中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共9条,第1-9条 帮助

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Application of deep generative model for design of Pyrrolo[2,3-d] pyrimidine derivatives as new selective TANK binding kinase 1 (TBK1) inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 247, 页码: 115034
作者:  
Song, Shukai;  Tang, Haotian;  Ran, Ting;  Fang, Feng;  Tong, Linjiang
  |  收藏  |  浏览/下载:11/0  |  提交时间:2024/03/27
Temperature-Controlled Divergent Synthesis of Tetrasubstituted Alkenes and Pyrrolo[1,2-a]indole Derivatives via Iridium Catalysis 期刊论文  OAI收割
ASIAN JOURNAL OF ORGANIC CHEMISTRY, 2021, 页码: 14
作者:  
Liu, Siyu;  Mao, Hui;  Qiao, Jin;  Zhang, Xiaoning;  Lu, Yangbin
  |  收藏  |  浏览/下载:56/0  |  提交时间:2021/11/04
Identification of methyl (5-(6-((4-(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinopyrrolo[2,1-f][1,2,4]triazin-2-yl)-4-(trifluoromethyl)pyridin-2-yl)carbamate (CYH33) as an orally bioavailable, highly potent, PI3K alpha inhibitor for the treatment of advanced solid tumors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 209, 页码: 10
作者:  
Xiang, Hao-Yue;  Wang, Xiang;  Chen, Yan-Hong;  Zhang, Xi;  Tan, Cun
  |  收藏  |  浏览/下载:28/0  |  提交时间:2021/05/24
Design, synthesis and antiproliferative activity evaluation of a series of pyrrolo [2,1-f] [1,2,4] triazine derivatives 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 12, 页码: 4
作者:  
Xiang, Hao-Yue;  Chen, Yan-Hong;  Wang, Yi;  Zhang, Xi;  Ding, Jian
  |  收藏  |  浏览/下载:39/0  |  提交时间:2020/07/01
Discovery of a Novel Series of 7-Azaindole Scaffold Derivatives as PI3K Inhibitors with Potent Activity 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 8, 期号: 8, 页码: 875-880
作者:  
Yang, Chengbin;  Zhang, Xi;  Wang, Yi;  Yang, Yongtai;  Liu, Xiaofeng
  |  收藏  |  浏览/下载:40/0  |  提交时间:2019/01/08
A tandem copper (II)-promoted synthesis of 2-substituted pyrrolo [2,1-f][1,2,4] triazin-4(3H)-ones 期刊论文  OAI收割
TETRAHEDRON, 2013, 卷号: 69, 期号: 13, 页码: 2714-2719
作者:  
Chen, Yanhong;  Xiang, Haoyue;  Tan, Cun;  Xie, Yuyuan;  Yang, Chunhao
  |  收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
Synthesis and characterization of thieno[3,4-c]pyrrole-4,6-dione and pyrrolo [3,4-c]pyrrole-1,4-dione-based random polymers for photovoltaic applications 期刊论文  OAI收割
POLYMER, 2012, 卷号: 53, 期号: 20, 页码: 4407-4412
作者:  
Zhang, Guobing;  Fu, Yingying;  Qiu, Longzhen;  Xie, Zhiyuan
  |  收藏  |  浏览/下载:16/0  |  提交时间:2019/04/09
Molecular docking-based 3D-QSAR studies of pyrrolo[3,4-c]pyrazole derivatives as Aurora-A inhibitors 期刊论文  OAI收割
MOLECULAR SIMULATION, 2011, 卷号: 37, 期号: 1, 页码: 31-42
He, G.; Qiu, M. H.; Li, R.; Song, X. R.; Zheng, X.; Shi, J. Y.; Xu, G. B.; Han, J.; Yu, L. T.; Yang, S. Y.; Chen, L. J.; Wei, Y. Q.
收藏  |  浏览/下载:25/0  |  提交时间:2012/10/12
Gold(I)-Catalyzed One-Pot Tandem Coupling/Cyclization: An Efficient Synthesis of Pyrrolo-/Pyrido[2,1-b]benzo[d][1,3]oxazin-1-ones 期刊论文  OAI收割
ADVANCED SYNTHESIS & CATALYSIS, 2010, 卷号: 352, 期号: 2-3, 页码: 373-378
作者:  
Zhou, Yu;  Zhai, Yun;  Ji, Xun;  Liu, Guannan;  Feng, Enguang
  |  收藏  |  浏览/下载:24/0  |  提交时间:2019/01/08