中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [71]
西北高原生物研究所 [48]
大连化学物理研究所 [15]
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期刊论文 [193]
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Discovery of GPX4 inhibitors through FP-based high-throughput screening
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:
Cao, Yu
;
Wu, Bin
;
Xu, Ying
;
Wang, Mingchen
;
Wu, Xinyu
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2024/02/27
GPX4 inhibitor
HTS assay
Ferroptosis
Fluorescence polarization
Zebrafish (Danio rerio) TR beta- and TTR-based electrochemical biosensors: Construction and application for the evaluation of thyroid-disrupting activity of bisphenols
期刊论文
OAI收割
ENVIRONMENTAL POLLUTION, 2023, 卷号: 330, 页码: 9
作者:
Li, Yuejiao
;
Zhang, Zhenzhong
;
Wang, Jun
;
Shan, Yeqi
;
Tian, Hua
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/12/07
Thyroid-disrupting chemicals
Thyroid hormone receptor beta
Transthyretin
In vitro screening Assay
Electrochemical biosensor
Constructing an MCF-7 breast cancer cell-based transient transfection assay for screening RAR? (Ant)agonistic activities of emerging phenolic compounds
期刊论文
OAI收割
JOURNAL OF HAZARDOUS MATERIALS, 2022, 卷号: 435, 期号: 0, 页码: 129024
作者:
Xu, Hanqing
;
Su, Jiahui
;
Ku, Tingting
;
Liu, Qian S.
;
Liang, Jiefeng
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2022/11/08
ACID RECEPTOR-ALPHA
RETINOIC ACID
GENE-EXPRESSION
DEPENDENT TRANSCRIPTION
GROWTH-INHIBITION
IN-VITRO
RXR
CONTAMINANTS
ANTAGONIST
ACTIVATION
Effect-directed analysis of estrogenic chemicals in sediments from an electronic-waste recycling area
期刊论文
OAI收割
ENVIRONMENTAL POLLUTION, 2022, 卷号: 306, 期号: 0, 页码: 119369
作者:
Ma, Qianchi
;
Yang, Xiaoxi
;
Guo, Yunhe
;
Wang, Yi
;
Liu, Yanna
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2022/11/08
POLYBROMINATED DIPHENYL ETHERS
RECEPTOR-MEDIATED ACTIVITIES
IN-VITRO
BODY-COMPOSITION
BISPHENOL-A
IDENTIFICATION
HORMONE
PROTEIN
ALPHA
WATER
A Multiwell-Based Assay for Screening Thyroid Hormone Signaling Disruptors Using thibz Expression as a Sensitive Endpoint in Xenopus laevis
期刊论文
OAI收割
MOLECULES, 2022, 卷号: 27, 期号: 3, 页码: 798
作者:
Li, Jinbo
;
Li, Yuanyuan
;
Zhu, Min
;
Song, Shilin
;
Qin, Zhanfen
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2022/11/08
GENE-EXPRESSION
BISPHENOL-A
IN-VITRO
POSTEMBRYONIC DEVELOPMENT
VERTEBRATE DEVELOPMENT
RECEPTOR DISRUPTORS
METAMORPHOSIS ASSAY
TRICLOSAN
TETRABROMOBISPHENOL
EXPOSURE
Screening for alpha-Glucosidase-Inhibiting Saponins from Pressurized Hot Water Extracts of Quinoa Husks
期刊论文
OAI收割
FOODS, 2022, 卷号: 11, 期号: 19
作者:
Su, R
;
Li, J
;
Hu, N
;
Wang, HL
;
Cao, JY
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2022/12/02
Histone deacetylase inhibitor givinostat alleviates liver fibrosis by regulating hepatic stellate cell activation
期刊论文
OAI收割
MOLECULAR MEDICINE REPORTS, 2021, 卷号: 23, 期号: 5, 页码: 12
作者:
Huang, He-Ming
;
Zhou, Xiao-Ru
;
Liu, Yan-Jun
;
Fan, Shi-Jie
;
Liao, Li-Ping
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2021/05/24
liver fibrosis
hepatic stellate cell
histone deacetylase inhibitor
epigenetics
givinostat
Gossypol, a novel modulator of VCP, induces autophagic degradation of mutant huntingtin by promoting the formation of VCP/p97-LC3-mHTT complex
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 卷号: 42, 期号: 10, 页码: 1556-1566
作者:
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/03/21
Huntington disease
mutant huntingtin protein
gossypol acetate
VCP
LC3
autophagic degradation
drug reposition
Targeting Protein Neddylation to Inactivate Cullin-RING Ligases by Gossypol: A Lucky Hit or a New Start?
期刊论文
OAI收割
DRUG DESIGN DEVELOPMENT AND THERAPY, 2021, 卷号: 15
作者:
Yu, Qing
;
Sun, Yi
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2021/03/15
anti-cancer drug
cullin-RING E3 ligases
natural product
high-throughput screen
neddylation
small-molecule inhibitors
Lipid production is more than doubled by manipulating a diacylglycerol acyltransferase in algae
期刊论文
OAI收割
GLOBAL CHANGE BIOLOGY BIOENERGY, 2020, 页码: 16
作者:
Zhang, Yu
;
Pan, Yufang
;
Ding, Wei
;
Hu, Hanhua
;
Liu, Jin
  |  
收藏
  |  
浏览/下载:98/0
  |  
提交时间:2020/12/31
biofuel
diacylglycerol acyltransferase
genetic manipulation
oleaginous alga
Phaeodactylum tricornutum
subcellular localization
triacylglycerol