中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [127]
采集方式
OAI收割 [127]
内容类型
期刊论文 [124]
会议论文 [3]
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2024 [1]
2023 [7]
2022 [10]
2021 [10]
2020 [4]
2019 [6]
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学科主题
Pharmacol... [12]
Plant Sci... [12]
Chemistry [9]
Biochemist... [4]
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浏览/检索结果:
共127条,第1-10条
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存缴方式:oaiharvest
专题:上海药物研究所
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Enzymatic Synthesis of Noncanonical α-Amino Acids Containing γ-Tertiary Alcohols
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2024, 页码: 9
作者:
Zhang, Rui
;
Zhang, Chenghua
;
Tan, Jiamu
;
He, Yifan
;
Zhuo, Dan
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/02/27
Asymmetric Synthesis
Biocatalysis
Noncanonical Amino Acids
Quantum Chemical Calculations
Tertiary Alcohols
A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:
Yang, Xin-Mei
;
Yang, Yang
;
Yao, Bu-Fan
;
Ye, Pan-Pan
;
Xu, Yan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/11
COVID-19
Simnotrelvir
Safety
Pharmacokinetics
Healthy subjects
Sesquiterpene lactones from Artemisia verlotorum and their anti-inflammatory activities
期刊论文
OAI收割
FITOTERAPIA, 2023, 卷号: 169, 页码: 11
作者:
Wang, Mengyu
;
Yang, Yue
;
Ke, Changqiang
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/10/17
Artemisia verlotorum
Verlotolides A -G
DFT NMR calculation
TDDFT ECD calculation
X-ray diffraction
Anti-inflammation
The first phytochemical investigation of Artemisia nujianensis: Eight new guaianolides and their anti-inflammatory activity
期刊论文
OAI收割
FITOTERAPIA, 2023, 卷号: 167, 页码: 9
作者:
Yu, Shan
;
Tang, Chunping
;
Ke, Chang-Qiang
;
Yao, Sheng
;
Feng, Zheling
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/10/17
Artemisia nujianensis
Guaianolide
Artenujianolides A-H
DFT NMR calculation
Anti-inflammatory activity
The First Phytochemical Investigation of Artemisia divaricate: Sesquiterpenes and Their Anti-Inflammatory Activity
期刊论文
OAI收割
MOLECULES, 2023, 卷号: 28, 期号: 10, 页码: 14
作者:
Yan, Siqi
;
Ke, Changqiang
;
Feng, Zheling
;
Tang, Chunping
;
Ye, Yang
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/10/17
Artemisia divaricate
sesquiterpene
divaricanolide A-I
anti-inflammatory activity
Extracellular vesicles mediate antibody-resistant transmission of SARS-CoV-2
期刊论文
OAI收割
CELL DISCOVERY, 2023, 卷号: 9, 期号: 1, 页码: 15
作者:
Xia, Bingqing
;
Pan, Xiaoyan
;
Luo, Rong-Hua
;
Shen, Xurui
;
Li, Shuangqu
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2023/04/10
Flavonoids from the roots and rhizomes of Sophora tonkinensis and their in vitro anti-SARS-CoV-2 activity
期刊论文
OAI收割
CHINESE JOURNAL OF NATURAL MEDICINES, 2023, 卷号: 21, 期号: 1, 页码: 65
作者:
Li Zhuo
;
Xie Hang
;
Tang Chunping
;
Feng Lu
;
Ke Changqiang
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/05/22
Sophora tonkinensis
Flavonoid
Anti-SARS-CoV-2 activity
SARS-CoV-2 3CLpro
SARS-CoV-2 PLpro
Discovery of HCD3514 as a potent EGFR inhibitor against C797S mutation in vitro and in vivo
期刊论文
OAI收割
JOURNAL OF CANCER, 2023, 卷号: 14, 期号: 1, 页码: 152-162
作者:
Lai, Mengzhen
;
Zhang, Tao
;
Chen, Hao
;
Song, Peiran
  |  
收藏
  |  
浏览/下载:80/0
  |  
提交时间:2023/04/10
fourth-generation EGFR inhibitor
EGFRC797S mutation
NSCLC
drug resistance
small molecular inhibitor
Fused-ring alpha-pyrones from intramolecular C-H activation and their lipids-lowering activity associated with LXR-IDOL-LDLR axis regulation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 244, 页码: 11
作者:
Mao, Yingle
;
Li, Jiaomeng
;
Tang, Chunping
;
Ma, Biao
;
Xu, Zhijian
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/04/10
C-H activation
One-pot intramolecular cyclization
?-Pyrone derivatives
LDL uptaking
LXR-IDOL-LDLR axis
In vivo lipids-lowering effect
ASK120067 potently suppresses B-cell or T-cell malignancies in vitro and in vivo by inhibiting BTK and ITK
期刊论文
OAI收割
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13, 页码: 9
作者:
Song, Peiran
;
Bai, Gang
;
Chan, Shingpan
;
Zhang, Tao
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2023/04/10
Bruton's tyrosine kinase
interleukin-2-inducible T cell kinase
ASK120067
B-cell lymphoma
T-cell leukemia