中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [12]
采集方式
OAI收割 [12]
内容类型
期刊论文 [12]
发表日期
2020 [1]
2016 [1]
2015 [2]
2014 [3]
2012 [3]
2009 [2]
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专题:上海药物研究所
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Design, Synthesis, and In Vitro Evaluation of Benzofuro[3,2-c]Quinoline Derivatives as Potential Antileukemia Agents
期刊论文
OAI收割
MOLECULES, 2020, 卷号: 25, 期号: 1, 页码: 13
作者:
Lin, Ying
;
Xing, Dong
;
Wu, Wen-Biao
;
Xu, Gao-Ya
;
Yu, Li-Fang
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2020/07/01
benzofuro[3,2-c]quinolines
3-(2-methoxyphenyl)quinolin-4(1H)one
MV-4-11 cell line
antileukemia activity
Effect of a hepatitis B virus inhibitor, NZ-4, on capsid formation
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2016, 卷号: 125, 页码: 25-33
作者:
Yang, Li
;
Wang, Ya-Juan
;
Chen, Hai Jun
;
Shi, Li-Ping
;
Tong, Xian-Kun
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/01/08
Anti-hepatitis B virus compound
Capsid formation
pgRNA packaging
Arg-rich domain I
Faster-migrating capsid
2-(3-Benzoylthioureido)-4,5,6,7-tetrahydrobenzo[b] thiophene-3-carboxylic acid ameliorates metabolic disorders in high-fat diet-fed mice
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2015, 卷号: 36, 期号: 4, 页码: 483-496
作者:
Zhang, Jin
;
Zhang, Li-na
;
Chen, Dong-mei
;
Fu, Yan-yun
;
Zhang, Feng
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2019/01/08
2-(3-benzoylthioureido)-4,5,6,7-tetrahydrobenzo[b] thiophene-3-carboxylic acid
lipogenesis
SREBP-1c
AMPK
mTOR
hepatic lipid accumulation
obesity
metabolic disorders
Platycodin D triggers autophagy through activation of extracellular signal-regulated kinase in hepatocellular carcinoma HepG2 cells
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACOLOGY, 2015, 卷号: 749, 页码: 81-88
作者:
Li, Ting
;
Tang, Zheng-Hai
;
Xu, Wen-Shan
;
Wu, Guo-Sheng
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
Platycodin D
Auto phagy
ERK
Chloroquine
Protective
HepG2
Design and discovery of flavonoid-based HIV-1 integrase inhibitors targeting both the active site and the interaction with LEDGF/p75
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2014, 卷号: 22, 期号: 12, 页码: 3146-3158
作者:
Li, Bo-Wen
;
Zhang, Feng-Hua
;
Serrao, Erik
;
Chen, Huan
;
Sanchez, Tino W.
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
HIV-1 integrase inhibitors
Flavonoid
Chelation
Strand transfer
LEDGF/p75
Synthesis and biological evaluation of novel bis-aromatic amides as novel PTP1B inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 8, 页码: 1889-1894
作者:
Wang, Wen-Long
;
Huang, Chao
;
Gao, Li-Xin
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/01/08
Bis-aromatic amides
PTP1B inhibitors
Selectivity
Cellular activity
Structure-activity relationships (SARs)
1H-2,3-Dihydroperimidine Derivatives: A New Class of Potent Protein Tyrosine Phosphatase 1B Inhibitors
期刊论文
OAI收割
MOLECULES, 2014, 卷号: 19, 期号: 1, 页码: 102-121
作者:
Wang, Wen-Long
;
Yang, Dong-Lin
;
Gao, Li-Xin
;
Tang, Chun-Lan
;
Ma, Wei-Ping
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
1H-2,3-dihydroperimidine derivatives
PTP1B
inhibitors
selectivity
structure-activity relationships (SAR)
Synthesis and biological evaluation of 4,4-dimethyl lithocholic acid derivatives as novel inhibitors of protein tyrosine phosphatase 1B
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 卷号: 22, 期号: 23, 页码: 7237-7242
作者:
He, Hai-Bing
;
Gao, Li-Xin
;
Deng, Qi-Feng
;
Ma, Wei-Ping
;
Tang, Chun-Lan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
4,4-Dimethyl lithocholic acids
Protein tyrosine phosphatase 1B
Inhibitor
SAR
Diabetes
DESIGN, SYNTHESIS AND BIOLOGICAL ACTIVITY EVALUATION OF 2,5-DIPHENYL-1,3,4-OXADIAZOLE DERIVATIVES AS NOVEL INHIBITORS OF FRUCTOSE-1,6-BISPHOSPHATASE
期刊论文
OAI收割
HETEROCYCLES, 2012, 卷号: 85, 期号: 11, 页码: 2693-2712
作者:
He, Hai-Bing
;
Gao, Li-Xin
;
Zhou, Yue-Yang
;
Liu, Ting
;
Tang, Jie
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
Fructose-1,6-bisphosphatase
2,5-Phenyl-1,3,4-oxadiazole
Type-2 Diabetes
Enzyme Inhibition
DESIGN, SYNTHESIS AND BIOLOGICAL ACTIVITY EVALUATION OF 2-MERCAPTO-4(3H)-QUINAZOLINONE DERIVATIVES AS NOVEL INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE 1B
期刊论文
OAI收割
HETEROCYCLES, 2012, 卷号: 85, 期号: 8, 页码: 1897-1911
作者:
Li, Hui
;
Wang, Jin-Ping
;
Yang, Fan
;
Liu, Ting
;
Qiu, Wen-Wei
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
PTP1B
TCPTP
Quinazolinone
Inhibition
Synthesis