中国科学院机构知识库网格
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A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:
Yang, Xin-Mei
;
Yang, Yang
;
Yao, Bu-Fan
;
Ye, Pan-Pan
;
Xu, Yan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/11
COVID-19
Simnotrelvir
Safety
Pharmacokinetics
Healthy subjects
Structure-based development and preclinical evaluation of the SARS-CoV-2 3C-like protease inhibitor simnotrelvir
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 15
作者:
Jiang, Xiangrui
;
Su, Haixia
;
Shang, Weijuan
;
Zhou, Feng
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/03/25
COVID-19-related Olfactory Dysfunction: Prevalence, Mechanism and Recovery
期刊论文
OAI收割
PROGRESS IN BIOCHEMISTRY AND BIOPHYSICS, 2023, 卷号: 50, 期号: 6, 页码: 1245-1260
作者:
Xing, Chen
;
Ma, Jing-Chao
;
Yun, Han-Qi
;
Liu, Qing-Jing
;
Chang, Xiao-Yue
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/10/09
COVID-19
olfactory dysfunction
SARS-CoV-2
SARS-CoV-2 variants
long COVID
olfactory training
Sensitivity-enhanced nanoplasmonic biosensor using direct immobilization of two engineered nanobodies for SARS-CoV-2 spike receptor-binding domain detection
期刊论文
OAI收割
SENSORS AND ACTUATORS B-CHEMICAL, 2023, 卷号: 383, 页码: 133575
作者:
Ma, Zhengtai
;
Sun, Zengchao
;
Lv, Xiaoqing
;
Chen, Hongda
;
Geng, Yong
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/03/27
Nanoplasmonics
Biosensor
COVID-19
Nanobody
Immobilization
High -throughput
Structure-Based Design of Potent Peptidomimetic Inhibitors Covalently Targeting SARS-CoV-2 Papain-like Protease
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2023, 卷号: 24, 期号: 10, 页码: 15
作者:
Wang, Qian
;
Chen, Guofeng
;
He, Jian
;
Li, Jiameng
;
Xiong, Muya
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/10/17
SARS-CoV-2
papain-like protease
covalent inhibitor
co-crystal structure
in vitro assay
Unraveling the catalytic mechanism of SARS-CoV-2 papain-like protease with allosteric modulation of C270 mutation using multiscale computational approaches
期刊论文
OAI收割
CHEMICAL SCIENCE, 2023, 卷号: 14, 期号: 18, 页码: 4681-4696
作者:
Shao, Qiang
;
Xiong, Muya
;
Li, Jiameng
;
Hu, Hangchen
;
Su, Haixia
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/03/27
Discovery, synthesis and mechanism study of 2,3,5-substituted [1,2,4]-thiadiazoles as covalent inhibitors targeting 3C-Like protease of SARS-CoV-2
期刊论文
OAI收割
European journal of medicinal chemistry, 2023, 卷号: 249, 页码: 115129
作者:
Ren, Pengxuan
;
Yu, Changyue
;
Zhang, Ruxue
;
Nie, Tianqing
;
Hu, Qiaoyu
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/03/26
Localized delivery of nanomedicine and antibodies for combating COVID-19
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 5, 页码: 1828-1846
作者:
Tu, Bin
;
Gao, Yanrong
;
An, Xinran
;
Wang, Huiyuan
;
Huang, Yongzhuo
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/10/17
SARS-CoV-2
COVID-19
Nanomedicine
Orally-inhaled delivery
Intranasal delivery
Antibody
Discovery of Polyphenolic Natural Products as SARS-CoV-2 Mpro Inhibitors for COVID-19
期刊论文
OAI收割
PHARMACEUTICALS, 2023, 卷号: 16, 期号: 2, 页码: 190
作者:
Kruger, Nadine
;
Kronenberger, Thales
;
Xie, Hang
;
Rocha, Cheila
;
Pohlmann, Stefan
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/03/27
antivirals
coronavirus
COVID-19
covalent drugs
dynamic light scattering
inhibitors
main protease
natural products
Ginkgolic acids inhibit SARS-CoV-2 and its variants by blocking the spike protein/ACE2 interplay
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2023, 卷号: 226, 页码: 780-792
作者:
Xiang, Yusen
;
Zhai, Guanglei
;
Li, Yaozong
;
Wang, Mengge
;
Chen, Xixiang
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2023/04/10
SARS-CoV-2
S-RBD
Ginkgolic acid