机构

• 上海药物研究所 [4]
• 长春光学精密机械与物... [3]
• 化学研究所 [2]
• 工程热物理研究所 [2]
• 自动化研究所 [1]
• 生态环境研究中心 [1]
• 更多

采集方式

• OAI收割 [13]

内容类型

• 期刊论文 [8]
• 会议论文 [4]
• 学位论文 [1]

发表日期

• 2022 [1]
• 2019 [2]
• 2015 [3]
• 2012 [3]
• 2007 [2]
• 2006 [1]
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浏览/检索结果: 共13条，第1-10条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择题名升序题名降序提交时间升序提交时间降序作者升序作者降序发表日期升序发表日期降序 Synthesis and Biochemical Evaluation of 8H-Indeno[1,2-d]thiazole Derivatives as Novel SARS-CoV-2 3CL Protease Inhibitors 期刊论文  OAI收割 MOLECULES, 2022, 卷号: 27, 期号: 10, 页码: 11 作者:  Wu, Jing;  Feng, Bo;  Gao, Li-Xin;  Zhang, Chun;  Li, Jia   |  收藏  |  浏览/下载：43/0  |  提交时间：2022/08/16 COVID-19  M-pro inhibitors  drug design and synthesis  structure-activity relationships (SAR)   Rational Design, synthesis and biological evaluation of novel triazole derivatives as potent and selective PRMT5 inhibitors with antitumor activity 期刊论文  OAI收割 JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2019, 卷号: 33, 期号: 8, 页码: 775-785 作者:  Zhu, Kongkai;  Shao, Jingwei;  Tao, Hongrui;  Yan, Xue;  Luo, Cheng   |  收藏  |  浏览/下载：31/0  |  提交时间：2020/07/01 PRMT5 inhibitor  Anti-proliferative  Cellular target validation  Design and synthesis   Robust global consensus tracking of linear multi-agent systems with input saturation via scheduled low-and-high gain feedback 期刊论文  OAI收割 IET CONTROL THEORY AND APPLICATIONS, 2019, 卷号: 13, 期号: 1, 页码: 69-77 作者:  Chu, Hongjun;  Chen, Jianliang;  Wei, Qinglai;  Zhang, Weidong   |  收藏  |  浏览/下载：64/0  |  提交时间：2019/07/12 reduced order systems  observers  multi-agent systems  linear systems  multi-robot systems  actuators  robust control  state feedback  feedback  control system synthesis  topology  robust global consensus tracking  input saturation  agent dynamics  general linear systems  actuator saturation  input additive uncertainties  state feedback protocol  disturbance rejection  reduced-order observer-based protocol design  linear multi-agent systems  scheduled low-and-high gain feedback  network topology   An MILP (mixed integer linear programming) model for optimal design of district-scale distributed energy resource systems 期刊论文  OAI收割 ENERGY, 2015, 卷号: 90, 页码: 1901-1915 作者:  Yang, Yun;  Zhang, Shijie;  Xiao, Yunhan 收藏  |  浏览/下载：28/0  |  提交时间：2016/03/09 Distributed energy resource  Optimal design  Synthesis and operation strategies  Energy distribution networks  Mixed integer linear programming   Optimal design of distributed energy resource systems coupled with energy distribution networks 期刊论文  OAI收割 ENERGY, 2015, 卷号: 85, 页码: 433-448 作者:  Yang, Yun;  Zhang, Shijie;  Xiao, Yunhan 收藏  |  浏览/下载：17/0  |  提交时间：2015/10/27 Distributed energy resource  Optimal design  Synthesis and operation strategies  Energy distribution networks  Mixed integer linear programming   synthesischaracterizationandbiologicalactivitiesof356trisubstituted124triazinederivatives 期刊论文  OAI收割 chinesejournaloforganicchemistry, 2015, 卷号: 35, 期号: 1, 页码: 191 作者:  Li YJ(李英俊);  Shi XL(史相玲);  Gao LX(高立信);  Jin K(靳焜);  Sheng L(盛丽)   |  收藏  |  浏览/下载：18/0  |  提交时间：2020/07/01 MICROWAVE-ASSISTED SYNTHESIS  BENZIMIDAZOLE DERIVATIVES  ANTITUMOR-ACTIVITY  COMPLEXES  CYTOTOXICITY  DESIGN  3,5,6-trisubstituted-1,2,4-triazine  benzimidazole  microwave irradiation  synthesis  crystal structure  Cdc25B and PTP1B inhibitors   Design,Synthesis and Evaluation of Indolebutylamines as a Novel Class of Selective Dopamine D3 Receptor Ligands 会议论文  OAI收割 作者:  Xu LL(徐丽丽);  Du P(杜鹏);  Yu KQ(于坤千);  Zhao WL(赵伟利);  Zhen XC(镇学初)   |  收藏  |  浏览/下载：26/0  |  提交时间：2019/01/08 Design,Synthesis and Evaluation of Indolebutylamines as a Novel Class of Selective Dopamine D3 Receptor Ligands   新型甲氧基丙烯酸酯类衍生物的设计合成及生物活性研究 学位论文  OAI收割 博士后, 北京: 中国科学院研究生院, 2012 张翔 收藏  |  浏览/下载：72/0  |  提交时间：2014/05/13 甲氧基丙烯酸酯  杀菌剂  嘧啶  生物活性：构效关系  分子设计与合成  Synthesis  Fungicide  Substituted Pyrimidine  Antifungal Activities  SAR  Molecular Design and Synthesis.   Accuracy synthesis of a 3-RPS parallel robot based on manufacturing costs (EI CONFERENCE) 会议论文  OAI收割 31st Chinese Control Conference, CCC 2012, July 25, 2012 - July 27, 2012, Hefei, China Yao T.-K.; Xi Z.; Feng Z.; Zhang L.-M.; Yong W. 收藏  |  浏览/下载：32/0  |  提交时间：2013/03/25 Pose accuracy is an important issue for parallel robot being used as mirror supporting system of telescope. One challenging topic is the accuracy synthesis which deals with the optimal design of the manufacturing and assembling tolerances of each component under the given pose accuracy. First  the error model of the 3-RPS parallel robot is built based on total derivation of the kinematic equations. And the error variable of each spherical or rotate joint can be expressed as a single boundary error parameter but not three independent position parameters. Then  the accuracy synthesis model is formulated taking the manufacturing costs as the optimization objective and the accuracy requirements as the constraint condition. Finally  the genetic algorithm is used to solve the optimization problem and a simulation example is given. The results show that the accuracy synthesis method based on manufacturing costs can satisfy the need of pose accuracy and is better for engineering application than the method based on error sensitivity. 2012 Chinese Assoc of Automati.   Super-resolved imaging system with oversampling technology (EI CONFERENCE) 会议论文  OAI收割 3rd International Symposium on Advanced Optical Manufacturing and Testing Technologies, AOMATT 2007: Advanced Optical Manufacturing Technologies, July 8, 2007 - July 12, 2007, Chengdu, China 作者:  Zhang X.;  Wang L.-J.;  Wang L.-J.;  Zhang J.-P.;  Liu Y. 收藏  |  浏览/下载：63/0  |  提交时间：2013/03/25 It has been a significant issue in the imaging filed to provide the highest possible resolution of an electro-optical imaging system(E-O imaging system). CCD arrays are inherently undersampled and spatial frequency above Nyquist frequency is distorted so as to create ambiguity and Moire patterns for targets imaged by E-O system.. As to this drawback  a system-design project is introduced and discussed in the paper. It's well known that many image quality metrics are linked to MTF. However  CCDs don't satisfy MTF condition  namely  the shift-invariant property  so MTF synthesis can't appraise the whole system simply by the MTF product of the few sub-system ones in E-O imaging system. Then it is depicted how to solve this problem in the following. Finally the analyses and comparisons of the imaging performance parameters with and without super-resolved technologies are shown.