中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
  • 上海药物研究所 [31]
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发表日期
  • 2019 [31]
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浏览/检索结果: 共31条,第1-10条 帮助

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Common activation mechanism of class A GPCRs 期刊论文  OAI收割
ELIFE, 2019, 卷号: 8, 页码: 31
作者:  
Zhou, Qingtong;  Yang, Dehua;  Wu, Meng;  Guo, Yu;  Guo, Wangjing
  |  收藏  |  浏览/下载:76/0  |  提交时间:2020/07/01
HRAS(G12s) mutant mediates resistance to a PI3K alpha inhibitor CYH33 in esophageal squamous cell carcinomas 期刊论文  OAI收割
MOLECULAR CANCER THERAPEUTICS, 2019, 卷号: 18, 期号: 12, 页码: 2
作者:  
Wang, Yuxiang;  Zhang, Xu;  Ma, Qingyang;  Zhang, Xi;  Yang, Chunhao
  |  收藏  |  浏览/下载:21/0  |  提交时间:2020/07/01
Design, synthesis, and biological evaluation of thieno[3,2-d]pyrimidine derivatives as potential simplified phosphatidylinositol 3-kinase alpha inhibitors 期刊论文  OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2019, 卷号: 94, 期号: 6, 页码: 2013-2022
作者:  
Yang, Xiuyan;  Deng, Meng;  Zhang, Xi;  Wang, Yi;  Song, Kun
  |  收藏  |  浏览/下载:31/0  |  提交时间:2020/07/01
Unbiased screening reveals that blocking exportin 1 overcomes resistance to PI3K alpha inhibition in breast cancer 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2019, 卷号: 4, 页码: 3
作者:  
Liu, Xue-Ling;  Wang, Bo-Bo;  Wang, Yi;  Wang, Yu-Xiang;  Yang, Chun-hao
  |  收藏  |  浏览/下载:11/0  |  提交时间:2020/07/01
Effects of traditional Chinese medicine formula Le-Cao-Shi on hepatitis B: In vivo and in vitro studies 期刊论文  OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2019, 卷号: 244, 页码: 10
作者:  
Zhao, Qing;  Ren, Xia;  Chen, Min;  Yue, Shi-Jun;  Zhang, Meng-Qi
  |  收藏  |  浏览/下载:34/0  |  提交时间:2020/07/01
Development and Characterization of a Fluorescent Probe for GLS1 and the Application for High-Throughput Screening of Allosteric Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 21, 页码: 9642-9657
作者:  
Xu, Xi;  Kuang, Zijian;  Han, Jie;  Meng, Ying;  Li, Lei
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/03/21
Current trends in drug metabolism and pharmacokinetics 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2019, 卷号: 9, 期号: 6, 页码: 1113-1144
作者:  
Li, Yuhua;  Meng, Qiang;  Yang, Mengbi;  Liu, Dongyang
  |  收藏  |  浏览/下载:35/0  |  提交时间:2020/07/01
Design, synthesis and antitumor study of a series of N-Cyclic sulfamoylaminoethyl substituted 1,2,5-oxadiazol-3-amines as new indoleamine 2, 3-dioxygenase 1 (IDO1) inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 179, 页码: 38-55
作者:  
Chen, Shulun;  Guo, Wei;  Liu, Xiaohua;  Sun, Pu;  Wang, Yi
  |  收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01
Structure-Based Discovery and Development of a Series of Potent and Selective Bromodomain and Extra-Terminal Protein Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 18, 页码: 8642-8663
作者:  
Hu, Jianping;  Tian, Chang-Qing
  |  收藏  |  浏览/下载:35/0  |  提交时间:2020/07/01
Cinerols, Nitrogenous Meroterpenoids from the Marine Sponge Dysidea cinerea 期刊论文  OAI收割
JOURNAL OF NATURAL PRODUCTS, 2019, 卷号: 82, 期号: 9, 页码: 2586-2593
作者:  
Jiao, Wei-Hua;  Li, Jing;  Wang, Dan;  Zhang, Meng-Meng;  Liu, Li-Yun
  |  收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01