中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共169条,第1-10条 帮助

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Distinct roles of the extracellular surface residues of glucagon-like peptide-1 receptor in B-arrestin 1/2 signaling 期刊论文  OAI收割
EUROPEAN JOURNAL OF PHARMACOLOGY, 2024, 卷号: 968, 页码: 17
作者:  
Lei, Saifei;  Meng, Qian;  Liu, Yanyun;  Liu, Qiaofeng;  Dai, Antao
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/05/22
Cryo-electron microscopy for GPCR research and drug discovery in endocrinology and metabolism 期刊论文  OAI收割
NATURE REVIEWS ENDOCRINOLOGY, 2024, 页码: 17
作者:  
Duan, Jia;  He, Xin-Heng;  Li, Shu-Jie;  Xu, H. Eric
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/07
Exploration of the potential association between GLP-1 receptor agonists and suicidal or self-injurious behaviors: a pharmacovigilance study based on the FDA Adverse Event Reporting System database 期刊论文  OAI收割
BMC MEDICINE, 2024, 卷号: 22, 期号: 1, 页码: 13
作者:  
Zhou, Jianxing;  Zheng, You;  Xu, Baohua;  Long, Songjun;  Zhu, Li-e
  |  收藏  |  浏览/下载:20/0  |  提交时间:2024/03/25
Molecular features of the ligand-free GLP-1R, GCGR and GIPR in complex with Gs proteins 期刊论文  OAI收割
CELL DISCOVERY, 2024, 卷号: 10, 期号: 1, 页码: 13
作者:  
Cong, Zhaotong;  Zhao, Fenghui;  Li, Yang;  Luo, Gan;  Mai, Yiting
  |  收藏  |  浏览/下载:26/0  |  提交时间:2024/03/13
Tail engagement of arrestin at the glucagon receptor 期刊论文  OAI收割
NATURE, 2023, 页码: 21
作者:  
Chen, Kun;  Zhang, Chenhui;  Lin, Shuling;  Yan, Xinyu;  Cai, Heng
  |  收藏  |  浏览/下载:15/0  |  提交时间:2023/10/17
Structural analysis of the dual agonism at GLP-1R and GCGR 期刊论文  OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2023, 卷号: 120, 期号: 33, 页码: 12
作者:  
Li, Yang;  Zhou, Qingtong;  Dai, Antao;  Zhao, Fenghui;  Chang, Rulue
  |  收藏  |  浏览/下载:0/0  |  提交时间:2024/05/07
Conserved class B GPCR activation by a biased intracellular agonist 期刊论文  OAI收割
NATURE, 2023, 页码: 25
作者:  
Zhao, Li-Hua;  He, Qian;  Yuan, Qingning;  Gu, Yimin;  He, Xinheng
  |  收藏  |  浏览/下载:10/0  |  提交时间:2023/10/17
Discovery of Novel 5,6-Dihydro-1,2,4-triazine Derivatives as Efficacious Glucagon-Like Peptide-1 Receptor Agonists 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 23
作者:  
Chen, Lili;  Yun, Ying;  Guo, Shimeng;  Wang, Xiaoyan;  Xiong, Muya
  |  收藏  |  浏览/下载:10/0  |  提交时间:2023/10/17
Design and exploration of gut-restricted bifunctional molecule with TGR5 agonistic and DPP4 inhibitory effects for treating ulcerative colitis 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 242, 页码: 114697
作者:  
Han, Fanghui;  Ning, Mengmeng;  Wang, Kai;  Gu, Yipei;  Qu, Hui
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/03/21
Structure insights into selective coupling of G protein subtypes by a class B G protein-coupled receptor 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2022, 卷号: 13, 期号: 1, 页码: 13
作者:  
Zhao, Li-Hua;  Lin, Jingyu;  Ji, Su-Yu;  Zhou, X. Edward;  Mao, Chunyou
  |  收藏  |  浏览/下载:15/0  |  提交时间:2023/04/10