14
作者:  
Yu, Jun-dong;  Wang, Jing-Yi;  Liu, Jia-yuan;  Xu, Ye-chun;  Zhang, Xue
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/02/27
Novel imidazo[1,2,4] triazole derivatives: Synthesis, fluorescence, bioactivity for SHP1 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 15
作者:  
Yan, Xue;  Zhang, Chun;  Gao, Li-Xin;  Liu, Min -Min;  Yang, Yu-Ting
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/02/27
Revisiting the Role of Valeric Acid in Manipulating Ulcerative Colitis 期刊论文  OAI收割
INFLAMMATORY BOWEL DISEASES, 2024, 页码: 12
作者:  
Liu, Moting;  Zhang, Yao;  Liu, Jia;  Xiang, Caigui;  Lu, Qiukai
  |  收藏  |  浏览/下载:6/0  |  提交时间:2024/02/19
Discovery of 5-trifluoromethyl-2-aminopyrimidine derivatives as potent dual inhibitors of FLT3 and CHK1 期刊论文  OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 14
作者:  
Deng, Minjie;  Gao, Yue;  Wang, Peipei;  Du, Wenjing;  Xu, Gaoya
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/02/19
Discovery of JN122, a Spiroindoline-Containing Molecule that Inhibits MDM2/p53 Protein-Protein Interaction and Exerts Robust In Vivo Antitumor Efficacy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 24, 页码: 16991-17025
作者:  
Cheng, Jing;  Yan, Ziqin;  Jiang, Kailong;  Liu, Chen;  Xu, Dehua
  |  收藏  |  浏览/下载:5/0  |  提交时间:2024/02/19
The claustrum-prelimbic cortex circuit through dynorphin/κ-opioid receptor signaling underlies depression-like behaviors associated with social stress etiology 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 17
作者:  
Wang, Yu-Jun;  Zan, Gui-Ying;  Xu, Cenglin;  Li, Xue-Ping;  Shu, Xuelian
  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/02/19
Design, synthesis and biological evaluation of 2-aminopyrimidine derivatives as potent FLT3 inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 96, 页码: 5
作者:  
Lian, Xuanmin;  Gao, Yue;  Li, Xuemei;  Wang, Peipei;  Tong, Lexian
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/12/11
Discovery of PVD-06 as a Subtype-Selective and Efficient PTPN2 Degrader 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 22, 页码: 15269-15287
作者:  
Hu, Linghao;  Li, Huiyun;  Qin, Junlin;  Yang, Dan;  Liu, Jieming
  |  收藏  |  浏览/下载:20/0  |  提交时间:2024/02/27
ABPP-CoDEL: Activity-Based Proteome Profiling-Guided Discovery of Tyrosine-Targeting Covalent Inhibitors from DNA-Encoded Libraries 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2023, 卷号: 145, 期号: 46, 页码: 25283-25292
作者:  
Jiang, Lulu;  Liu, Sixiu;  Jia, Xinglong;  Gong, Qinting;  Wen, Xin
  |  收藏  |  浏览/下载:24/0  |  提交时间:2024/01/16
Anxiolytic effect of antidiabetic metformin is mediated by AMPK activation in mPFC inhibitory neurons 期刊论文  OAI收割
MOLECULAR PSYCHIATRY, 2023, 页码: 11
作者:  
Zhang, Yong-mei;  Zong, Hai-chao;  Qi, Ying-bei;  Chang, Liu-liu;  Gao, Ya-nan
  |  收藏  |  浏览/下载:10/0  |  提交时间:2023/12/08