中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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Excessive fatty acids activate PRMT5/MDM2/Drosha pathway to regulate miRNA biogenesis and lipid metabolism
期刊论文
OAI收割
LIVER INTERNATIONAL, 2024, 页码: 17
作者:
Hou, Aijun
;
Xu, Xiaoding
;
Zhang, Yu
;
He, Hongxiu
;
Feng, Yihan
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Drosha degradation
lipid metabolism
miRNA biogenesis
NAFLD
PRMT5
Synthesis and Biological Evaluation of β-Lactam Derivatives Targeting Speckle-Type POZ Protein (SPOP)
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 15, 期号: 2, 页码: 270-279
作者:
Zhou, Chenmao
;
Hao, Xinyue
;
Chen, Zhengyang
;
Zhang, Runze
;
Zhou, Qian
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/03/13
Speckle-type POZ protein (SPOP)
SPOP inhibitors
Clear cell renal cell carcinoma (ccRCC)
Structure-activityrelationship (SAR)
Role of F-box proteins in human upper gastrointestinal tumors
期刊论文
OAI收割
BIOCHIMICA ET BIOPHYSICA ACTA-REVIEWS ON CANCER, 2024, 卷号: 1879, 期号: 1, 页码: 16
作者:
Zhang, Che
;
Pan, Guangzhao
;
Qin, Jiang-Jiang
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2024/02/27
F-box protein
Upper gastrointestinal cancer
E3 ubiquitin ligase
Ubiquitin
The new direction of drug development: Degradation of undruggable targets through targeting chimera technology
期刊论文
OAI收割
MEDICINAL RESEARCH REVIEWS, 2023, 页码: 54
作者:
Liang, Xuewu
;
Ren, Hairu
;
Han, Fengyang
;
Liang, Renwen
;
Zhao, Jiayan
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2024/01/16
chimeric design
degradation System
PROTAC
targeted degradation technology
undruggable targets
Deubiquitylating Enzymes in Cancer and Immunity
期刊论文
OAI收割
ADVANCED SCIENCE, 2023, 页码: 37
作者:
Ren, Jiang
;
Yu, Peng
;
Liu, Sijia
;
Li, Ran
;
Niu, Xin
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/12/08
cancer
deubiquitylating enzymes (DUBs)
immunity
therapeutic approach
MAVS-loaded unanchored Lys63-linked polyubiquitin chains activate the RIG-I-MAVS signaling cascade
期刊论文
OAI收割
CELLULAR & MOLECULAR IMMUNOLOGY, 2023, 页码: 17
作者:
Liu, Feng
;
Zhuang, Wanxin
;
Song, Bin
;
Yang, Yuan
;
Liu, Junqi
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/10/17
MAVS
Aggregation
Unanchored K63-linked polyubiquitin chains
RIG-I
USP10
Selective degradation of cellular BRD3 and BRD4-L promoted by PROTAC molecules in six cancer cell lines
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 254, 页码: 17
作者:
Yan, Ziqin
;
Lyu, Xilin
;
Lin, Dongze
;
Wu, Gaoxing
;
Gong, Yang
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2023/10/17
Stimuli-activatable PROTACs for precise protein degradation and cancer therapy
期刊论文
OAI收割
SCIENCE BULLETIN, 2023, 卷号: 68, 期号: 10, 页码: 1069-1085
作者:
Gao, Jing
;
Yang, Lei
;
Lei, Shumin
;
Zhou, Feng
;
Nie, Huijun
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/10/17
PROTAC
Stimuli-activatable prodrug
Precise protein degradation
Nanomedicine
Combinatory therapy
Goliath induces inflammation in obese mice by linking fatty acid β-oxidation to glycolysis
期刊论文
OAI收割
EMBO REPORTS, 2023, 卷号: 24, 期号: 4
作者:
Hao, Shumeng
;
Zhang, Sulin
;
Ye, Jialin
;
Chen, Lifan
;
Wang, Yan
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/03/27
FAO
glycolysis
Goliath
inflammation
obesity
E3 ligase ligand optimization of Clinical PROTACs
期刊论文
OAI收割
FRONTIERS IN CHEMISTRY, 2023, 卷号: 11, 页码: 15
作者:
Jiang, Hanrui
;
Xiong, Huan
;
Gu, Shuang-Xi
;
Wang, Mingliang
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/04/10
PROTACs
E3 ubiquitin ligase ligand
structure optimization
clinical trials
CRBN