中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [41]
采集方式
OAI收割 [41]
内容类型
期刊论文 [41]
发表日期
2024 [2]
2023 [3]
2022 [5]
2021 [3]
2020 [2]
2019 [2]
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浏览/检索结果:
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专题:上海药物研究所
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Ent-labdane-type diterpene glycosides obtained from
Rubus
chingii
Hu and their inhibitory effects on PDE5A activity
期刊论文
OAI收割
FITOTERAPIA, 2024, 卷号: 173, 页码: 14
作者:
Yu, Jun-dong
;
Wang, Jing-Yi
;
Liu, Jia-yuan
;
Xu, Ye-chun
;
Zhang, Xue
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/02/27
diterpene glycosides
Rubus Chingii Hu
PDE5A inhibitory activity
ent-labdane
Pharmacologically significant constituents collectively responsible for anti-sepsis action of XueBiJing, a Chinese herb-based intravenous formulation
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 16
作者:
Cheng, Chen
;
Ren, Chao
;
Li, Mu-zi
;
Liu, Yi-hui
;
Yao, Ren-qi
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/02/27
Traditional Chinese medicine
XueBiJing
sepsis
mortality
pharmacokinetic compatibility
polypharmacology
A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:
Yang, Xin-Mei
;
Yang, Yang
;
Yao, Bu-Fan
;
Ye, Pan-Pan
;
Xu, Yan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/11
COVID-19
Simnotrelvir
Safety
Pharmacokinetics
Healthy subjects
Design, Synthesis and Evaluation of Fluorescent Properties of Benzothiazole Derivatives
期刊论文
OAI收割
CHEMPHYSCHEM, 2023, 页码: 13
作者:
Sun, Yi-Tao
;
Zhang, Chun
;
Gao, Li-Xin
;
Liu, Min-Min
;
Yang, Yuting
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/10/17
A study on optical properties of various hot drug molecules by 2020
期刊论文
OAI收割
NEW JOURNAL OF CHEMISTRY, 2023, 卷号: 47, 期号: 21, 页码: 10046-10060
作者:
Zhang, Chun
;
Yang, Yuting
;
Yan, Xue
;
Sun, Yi-Tao
;
Shao, Andong
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/10/17
Targeting UHRF1-SAP30-MXD4 axis for leukemia initiating cell eradication in myeloid leukemia
期刊论文
OAI收割
CELL RESEARCH, 2022, 页码: 19
作者:
Hu, Cheng-Long
;
Chen, Bing-Yi
;
Li, Zijuan
;
Yang, Tianbiao
;
Xu, Chun-Hui
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/12/13
Absorption, distribution, metabolism, and excretion of [C-14]Mefuparib (CVL218), a novel PARP1/2 inhibitor, in rats
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2022, 页码: 12
作者:
Li, Xin-mei
;
Zheng, Yuan-dong
;
Zhang, Yi-fan
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/12/13
[C-14]Mefuparib
Mefuparib (CVL218)
Blood-brain barrier
Mass balance
Tissue distribution
GastroPlus simulation
Deletion of Schizophrenia Susceptibility Gene Ulk4 Leads to Abnormal Cognitive Behaviors via Akt-GSK-3 Signaling Pathway in Mice
期刊论文
OAI收割
SCHIZOPHRENIA BULLETIN, 2022, 页码: 10
作者:
Hu, Ling
;
Zhou, Bing-Yao
;
Yang, Cui-Ping
;
Lu, Da-Yun
;
Tao, Yun-Chao
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/06/15
Unc-51-like kinase 4
schizophrenia
sensorimotor gating
Akt
GSK-3
cerebral cortex
Synthesis and Biochemical Evaluation of 8H-Indeno[1,2-d]thiazole Derivatives as Novel SARS-CoV-2 3CL Protease Inhibitors
期刊论文
OAI收割
MOLECULES, 2022, 卷号: 27, 期号: 10, 页码: 11
作者:
Wu, Jing
;
Feng, Bo
;
Gao, Li-Xin
;
Zhang, Chun
;
Li, Jia
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/08/16
COVID-19
M-pro inhibitors
drug design and synthesis
structure-activity relationships (SAR)
Repressing MYC by targeting BET synergizes with selective inhibition of PI3K alpha against B cell lymphoma
期刊论文
OAI收割
CANCER LETTERS, 2022, 卷号: 524, 页码: 206-218
作者:
Chen, Zi-qi
;
Cao, Zhe-rui
;
Wang, Yi
;
Zhang, Xi
;
Xu, Lan
  |  
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2021/12/16
CYH33
MYC
P300
BET
B cell lymphoma
PI3K