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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [14]
采集方式
OAI收割 [14]
内容类型
期刊论文 [14]
发表日期
2024 [1]
2022 [1]
2021 [4]
2018 [2]
2017 [1]
2014 [2]
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浏览/检索结果:
共14条,第1-10条
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存缴方式:oaiharvest
专题:上海药物研究所
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Discovery of betulinic acid derivatives as gut-restricted TGR5 agonists: Balancing the potency and physicochemical properties
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 144, 页码: 18
作者:
Zhuo, Ning
;
Yun, Ying
;
Zhang, Chenlu
;
Guo, Shimeng
;
Yin, Jianpeng
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/03/25
Type 2 Diabetes
TGR5 agonist
Betulinic acid
Gut-restricted
Gallbladder-filling effects
Kinetophores
Copy Number Analyses Identified a Novel Gene: APOBEC3A Related to Lipid Metabolism in the Pathogenesis of Preeclampsia
期刊论文
OAI收割
FRONTIERS IN CARDIOVASCULAR MEDICINE, 2022, 卷号: 9, 页码: 13
作者:
Liu, Nan
;
Guo, Yu-Na
;
Wang, Xiao-Jin
;
Ma, Jue
;
He, Yun-Ting
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/08/16
preeclampsia
APOBEC3A
lipid metabolism
copy number variation
genetics
Identification of Betulinic Acid Derivatives as Potent TGR5 Agonists with Antidiabetic Effects via Humanized TGR5(H88Y) Mutant Mice
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12181-12199
作者:
Yun, Ying
;
Zhang, Chenlu
;
Guo, Shimeng
;
Liang, Xiaoying
;
Lan, Yuan
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2021/11/04
Iridoid Constituents of Viburnum brachybotryum
期刊论文
OAI收割
JOURNAL OF NATURAL PRODUCTS, 2021, 卷号: 84, 期号: 7, 页码: 1915-1923
作者:
Rao, Li
;
Li, Yao
;
He, Qian
;
Liu, Yu
;
Su, Yu
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/11/04
Acylphloroglucinol derivatives with ATP citrate lyase inhibitory activities from Syzygium oblatum Wall
期刊论文
OAI收割
PHYTOCHEMISTRY, 2021, 卷号: 187, 页码: 7
作者:
Huang, Jin-Chang
;
Liu, Yi-Nan
;
Tao, Yun-Hua
;
Chen, Bai-Yu
;
Lei, Chun
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2021/08/17
Syzygium oblatum Wall
Myrtaceae
Acylphloroglucinols
Oblatones A-I
ATP citrate lyase
Discovery of HN37 as a Potent and Chemically Stable Antiepileptic Drug Candidate
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 9, 页码: 5816-5837
作者:
Zhang, Yang-Ming
;
Xu, Hai-Yan
;
Hu, Hai-Ning
;
Tian, Fu-Yun
;
Chen, Fei
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/03/21
Identification of compound D2923 as a novel anti-tumor agent targeting CSF1R
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 11, 页码: 1768-1776
作者:
Liu, Ying-Qiang
;
Wang, Ya-Nan
;
Lu, Xiao-Yun
;
Tong, Lin-Jiang
;
Li, Yan
  |  
收藏
  |  
浏览/下载:110/0
  |  
提交时间:2019/01/08
CSF-1R
small-molecule inhibitor
macrophage
myeloid leukemia
Discovery of novel propargylamine-modified 4-aminoalkyl imidazole substituted pyrimidinylthiourea derivatives as multifunctional agents for the treatment of Alzheimer's disease
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 143, 页码: 33-47
作者:
Xu, Yi-xiang
;
Wang, Huan
;
Li, Xiao-kang
;
Dong, Sheng-nan
;
Liu, Wen-wen
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
Multifunctional agents
AChE inhibitors
MAO-B inhibitors
Metal chelating agents
Alzheimer's disease
The synthesis and antistaphylococcal activity of 9, 13-disubstituted berberine derivatives
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 127, 页码: 424-433
作者:
Wang, Jing
;
Yang, Teng
;
Chen, Huang
;
Xu, Yun-Nan
;
Yu, Li-Fang
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
Berberine derivatives
Antistaphylococcal activity
Multidrug-resistant
Cytotoxicity
Azoxystrobin, a mitochondrial complex III Q(o) site inhibitor, exerts beneficial metabolic effects in vivo and in vitro
期刊论文
OAI收割
BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS, 2014, 卷号: 1840, 期号: 7, 页码: 2212-2221
作者:
Gao, An-Hui
;
Fu, Yan-Yun
;
Zhang, Kun-Zhi
;
Zhang, Mei
;
Jiang, Hao-Wen
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
Azoxystrobin
Mitochondria complex III
Metabolic diseases
AMP-activated protein kinase