中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [8]
金属研究所 [2]
地理科学与资源研究所 [1]
化学研究所 [1]
大连化学物理研究所 [1]
合肥物质科学研究院 [1]
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OAI收割 [14]
内容类型
期刊论文 [14]
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2024 [2]
2020 [2]
2017 [1]
2016 [2]
2014 [2]
2009 [1]
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学科主题
Oncology [1]
Pharmacolo... [1]
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Discovery of betulinic acid derivatives as gut-restricted TGR5 agonists: Balancing the potency and physicochemical properties
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 144, 页码: 18
作者:
Zhuo, Ning
;
Yun, Ying
;
Zhang, Chenlu
;
Guo, Shimeng
;
Yin, Jianpeng
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2024/03/25
Type 2 Diabetes
TGR5 agonist
Betulinic acid
Gut-restricted
Gallbladder-filling effects
Kinetophores
Discovery and exploration of novel somatostatin receptor subtype 5 (SSTR5) antagonists for the treatment of cholesterol gallstones
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 264, 页码: 16
作者:
Han, Fanghui
;
Zhao, Tingting
;
Zhang, Yanglong
;
Yun, Ying
;
Xu, Yuanyuan
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/02/19
SSTR5 antagonist
Gallbladder emptying
Cholesterol gallstones
Survival analysis of patients with primary gallbladder cancer from 2010 to 2015 A retrospective study based on SEER data
期刊论文
OAI收割
MEDICINE, 2020, 卷号: 99, 期号: 40, 页码: 6
作者:
Zhu, Xiaolei
;
Zhang, Xiaochang
;
Hu, Xiao
;
Ren, Hongyan
;
Wu, Shenghui
  |  
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2021/03/16
primary gallbladder cancer
prognosis
survival
Design of G-protein-coupled bile acid receptor 1 (GPBAR1, TGR5) soft drugs with reduced gallbladder-filling effects
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 12
作者:
Han, Fanghui
;
Ning, Mengmeng
;
Cao, Hua
;
Ye, Yangliang
;
Feng, Ying
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/12/21
Soft drug
TGR5
GLP-1
Gallbladder-filling effects
Rapid metabolism
Carboxylic ester
Long non-coding RNA expression profiles in gallbladder carcinoma identified using microarray analysis
期刊论文
OAI收割
ONCOLOGY LETTERS, 2017, 卷号: 13, 期号: 5, 页码: 3508-3516
作者:
Wang, Jiwen
;
Liu, Han
;
Shen, Xiaokun
;
Wang, Yueqi
;
Zhang, Dexiang
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
computational biology
expression profile
gallbladder neoplasms
long non-coding RNA
gene microarray analysis
OL3, a novel low-absorbed TGR5 agonist with reduced side effects, lowered blood glucose via dual actions on TGR5 activation and DPP-4 inhibition
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 10, 页码: 1359-1369
作者:
Ma, Shan-yao
;
Ning, Meng-meng
;
Zou, Qing-an
;
Feng, Ying
;
Ye, Yang-liang
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2019/01/08
OL3
MN6
linagliptin
TGR5 agonist
DPP4 inhibitor
GLP-1
low-absorbed
gallbladder filling
type 2 diabetes mellitus
ol3anovellowabsorbedtgr5agonistwithreducedsideeffectsloweredbloodglucoseviadualactionsontgr5activationanddpp4inhibition
期刊论文
OAI收割
actapharmacologicasinica, 2016, 卷号: 000, 期号: 010, 页码: 1359
作者:
Ma Shanyao
;
Ning Mengmeng
;
Zou Qingan
;
Feng Ying
;
Ye Yangliang
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/07/01
OL3
MN6
linagliptin
TGR5 agonist
DPP4 inhibitor
GLP-1
low-absorbed
gallbladder filling
type 2 diabetes mellitus
4-Benzofuranyloxynicotinamide derivatives are novel potent and orally available TGR5 agonists
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 82, 页码: 1-15
作者:
Zou, Qingan
;
Duan, Hongliang
;
Ning, Mengmeng
;
Liu, Jia
;
Feng, Ying
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
TGR5
4-Benzofuranyloxynicotinamide
Gallbladder toxicity
Caco-2 permeability
Scalp metastasis from gallbladder cancer: an unusual case
期刊论文
OAI收割
CHINESE MEDICAL JOURNAL, 2014, 卷号: 127
-
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/10/26
CARCINOMA
gallbladder cancer
scalp
metastasis