中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [10]
采集方式
OAI收割 [10]
内容类型
期刊论文 [10]
发表日期
2023 [10]
学科主题
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发表日期:2023
专题:上海药物研究所
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Asponchimides A-E: new enantiomeric N-acetyldopamine trimers from Aspongopus chinensis
期刊论文
OAI收割
CHINESE JOURNAL OF NATURAL MEDICINES, 2023, 卷号: 21, 期号: 11, 页码: 859-867
作者:
Nie, Jinchun
;
Mei, Fang
;
Zheng, Yueyuan
;
Wen, Qiuyi
;
Li, Zhenwei
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/01/26
Aspongopus chinensis
N-acetyldopamine trimer
ECD calculations
NO inhibitory activity
Structural insights into the interaction of three Y- shaped ligands with PI3Kα
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2023, 卷号: 120, 期号: 34, 页码: 9
作者:
Zhou, Qingtong
;
Liu, Xiao
;
Neri, Dario
;
Li, Wenxin
;
Favalli, Nicholas
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/12/08
phosphoinositide 3-kinase
drug target
ligand
binding pocket
chemical scaffold
OTTM: an automated classification tool for translational drug discovery from omics data
期刊论文
OAI收割
BRIEFINGS IN BIOINFORMATICS, 2023, 页码: 12
作者:
Yang, Xiaobo
;
Zhang, Bei
;
Wang, Siqi
;
Lu, Ye
;
Chen, Kaixian
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/10/17
OTTM
omics data
translational drug discovery
literature mining
hepatocellular carcinoma
The first phytochemical investigation of Artemisia nujianensis: Eight new guaianolides and their anti-inflammatory activity
期刊论文
OAI收割
FITOTERAPIA, 2023, 卷号: 167, 页码: 9
作者:
Yu, Shan
;
Tang, Chunping
;
Ke, Chang-Qiang
;
Yao, Sheng
;
Feng, Zheling
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2023/10/17
Artemisia nujianensis
Guaianolide
Artenujianolides A-H
DFT NMR calculation
Anti-inflammatory activity
Design, synthesis of novel benzimidazole derivatives as ENL inhibitors suppressing leukemia cells viability via downregulating the expression of MYC
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 248, 页码: 14
作者:
Guo, Siqi
;
Jia, Tongguan
;
Xu, Xiaoming
;
Yang, Feng
;
Xiao, Senhao
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/04/10
ENL Inhibitor
YEATS domain
Histone lysine acetylation
Benzimidazole derivatives
Acute myeloid leukemia
New cembranoids from the leaves and twigs of Croton yanhuii Y. T. Chang
期刊论文
OAI收割
NATURAL PRODUCT RESEARCH, 2023, 页码: 7
作者:
Zhang, Daidi
;
Wang, Didi
;
Li, Zhenwei
;
Guo, Dean
;
Li, Wei
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/04/10
Euphorbiaceae
Croton yanhuii Y
T
Chang
cembranoids
ECD calculations
NO inhibitory activity
Coumaronochromones, flavanones, and isoflavones from the twigs and leaves of Erythrina subumbrans inhibit PTP1B and nitric oxide production
期刊论文
OAI收割
PHYTOCHEMISTRY, 2023, 卷号: 206, 页码: 12
作者:
Liu, Cai-Ying
;
Deng, Pan
;
Wang, Bin
;
Liu, Ai-Hong
;
Wang, Meng-Ge
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/04/10
Erythrina subumbrans
Fabaceae
Sesquiterpenoids
Coumaronochromones
Flavanones
Isoflavones
Nitric oxide production inhibition
PTP1B inhibition
Cembrane Diterpenes Possessing Nonaromatic Oxacycles from the Hainan Soft Coral Sarcophyton mililatensis
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2023, 卷号: 24, 期号: 3, 页码: 1979
作者:
Zhang, Ling
;
Yang, Min
;
Chen, Zi-Hui
;
Ge, Zeng-Yue
;
Li, Song-Wei
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/03/27
soft coral
Sarcophyton mililatensis
cembrane diterpene
absolute configuration
TNF-alpha inhibitory
binding mode
Five New Diarylbutyrolactones and Sesquilignans from Saussurea medusa and Their Inhibitory Effects on LPS-induced NO Production
期刊论文
OAI收割
PLANTA MEDICA, 2023, 页码: 11
作者:
Cao, Jing-Ya
;
Wang, Zhi-Yao
;
Stewart, Alan J. J.
;
Dong, Qi
;
Zhao, Ye
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/04/10
Saussurea medusa
Asteraceae
diarylbutyrolactone lignan
sesquilignan
anti-inflammatory activity
molecular docking
Combined inhibition of PARP and ATR synergistically potentiates the antitumor activity of HER2-targeting antibody-drug conjugate in HER2-positive cancers
期刊论文
OAI收割
AMERICAN JOURNAL OF CANCER RESEARCH, 2023, 卷号: 13, 期号: 1, 页码: 161-+
作者:
Li, Yongpeng
;
Li, Lin
;
Fu, Haoyu
;
Yao, Qing
;
Wang, Lei
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/10/17
Antibody-drug conjugate
DS-8201
PARP
ATR
synergy
DNA damage