中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [8]
海洋研究所 [3]
新疆理化技术研究所 [2]
昆明植物研究所 [1]
中国科学院大学 [1]
合肥物质科学研究院 [1]
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期刊论文 [16]
学位论文 [1]
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2021 [6]
2018 [2]
2017 [1]
2015 [1]
2014 [1]
2013 [3]
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Pharmacolo... [2]
天然产物分离与分析 [1]
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Development of FABP4/5 inhibitors with potential therapeutic effect on type 2 Diabetes Mellitus
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 224, 页码: 14
作者:
He, Yu-Long
;
Chen, Meng-Ting
;
Wang, Ting
;
Zhang, Ming-Ming
;
Li, Ying-Xia
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2021/11/04
Type 2 diabetes mellitus
Dual FABP4/5 inhibitors
Anti-lipolytic and anti-inflammatory effects
Metabolic stability
Anti-diabetic activities
Novel tetrahydrobenzo[b]thiophen-2-yl)urea derivatives as novel alpha-glucosidase inhibitors: Synthesis, kinetics study, molecular docking, and in vivo anti-hyperglycemic evaluation
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 115, 页码: 17
作者:
Xie, Hong-Xu
;
Zhang, Juan
;
Li, Yue
;
Zhang, Jin-He
;
Liu, Shan-Kui
  |  
收藏
  |  
浏览/下载:81/0
  |  
提交时间:2021/11/04
Tetrahydrobenzo[b]thiophen-2-yl)urea
alpha-Glucosidase inhibitors
Non-competitive inhibitor
Molecular docking
Anti-hyperglycaemic activity
Type 2 diabetes
A novel GPR120-selective agonist promotes insulin secretion and improves chronic inflammation
期刊论文
OAI收割
LIFE SCIENCES, 2021, 卷号: 269, 页码: 8
作者:
Yang, Liu
;
Lei, Xian-Tao
;
Huang, Qi
;
Wang, Ting
;
Sun, Hong-Bin
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2021/05/24
GPR120 agonist
Insulin secretion
Anti-inflammation
Insulin resistance
Type 2 diabetes mellitus
Discovery of 5-(3-bromo-2-(2,3-dibromo-4,5-dimethoxybenzyl)-4,5-dimethoxybenzylidene)thiazolidine-2,4-dione as a novel potent protein tyrosine phosphatase 1B inhibitor with antidiabetic properties
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 108, 页码: 13
作者:
Jiang, Bo
;
Luo, Jiao
;
Guo, Shuju
;
Wang, Lijun
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2021/05/11
Type 2 diabetes mellitus
Protein tyrosine phosphatase 1B inhibitors
Thiazolidinedione
Insulin signaling
Anti-diabetic activities
Dynamic folding modulation generates FGF21 variant against diabetes
期刊论文
OAI收割
EMBO REPORTS, 2021, 卷号: 22
作者:
Zhu, Lei
;
Zhao, Hongxin
;
Liu, Juanjuan
;
Cai, Hao
;
Wu, Bo
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2021/08/30
anti‐
diabetes
disulfide bond mutation
FGF21
folding dynamics
NMR
Multiple in vitro biological effects of phenolic compounds from Terminalia chebula var. tomentella
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2021, 卷号: 275, 页码: 114135
作者:
Zhang,Xiao-Rui
;
Qiao,Yi-Jun
;
Zhu,Hong-Tao
;
Kong,Qing-Hua
;
Wang,Dong
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2022/04/02
Terminalia chebula var
tomentella
Combretaceae
Fructus Chebulae
Hydrolyzed tannins
Simple phenolic compounds
Anti-inflammation
Anti-diabetes
NITRIC-OXIDE
ANTIOXIDANT
TANNINS
CONSTITUENTS
VALIDATION
ALGORITHM
ESTERS
FRUITS
Anti-diabetic Effect of Punica granatum Flower Polyphenols Extract in Type 2 Diabetic Rats: Activation of Akt/GSK-3 beta and Inhibition of IRE1 alpha-XBP1 Pathways
期刊论文
OAI收割
FRONTIERS IN ENDOCRINOLOGY, 2018, 卷号: 9
作者:
Tang, Dan
;
Liu, Liu
;
Ajiakber, Dildar
;
Ye, Jianping
;
Xu, Jianjun
  |  
收藏
  |  
浏览/下载:79/0
  |  
提交时间:2019/01/08
type 2 diabetes mellitus
Punica granatum L. flower
anti-diabetic herb
oral glucose tolerance test
endoplasmic reticulum stress
insulin resistance
Anti-diabetic effect and mechanism of Kursi Wufarikun Ziyabit in L6 rat skeletal muscle cells
期刊论文
OAI收割
JOURNAL OF PHARMACOLOGICAL SCIENCES, 2018, 卷号: 137, 期号: 2, 页码: 212-219
作者:
Edirs, S (Edirs, Salamet)[ 1,3 ]
;
Jiang, L (Jiang, Lan)[ 1,2 ]
;
Xin, XL (Xin, XueLei)[ 1,2 ]
;
Aisa, HA (Aisa, Haji Akber)[ 1,2 ]
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2018/09/27
Type 2 Diabetes
Kursi Wufarikun Ziyabit
Anti-diabetic Activity
Insulin Signaling Pathway
Endoplasmic Reticulum Stress
Anti-diabetic effect of three new norditerpenoid alkaloids in vitro and potential mechanism via PI3K/Akt signaling pathway
期刊论文
OAI收割
BIOMEDICINE & PHARMACOTHERAPY, 2017, 卷号: 87, 期号: 3, 页码: 145-152
作者:
Tang, D (Tang, Dan)
;
Chen, QB (Chen, Qi-Bin)
;
Xin, XL (Xin, Xue-Lei)
;
Aisa, HA (Aisa, Haji-Akber)
;
Aisa, HA
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2017/04/05
Diabetes
Norditerpenoid alkaloids
Anti-diabetic activity
Glucose metabolism
Protein tyrosine phosphatase 1B
PI3K/Akt signaling pathway
Anti-Diabetic Effects of Madecassic Acid and Rotundic Acid
期刊论文
OAI收割
NUTRIENTS, 2015, 卷号: 7, 期号: 12, 页码: 10065-10075
作者:
Hsu, Yuan-Man
;
Hung, Yi-chih
;
Hu, Lihong
;
Lee, Yi-ju
;
Yin, Mei-chin
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2019/01/08
madecassic acid
rotundic acid
diabetes
coagulation
anti-lipid