中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [20]
昆明植物研究所 [2]
上海生物化学与细胞生... [2]
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OAI收割 [29]
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期刊论文 [28]
学位论文 [2]
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2023 [5]
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2008 [3]
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Immunology... [1]
Virology [1]
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A viral RNA-dependent RNA polymerase inhibitor VV116 broadly inhibits human coronaviruses and has synergistic potency with 3CLpro inhibitor nirmatrelvir
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 10
作者:
Zhang, Yumin
;
Sun, Yuan
;
Xie, Yuanchao
;
Shang, Weijuan
;
Wang, Zhen
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2023/12/08
Design, synthesis and biological evaluation of peptidomimetic benzothiazolyl ketones as 3CLpro inhibitors against SARS-CoV-2
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 257, 页码: 13
作者:
Yang, Hanxi
;
You, Mengyuan
;
Shu, Xiaoyang
;
Zhen, Jingyao
;
Zhu, Mengwei
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/10/17
Peptidomimetics
Benzothiazolyl ketone
3CLpro inhibitor
Pharmacokinetic properties
SARS-CoV-2
Efficacy and safety of SIM0417 (SSD8432) plus ritonavir for COVID-19 treatment: a randomised, double-blind, placebo- controlled, phase 1b trial
期刊论文
OAI收割
LANCET REGIONAL HEALTH-WESTERN PACIFIC, 2023, 卷号: 38, 页码: 13
作者:
Wang, Fuxiang
;
Xiao, Wen
;
Tang, Yimin
;
Cao, Mengli
;
Shu, Dan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Covid-19
3CL protease inhibitor
SARS-CoV-2 viral load
Alleviation of COVID-19 symptoms
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors
期刊论文
OAI收割
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1, 页码: 17-27
作者:
Zang, Yi
;
Su, Mingbo
;
Wang, Qingxing
;
Cheng, Xi
;
Zhang, Wenru
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/03/27
high-throughput screening
SARS
CoV-2
main
papain-like
proteases
Flavonoids from the roots and rhizomes of Sophora tonkinensis and their in vitro anti-SARS-CoV-2 activity
期刊论文
OAI收割
CHINESE JOURNAL OF NATURAL MEDICINES, 2023, 卷号: 21, 期号: 1, 页码: 65
作者:
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/05/22
Sophora tonkinensis
Flavonoid
Anti-SARS-CoV-2 activity
SARS-CoV-2 3CLpro
SARS-CoV-2 PLpro
In vitro and in vivo evaluation of the main protease inhibitor FB2001 against SARS-CoV-2
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2022, 卷号: 208, 页码: 10
作者:
Shang, Weijuan
;
Dai, Wenhao
;
Yao, Cheng
;
Xu, Ling
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/04/10
SARS-CoV-2
SARS-CoV-2 variants
FB2001
Main protease
PBPK
Anti-SARS-CoV-2 in vivo
Predicting In Vitro and In Vivo Anti-SARS-CoV-2 Activities of Antivirals by Intracellular Bioavailability and Biochemical Activity
期刊论文
OAI收割
ACS OMEGA, 2022, 页码: 13
作者:
Zhang, Jinwen
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/04/10
Mililatensols A-C, New Records of Sarsolenane and Capnosane Diterpenes from Soft Coral Sarcophyton mililatensis
期刊论文
OAI收割
MARINE DRUGS, 2022, 卷号: 20, 期号: 9, 页码: 10
作者:
Bu, Qing
;
Yang, Min
;
Yan, Xian-Yun
;
Li, Song-Wei
;
Ge, Zeng-Yue
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/11/11
soft coral
Sarcophyton mililatensis
sarsolenane
capnosane
stereochemistry
anti-inflammatory activity
Synthesis and anti-SARS-CoV-2 activity of deuterated GS-441524 analogs
期刊论文
OAI收割
TETRAHEDRON LETTERS, 2022, 卷号: 104, 页码: 9
作者:
Zheng, Wei
;
Hu, Tianwen
;
Zhang, Yumin
;
Wei, Daibao
;
Xie, Yuanchao
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2022/11/11
SARS-CoV-2
GS-441524
Deuterated
Structures of the Omicron spike trimer with ACE2 and an anti-Omicron antibody
期刊论文
OAI收割
SCIENCE, 2022, 卷号: 375, 期号: 6584, 页码: 1048-+
作者:
Yin, Wanchao
;
Xu, Youwei
;
Xu, Peiyu
;
Cao, Xiaodan
;
Wu, Canrong
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/06/15