中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [474]
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Discovery of betulinic acid derivatives as gut-restricted TGR5 agonists: Balancing the potency and physicochemical properties 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 144, 页码: 18
作者:  
Zhuo, Ning;  Yun, Ying;  Zhang, Chenlu;  Guo, Shimeng;  Yin, Jianpeng
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/03/25
Eleven highly oxygenated and anti-inflammatory guaian-8,12-olides from Hedyosmum orientale 期刊论文  OAI收割
TETRAHEDRON, 2024, 卷号: 152, 页码: 8
作者:  
Fan, Yao-Yue;  Zhang, Xin-Ru;  Zheng, Cheng-Yu;  Li, Ying;  Yue, Jian-Min
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/03/25
Novel imidazo[1,2,4] triazole derivatives: Synthesis, fluorescence, bioactivity for SHP1 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 15
作者:  
Yan, Xue;  Zhang, Chun;  Gao, Li-Xin;  Liu, Min -Min;  Yang, Yu-Ting
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/02/27
Metabolic regulation of homologous recombination repair by MRE11 lactylation 期刊论文  OAI收割
CELL, 2024, 卷号: 187, 期号: 2, 页码: 40
作者:  
Chen, Yuping;  Wu, Jinhuan;  Zhai, Linhui;  Zhang, Tingting;  Yin, Hui
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/04/09
Discovery and exploration of novel somatostatin receptor subtype 5 (SSTR5) antagonists for the treatment of cholesterol gallstones 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 264, 页码: 16
作者:  
Han, Fanghui;  Zhao, Tingting;  Zhang, Yanglong;  Yun, Ying;  Xu, Yuanyuan
  |  收藏  |  浏览/下载:3/0  |  提交时间:2024/02/19
A novel capsid-XL32-derived adeno-associated virus serotype prompts retinal tropism and ameliorates choroidal neovascularization 期刊论文  OAI收割
BIOMATERIALS, 2024, 卷号: 304, 页码: 13
作者:  
Luo, Lin-Lin;  Xu, Jie;  Wang, Bing-Qiao;  Chen, Chen;  Chen, Xi
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/01/26
Discovery of a novel GPR35 agonist with high and equipotent species potency for oral treatment of IBD 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 96, 页码: 12
作者:  
Song, Zhaoxiang;  Lu, Dan;  Sun, Jun;  Ye, Yangliang;  Fang, Jiahui
  |  收藏  |  浏览/下载:26/0  |  提交时间:2024/01/16
GPR35  IBD  Lodoxamide  
Exploring the mechanism of the PTP1B inhibitors by molecular dynamics and experimental study 期刊论文  OAI收割
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2023, 卷号: 125, 页码: 12
作者:  
Zhao, Tian-Tian;  Hu, Hao-Jie;  Gao, Li-Xin;  Zhou, Yu-Bo;  Zhu, Yun-Long
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/10/17
A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects 期刊论文  OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:  
Yang, Xin-Mei;  Yang, Yang;  Yao, Bu-Fan;  Ye, Pan-Pan;  Xu, Yan
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/12/11
CD47 and PD-L1 overexpression in proliferating human hepatocytes attenuated immune responses and ameliorated acute liver injury in mice 期刊论文  OAI收割
AMERICAN JOURNAL OF TRANSPLANTATION, 2023, 卷号: 23, 期号: 12, 页码: 1832-1844
作者:  
Ma, Chen;  Cao, Huiying;  Sun, Zhen;  Deng, Qiangqiang;  Liu, Wenjing
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/02/27