中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [19]
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Identification of [1,2,4]Triazolo[4,3-a]pyrazine PARP1 inhibitors with overcome acquired resistance activities 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 19
作者:  
Wang, Pingyuan;  Zhu, Wen-Ting;  Wang, Yajing;  Song, Shan-Shan;  Xi, Yong
  |  收藏  |  浏览/下载:58/0  |  提交时间:2023/10/17
Structure-Activity Relationship Study of 1H-Pyrrole-3-carbonitrile Derivatives as STING Receptor Agonists 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2023, 页码: 9
作者:  
Shen, Chang;  Xu, Peijia;  Zhang, Changfa;  Su, Zhaoming;  Shan, Bin
  |  收藏  |  浏览/下载:24/0  |  提交时间:2023/10/17
Design, Synthesis, and Biological Evaluation of Bipyridazine Derivatives as Stimulator of Interferon Genes (STING) Receptor Agonists 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 5, 页码: 3327-3347
作者:  
Shan, Bin;  Hou, Hui;  Zhang, Keke;  Li, Rui;  Shen, Chang
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/03/27
Thioparib inhibits homologous recombination repair, activates the type I IFN response, and overcomes olaparib resistance 期刊论文  OAI收割
EMBO MOLECULAR MEDICINE, 2023, 页码: 24
作者:  
Wang, Li-Min;  Wang, Pingyuan;  Chen, Xiao-Min;  Yang, Hui;  Song, Shan-Shan
  |  收藏  |  浏览/下载:21/0  |  提交时间:2023/04/10
Identification of HGD and GSTZ1 as Biomarkers Involved Metabolic Reprogramming in Kidney Renal Clear Cell Carcinoma 期刊论文  OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2022, 卷号: 23, 期号: 9, 页码: 14
作者:  
Wang, Jiyan;  Chang, Hongkai;  Su, Meng;  Qiao, Yaya;  Sun, Huanran
  |  收藏  |  浏览/下载:16/0  |  提交时间:2022/08/16
Optimization of Brigatinib as New Wild-Type Sparing Inhibitors of EGFR(T790M/C797S) Mutants 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2022, 页码: 7
作者:  
Li, Shan;  Zhang, Tao;  Zhu, Su-Jie;  Lei, Chong;  Lai, Mengzhen
  |  收藏  |  浏览/下载:25/0  |  提交时间:2022/06/15
Anti-SARS-CoV-2 activities in vitro of Shuanghuanglian preparations and bioactive ingredients 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:  
Su, Hai-xia;  Yao, Sheng;  Zhao, Wen-feng;  Li, Min-jun;  Liu, Jia
  |  收藏  |  浏览/下载:62/0  |  提交时间:2020/12/24
Poly(ADP-ribose)polymerase (PARP) inhibition and anticancer activity of simmiparib, a new inhibitor undergoing clinical trials 期刊论文  OAI收割
CANCER LETTERS, 2017, 卷号: 386, 页码: 47-56
作者:  
Yuan, Bo;  Ye, Na;  Song, Shan-Shan;  Wang, Yu-Ting;  Song, Zilan
  |  收藏  |  浏览/下载:43/0  |  提交时间:2019/01/08
Novel PARP1/2 inhibitor mefuparib hydrochloride elicits potent in vitro and in vivo anticancer activity, characteristic of high tissue distribution 期刊论文  OAI收割
ONCOTARGET, 2017, 卷号: 8, 期号: 3, 页码: 4156-4168
作者:  
He, Jin-Xue;  Wang, Meng;  Huan, Xia-Juan;  Chen, Chuan-Huizi;  Song, Shan-Shan
  |  收藏  |  浏览/下载:35/0  |  提交时间:2019/01/08
Dual pH-sensitive micelles with charge-switch for controlling cellular uptake and drug release to treat metastatic breast cancer 期刊论文  OAI收割
BIOMATERIALS, 2017, 卷号: 114, 页码: 44-53
作者:  
Tang, Shan;  Meng, Qingshuo;  Sun, Huiping;  Su, Jinghan;  Yin, Qi
  |  收藏  |  浏览/下载:37/0  |  提交时间:2019/01/08