中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共889条,第1-10条 帮助

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Worm-like micelles facilitate the intestinal mucus diffusion and drug accumulation for enhancing colorectal cancer therapy 期刊论文  OAI收割
Chinese Chemical Letters, 2024, 卷号: 35, 期号: 6, 页码: 108967
作者:  
Zhou, Yihan;  Gao, Duo;  Wang, Yaying;  Liang, Li;  Zhang, Qingyu
  |  收藏  |  浏览/下载:25/0  |  提交时间:2024/03/26
Structure-based discovery of a new series of nucleoside-derived ring-opening PRMT5 inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 267, 页码: 19
作者:  
Chen, Yuting;  Wang, Zekun;  Zhang, Junjie;  Shi, Qiongyu;  Yang, Hong
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/07
Discovery of Pyrido[2,3-d]pyrimidin-7-one Derivatives as Highly Potent and Efficacious Ectonucleotide Pyrophosphatase/Phosphodiesterase 1 (ENPP1) Inhibitors for Cancer Treatment 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 5, 页码: 3986-4006
作者:  
Sun, Yaoliang;  Chen, Manman;  Han, Yuyan;  Li, Weiqiang;  Ma, Xiaoyu
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/07
Development of Potent MALT1 Inhibitors Featuring a Novel "2-Thioxo-2,3-dihydrothiazolo[4,5-d]pyrimidin-7(6H)-one" Scaffold for the Treatment of B Cell Lymphoma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 4, 页码: 2884-2906
作者:  
Liang, Xuewu;  Yu, Haolan;  Liang, Renwen;  Feng, Zhuanghui;  Saidahmatov, Abdusaid
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/04/09
Regulating protein corona on nanovesicles by glycosylated polyhydroxy polymer modification for efficient drug delivery 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2024, 卷号: 15, 期号: 1, 页码: 20
作者:  
Miao, Yunqiu;  Li, Lijun;  Wang, Ying;  Wang, Jiangyue;  Zhou, Yihan
  |  收藏  |  浏览/下载:17/0  |  提交时间:2024/03/13
Discovery of a 1,6-naphthyridin-4-one-based AXL inhibitor with improved pharmacokinetics and enhanced in vivo antitumor efficacy 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 17
作者:  
Lan, Yaohan;  Peng, Xia;  Ji, Yinchun;  Su, Yi;  Duan, Wenhu
  |  收藏  |  浏览/下载:12/0  |  提交时间:2024/02/27
pH-responsive nanogels with enhanced antioxidant and antitumor activities on drug delivery and smart drug release 期刊论文  OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2024, 卷号: 257, 页码: 16
作者:  
Ma, Bing;  Li, Qing;  Mi, Yingqi;  Zhang, Jingjing;  Tan, Wenqiang
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/01/26
Discovery, Optimization, and Evaluation of Novel Pyridin-2(1H)-one Analogues as Potent TRK Inhibitors for Cancer Treatment 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1168-1183
作者:  
Xu, Zichao;  Peng, Xia;  Zhang, Renjie;  Ji, Yinchun;  You, Mengke
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/02/27
Low-Dose Chemotherapy Preferentially Shapes the Ileal Microbiome and Augments the Response to Immune Checkpoint Blockade by Activating AIM2 Inflammasome in Ileal Epithelial Cells 期刊论文  OAI收割
ADVANCED SCIENCE, 2024, 页码: 17
作者:  
Pu, Congying;  Li, Yize;  Fu, Yixian;  Yan, Yiyang;  Tao, Siyao
  |  收藏  |  浏览/下载:26/0  |  提交时间:2024/02/27
Effect of Hydrophobic Chain Length in Amphiphilic Chitosan Conjugates on Intracellular Drug Delivery and Smart Drug Release of Redox-Responsive Micelle 期刊论文  OAI收割
MARINE DRUGS, 2024, 卷号: 22, 期号: 1, 页码: 18
作者:  
Yuan, Yuting;  Tan, Wenqiang;  Mi, Yingqi;  Wang, Linqing;  Qi, Zhen
  |  收藏  |  浏览/下载:0/0  |  提交时间:2024/05/07