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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [41]
大连化学物理研究所 [3]
过程工程研究所 [3]
金属研究所 [2]
西北高原生物研究所 [2]
生态环境研究中心 [2]
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OAI收割 [56]
内容类型
期刊论文 [55]
会议论文 [1]
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2025 [4]
2024 [5]
2023 [3]
2022 [4]
2021 [1]
2020 [3]
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Pharmacolo... [3]
Chemistry [2]
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Surface enhanced Raman scattering (SERS) for traditional Chinese medicine analysis: Current status and future perspectives
期刊论文
OAI收割
TRAC-TRENDS IN ANALYTICAL CHEMISTRY, 2025, 卷号: 193, 页码: 22
作者:
Zhao, Rui
;
Wang, Qishuo
;
Wang, Yunqing
;
Mei, Rongchao
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2025/11/10
Traditional Chinese medicine
Surface-enhanced Raman scattering
Quality assessment
Safety evaluation
Active ingredient screening
Pharmacokinetic analysis
Conformational restriction enables discovering a series of chroman derivatives as potent and selective NaV1.8 inhibitors with improved pharmacokinetic properties
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 293, 页码: 24
作者:
Li, Na
;
Wang, Linlin
;
Hu, Xinyuan
;
Xu, Haiyan
;
Yang, Bowen
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2025/08/20
Voltage-gated sodium channel 1.8
Conformational restriction
Pharmacokinetic
Structure-activity relationship
Analgesic
Guiding precision medicine strategy for intravenous ginsenosides via pharmacokinetic-informed bioinformatic approaches: a study on XueShuanTong
期刊论文
OAI收割
PHYTOMEDICINE, 2025, 卷号: 143, 页码: 18
作者:
Jia, Wei-Wei
;
Tian, Nan-Nan
;
Song, Zi-Jing
;
Lan, Xiao-Fang
;
Yang, Xi-He
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2025/08/20
Precision medicine
Physiologically based pharmacokinetic model
Ginsenoside
Albumin-facilitated dissociation
Drug interaction
Drug transporter
Hepatic impairment
Characterization of preclinical radio ADME properties of ARV-471 for predicting human PK using PBPK modeling
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL ANALYSIS, 2025, 卷号: 15, 期号: 5, 页码: 15
作者:
He, Yifei
;
Zhu, Chenggu
;
Lei, Peng
;
Yang, Chen
;
Zhang, Yifan
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2025/08/20
PROTAC
Vepdegestrant (ARV-471)
Radiolabeling
In vitro-in vivo extrapolation (IVIVE)
Physiologically based pharmacokinetic
(PBPK) model
Design and synthesis of pyridazin-4-one derivatives as necroptosis inhibitors
期刊论文
OAI收割
ARCHIV DER PHARMAZIE, 2024, 页码: 16
作者:
An, Yuxiang
;
Peng, Xia
;
Wang, Tianchen
;
Liu, Kaiyuan
;
Feng, Dazhi
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2024/12/25
inhibitor
pharmacokinetic study
pyridazin-4-one
receptor-interacting protein kinase 1
selectivity
Prediction of Multi-Pharmacokinetics Property in Multi-Species: Bayesian Neural Network Stacking Model with Uncertainty
期刊论文
OAI收割
MOLECULAR PHARMACEUTICS, 2024, 页码: 16
作者:
Zhang, Yuanyuan
;
Xie, Zhiyin
;
Xiao, Fu
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/12/11
pharmacokinetic parameters
machine learning
uncertainty
stacking
multitask learning
ADME
Strap-on Buoyant Device to Enhance Gastrointestinal Tract Retention of Felodipine Osmotic Pump Tablets
期刊论文
OAI收割
AAPS PHARMSCITECH, 2024, 卷号: 25, 期号: 8, 页码: 14
作者:
Ni, Qijia
;
Li, Zeru
;
Baqing, Libumo
;
Li, Tianfu
;
Xu, Huipeng
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2024/12/11
Gastro-retentive floating device
Osmotic pump
Pharmacokinetic
Stereolithography three-dimensional printing
Discovery and optimization of 3-(indolin-5-yloxy)pyridin-2-amine derivatives as potent necroptosis inhibitors
期刊论文
OAI收割
ARCHIV DER PHARMAZIE, 2024, 页码: 21
作者:
Lan, Yaohan
;
Ji, Yinchun
;
Peng, Xia
;
Duan, Wenhu
;
Geng, Meiyu
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/08/22
autoimmune disease
necroptosis inhibitor
pharmacokinetic profile
receptor interacting protein kinase 1 (RIPK1)
structural optimization
Pharmacologically significant constituents collectively responsible for anti-sepsis action of XueBiJing, a Chinese herb-based intravenous formulation
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 16
作者:
Cheng, Chen
;
Ren, Chao
;
Li, Mu-zi
;
Liu, Yi-hui
;
Yao, Ren-qi
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2024/02/27
Traditional Chinese medicine
XueBiJing
sepsis
mortality
pharmacokinetic compatibility
polypharmacology
Design, synthesis and biological evaluation of peptidomimetic benzothiazolyl ketones as 3CLpro inhibitors against SARS-CoV-2
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 257, 页码: 13
作者:
Yang, Hanxi
;
You, Mengyuan
;
Shu, Xiaoyang
;
Zhen, Jingyao
;
Zhu, Mengwei
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2023/10/17
Peptidomimetics
Benzothiazolyl ketone
3CLpro inhibitor
Pharmacokinetic properties
SARS-CoV-2