中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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YC-1 inhibits proliferation of breast cancer cells by downregulating EZH2 expression via activation of c-Cbl and ERK
期刊论文
OAI收割
出版物, 3111, 期号: 0, 页码: 1-46
作者:
Ling-Chu Chang
;
Hui-Yi Lin
;
Meng-Tung Tsai
;
Ruey-Hwang Chou
;
Fang-Yu Lee
  |  
收藏
  |  
浏览/下载:259/0
  |  
提交时间:2017/07/24
Yc-1
Triple-negative Breast Cancer
Erk
Ezh2
C-cbl
The Tyrosine Kinase Inhibitor Bafetinib Inhibits PAR2-induced Activation of TRPV4 In Vitro and Pain In Vivo1
期刊论文
OAI收割
出版物, 2111, 页码: 1-44
作者:
1M S Grace
;
T Lieu
;
B Darby
;
F C Abogadie
;
N Veldhuis N W Bunnett
;
P McIntyre
  |  
收藏
  |  
浏览/下载:220/0
  |  
提交时间:2017/07/24
Transient Receptor Potential Ion Channel
Trpv4
Protease Activated Receptor
Par2
Pain
Tyrosine Kinase
Bafetinib
Synthesis of 1,4-epoxy-2-aryltetrahydro-1-benzazepines
via
rhodium(
iii
)-catalyzed C-H allylation/intramolecular 1,3-dipolar cycloaddition
期刊论文
OAI收割
CHEMICAL COMMUNICATIONS, 2024, 卷号: 60, 期号: 17, 页码: 2401-2404
作者:
Wang, Xuan
;
Li, Jianlong
;
Du, Haifang
;
Liang, Weihong
;
Luo, Cheng
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/03/13
Gold-catalyzed
endo
-selective Ring-opening of Epoxides and its Application in Construction of Poly-ethers
期刊论文
OAI收割
CHEMISTRY-A EUROPEAN JOURNAL, 2024, 页码: 10
作者:
Wu, Kehuan
;
Kang, Kaiwen
;
Liu, Dan
;
Zhang, Chiyue
;
Wang, Xinyu
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/03/25
6-endo ring-opening of epoxide
Baldwin's rules
gold-catalyzed reactions
marine ladder-like poly-ethers
Nakanishi hypothesis
Thermal stimulus task fMRI in the cervical spinal cord at 7 Tesla
期刊论文
OAI收割
HUMAN BRAIN MAPPING, 2024, 卷号: 45, 期号: 3, 页码: 14
作者:
Seifert, Alan C.
;
Xu, Junqian
;
Kong, Yazhuo
;
Eippert, Falk
;
Miller, Karla L.
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/04/01
7 T MRI
fMRI
spinal cord fMRI
ultra-high field
Fucoxanthin Alleviates Dextran Sulfate Sodium-Induced Colitis and Gut Microbiota Dysbiosis in Mice
期刊论文
OAI收割
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2024, 卷号: 72, 期号: 8, 页码: 4142-4154
作者:
Yang, Yu-Hong
;
Chen, Chen
;
Zheng, Yan
;
Wu, Zi-Jian
;
Zhou, Meng-Qing
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/04/07
fucoxanthin
colitis
intestinal barrier function
anti-inflammation
antioxidation
gut microbiota
Palladium-Catalyzed Deuteration of Arylketone Oxime Ethers
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2024, 页码: 7
作者:
Wang, Zhen-Yu
;
Zhang, Xu
;
Chen, Wen-Qing
;
Sun, Guo-Dong
;
Wang, Xing
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/03/13
C-C Bond Cleavage
Deacylation
Regioselective Deuteration
Difunctionalization
Palladium Catalysis
Discovery of a 1,6-naphthyridin-4-one-based AXL inhibitor with improved pharmacokinetics and enhanced in vivo antitumor efficacy
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 17
作者:
Lan, Yaohan
;
Peng, Xia
;
Ji, Yinchun
;
Su, Yi
;
Duan, Wenhu
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/02/27
AXL inhibitor
In vivo antitumor efficacy
6-Naphthyridin-4-one derivatives
Scaffold hopping
Structure-based drug design
Discovery of a CB2 and 5-HT1A receptor dual agonist for the treatment of depression and anxiety
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 20
作者:
Yang, Wenjiao
;
Gong, Xudong
;
Sun, Haiguo
;
Wu, Chunhui
;
Suo, Jin
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/03/06
CB2R agonist
5-HT1AR agonist
CB1R antagonist
Antidepressant
Anxiolytic
An LQT2-related mutation in the voltage-sensing domain is involved in switching the gating polarity of hERG
期刊论文
OAI收割
BMC BIOLOGY, 2024, 卷号: 22, 期号: 1, 页码: 14
作者:
Liu, Zhipei
;
Wang, Feng
;
Yuan, Hui
;
Tian, Fuyun
;
Yang, Chuanyan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/03/13
hERG
K525N
Gating Polarity
Voltage-Sensing Domain
LQT2