中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [21]
采集方式
OAI收割 [21]
内容类型
期刊论文 [21]
发表日期
2023 [2]
2021 [1]
2020 [1]
2019 [1]
2018 [2]
2017 [1]
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浏览/检索结果:
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专题:上海药物研究所
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Exploration of novel four-membered-heterocycle constructed peptidyl proteasome inhibitors with improved metabolic stability for cancer treatment
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 138, 页码: 22
作者:
Wang, Hanlin
;
Wu, Zhaoxiao
;
Cao, Yu
;
Gao, Lixin
;
Shao, Jiaan
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/10/17
Metabolic stability
Four-membered heterocycles
Proteasome inhibitors
Multiple myeloma
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors
期刊论文
OAI收割
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1, 页码: 17-27
作者:
Zang, Yi
;
Su, Mingbo
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/03/27
high-throughput screening
SARS
CoV-2
main
papain-like
proteases
Rational Design and Development of Novel CDK9 Inhibitors for the Treatment of Acute Myeloid Leukemia
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14647-14663
作者:
Han, Xu
;
Song, Ning
;
Saidahmatov, Abdusaid
;
Wang, Peipei
;
Wang, Yong
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2021/12/16
Efficient synthesis, biological evaluation, and docking study of isatin based derivatives as caspase inhibitors
期刊论文
OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2020, 卷号: 35, 期号: 1, 页码: 1674-1684
作者:
Firoozpour, Loghman
;
Gao, Lixin
;
Moghimi, Setareh
;
Pasalar, Parvin
;
Davoodi, Jamshid
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/12/24
Caspase inhibitor
Isatin sulphonamides
docking studies
Pharmacophore
apoptosis
SNX10 (sorting nexin 10) inhibits colorectal cancer initiation and progression by controlling autophagic degradation of SRC
期刊论文
OAI收割
AUTOPHAGY, 2019, 页码: 15
作者:
Zhang, Sulin
;
Yang, Zhiwen
;
Bao, Weilian
;
Liu, Lixin
;
You, Yan
  |  
收藏
  |  
浏览/下载:94/0
  |  
提交时间:2020/07/01
Colorectal cancer
macroautophagy
SNX10
SRC
tumor growth
Pyrazolo[4,3-b]pyrimido[4,5-e][1,4]diazepine derivatives as new multi-targeted inhibitors of Aurora A/B and KDR
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 428-441
作者:
Zhang, Qiumeng
;
Shen, Qianqian
;
Gao, Lixin
;
Tong, Linjiang
;
Li, Jia
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2019/01/08
Aurora A
Aurora B
KDR
Multi-targeted
Anticancer
Heterocyclic
Enhanced doxorubicin delivery to hepatocellular carcinoma cells via CD147 antibody-conjugated immunoliposomes
期刊论文
OAI收割
NANOMEDICINE-NANOTECHNOLOGY BIOLOGY AND MEDICINE, 2018, 卷号: 14, 期号: 6, 页码: 1949-1961
作者:
Wang, Jian
;
Wu, Zhitao
;
Pan, Guoyu
;
Ni, Junsheng
;
Xie, Fangyuan
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2019/01/08
CD147
Antibody
Liposomes
Doxorubicin
Hepatocellular carcinoma
Simultaneous determination of eight B-vitamins in rat intestinal perfusate to identify effects of osmotic pressures on absorptions
期刊论文
OAI收割
BIOMEDICAL CHROMATOGRAPHY, 2017, 卷号: 31, 期号: 9
作者:
Wang, Xiaobo
;
Xiao, Jian
;
Zhou, Hui
;
Qiu, Ying
;
Peng, Hui
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
B-vitamins
HPLC-DAD
intestinal perfusate
osmotic pressures
designsynthesisandbiologicalevaluationofbiphenylureaderivativesasvegfr2kinaseinhibitorsii
期刊论文
OAI收割
chinesechemicalletters, 2016, 卷号: 27, 期号: 2, 页码: 200
作者:
Gao Guorui
;
Li Mengyuan
;
Lv Yongcong
;
Cao Sufen
;
Tong Linjiang
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2020/07/01
GROWTH-FACTOR RECEPTOR-2
POTENT
ANGIOGENESIS
DISCOVERY
SORAFENIB
TOXICITY
CANCER
Angiogenesis
Kinase
Inhibitor
VEGFR-2
dw10075anovelselectiveandsmallmoleculeinhibitorofvegfrexhibitsantitumoractivitiesbothinvitroandinvivo
期刊论文
OAI收割
actapharmacologicasinica, 2016, 卷号: 37, 期号: 3, 页码: 398
作者:
Ll Mengyuan
;
Lv Yongcong
;
Tong Linjiang
;
Peng Ting
;
Qu Rong
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/07/01
DW10075
VEGF/VEGF receptor inhibitor
Antitumor
Angiogenesis
U87-MG human glioblastoma